Compile Data Set for Download or QSAR
Found 139 with Last Name = 'puri' and Initial = 's'
TargetMonocarboxylate transporter 1(Rattus norvegicus (Rat))TBA
LigandPNGBDBM50606662(CHEMBL5221129)copy SMILES
Ligand InfoPC cidPC sid
In DepthDetails
TargetMonocarboxylate transporter 2(Rattus norvegicus)TBA
LigandPNGBDBM50606662(CHEMBL5221129)copy SMILES
Ligand InfoPC cidPC sid
In DepthDetails
TargetMonocarboxylate transporter 2(Homo sapiens)TBA
LigandPNGBDBM50103571(CHEMBL3335793)copy SMILES
Affinity DataKi:  20nMMore data for this Ligand-Target Pair
In DepthDetails
TargetMonocarboxylate transporter 4(Homo sapiens (Human))TBA
LigandPNGBDBM50608641(AF 2838 | AF-2838 | BINDARIT | Bindarit)copy SMILES
Affinity DataKi:  3.02E+4nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
TargetMonocarboxylate transporter 4(Homo sapiens (Human))TBA
LigandPNGBDBM356917(US10214492, Example 268 | US11292767, Example 268)copy SMILEScopy InChI
Affinity DataIC50: 0.300nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
TargetMonocarboxylate transporter 4(Homo sapiens (Human))TBA
LigandPNGBDBM356915(US10214492, Example 266 | US11292767, Example 266)copy SMILEScopy InChI
Affinity DataIC50: 0.360nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
TargetMonocarboxylate transporter 4(Homo sapiens (Human))TBA
LigandPNGBDBM356916(US10214492, Example 267 | US11292767, Example 267)copy SMILEScopy InChI
Affinity DataIC50: 0.570nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
TargetMonocarboxylate transporter 1(Homo sapiens (Human))TBA
LigandPNGBDBM50092069(CHEMBL3582422 | US9296728, 20)copy SMILEScopy InChI
In DepthDetails
TargetTransient receptor potential cation channel subfamily M member 8(Homo sapiens (Human))
Glenmark Pharmaceuticals Ltd.

Curated by ChEMBL
LigandPNGBDBM50442406(CHEMBL2443061)copy SMILEScopy InChI
Affinity DataIC50: 8.90nMAssay Description:Antagonist activity at human TRPM8 expressed in CHO cells assessed as inhibition of icilin-induced 45Ca2+ uptake incubated for 10 mins prior to icili...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TH8P5SPubMed
TargetMonocarboxylate transporter 1(Homo sapiens (Human))TBA
LigandPNGBDBM50092072(CHEMBL3582419 | US9296728, 14)copy SMILEScopy InChI
In DepthDetails
TargetTransient receptor potential cation channel subfamily M member 8(Homo sapiens (Human))
Glenmark Pharmaceuticals Ltd.

Curated by ChEMBL
LigandPNGBDBM50442408(CHEMBL2443079)copy SMILEScopy InChI
Affinity DataIC50: 9.5nMAssay Description:Antagonist activity at human TRPM8 expressed in CHO cells assessed as inhibition of icilin-induced 45Ca2+ uptake incubated for 10 mins prior to icili...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TH8P5SPubMed
TargetMonocarboxylate transporter 1(Homo sapiens (Human))TBA
LigandPNGBDBM50092071(CHEMBL3582420 | US9296728, 18)copy SMILEScopy InChI
Affinity DataIC50: 11nMMore data for this Ligand-Target Pair
In DepthDetails
TargetMonocarboxylate transporter 1(Rattus norvegicus (Rat))TBA
LigandPNGBDBM50608638(CHEMBL4303684)copy SMILES
Affinity DataIC50: 13nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails
TargetTransient receptor potential cation channel subfamily M member 8(Homo sapiens (Human))
Glenmark Pharmaceuticals Ltd.

Curated by ChEMBL
LigandPNGBDBM50442406(CHEMBL2443061)copy SMILEScopy InChI
Affinity DataIC50: 13nMAssay Description:Antagonist activity at human TRPM8 expressed in CHO cells assessed as inhibition of icilin-induced 45Ca2+ uptake incubated for 10 mins prior to icili...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TH8P5SPubMed
TargetMonocarboxylate transporter 4(Homo sapiens (Human))TBA
LigandPNGBDBM50092072(CHEMBL3582419 | US9296728, 14)copy SMILEScopy InChI
Affinity DataIC50: 14nMMore data for this Ligand-Target Pair
In DepthDetails
TargetTransient receptor potential cation channel subfamily M member 8(Homo sapiens (Human))
Glenmark Pharmaceuticals Ltd.

Curated by ChEMBL
LigandPNGBDBM50442404(CHEMBL2443063)copy SMILEScopy InChI
Affinity DataIC50: 17nMAssay Description:Antagonist activity at human TRPM8 expressed in CHO cells assessed as inhibition of icilin-induced 45Ca2+ uptake incubated for 10 mins prior to icili...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TH8P5SPubMed
TargetTransient receptor potential cation channel subfamily M member 8(Rattus norvegicus (Rat))
Glenmark Pharmaceuticals Ltd.

Curated by ChEMBL
LigandPNGBDBM50442406(CHEMBL2443061)copy SMILEScopy InChI
Affinity DataIC50: 17nMAssay Description:Antagonist activity at rat TRPM8 by 45Ca2+ uptake assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TH8P5SPubMed
TargetMonocarboxylate transporter 4(Homo sapiens (Human))TBA
LigandPNGBDBM50092071(CHEMBL3582420 | US9296728, 18)copy SMILEScopy InChI
Affinity DataIC50: 17nMMore data for this Ligand-Target Pair
In DepthDetails
TargetTransient receptor potential cation channel subfamily M member 8(Homo sapiens (Human))
Glenmark Pharmaceuticals Ltd.

Curated by ChEMBL
LigandPNGBDBM50442426(CHEMBL2443085)copy SMILEScopy InChI
Affinity DataIC50: 19nMAssay Description:Antagonist activity at human TRPM8 expressed in CHO cells assessed as inhibition of icilin-induced 45Ca2+ uptake incubated for 10 mins prior to icili...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TH8P5SPubMed
TargetTransient receptor potential cation channel subfamily M member 8(Homo sapiens (Human))
Glenmark Pharmaceuticals Ltd.

Curated by ChEMBL
LigandPNGBDBM50442405(CHEMBL2443062)copy SMILEScopy InChI
Affinity DataIC50: 20nMAssay Description:Antagonist activity at human TRPM8 expressed in CHO cells assessed as inhibition of icilin-induced 45Ca2+ uptake incubated for 10 mins prior to icili...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TH8P5SPubMed
TargetMonocarboxylate transporter 4(Homo sapiens (Human))TBA
LigandPNGBDBM50092069(CHEMBL3582422 | US9296728, 20)copy SMILEScopy InChI
Affinity DataIC50: 23nMMore data for this Ligand-Target Pair
In DepthDetails
TargetTransient receptor potential cation channel subfamily M member 8(Homo sapiens (Human))
Glenmark Pharmaceuticals Ltd.

Curated by ChEMBL
LigandPNGBDBM50442408(CHEMBL2443079)copy SMILEScopy InChI
Affinity DataIC50: 23nMAssay Description:Antagonist activity at human TRPM8 expressed in CHO cells assessed as inhibition of icilin-induced 45Ca2+ uptake incubated for 10 mins prior to icili...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TH8P5SPubMed
TargetMonocarboxylate transporter 1(Homo sapiens (Human))TBA
LigandPNGBDBM50608633(CHEMBL3582501)copy SMILES
Affinity DataIC50: 25nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
TargetMonocarboxylate transporter 4(Homo sapiens (Human))TBA
LigandPNGBDBM214697(US9296728, 19)copy SMILEScopy InChI
Affinity DataIC50: 32nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
TargetMonocarboxylate transporter 1(Homo sapiens (Human))TBA
LigandPNGBDBM50092070(CHEMBL3582421 | US9296728, 15)copy SMILEScopy InChI
Affinity DataIC50: 34nMMore data for this Ligand-Target Pair
In DepthDetails
TargetTransient receptor potential cation channel subfamily V member 1(Homo sapiens (Human))
Glenmark Pharmaceuticals Ltd.

Curated by ChEMBL
LigandPNGBDBM50133817(4-(3-Chloro-pyridin-2-yl)-piperazine-1-carboxylic ...)copy SMILEScopy InChI
Affinity DataIC50: 35nMAssay Description:Inhibition of TRPV1 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TH8P5SPubMed
TargetMonocarboxylate transporter 1(Homo sapiens (Human))TBA
LigandPNGBDBM214697(US9296728, 19)copy SMILEScopy InChI
Affinity DataIC50: 37nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
TargetTransient receptor potential cation channel subfamily M member 8(Homo sapiens (Human))
Glenmark Pharmaceuticals Ltd.

Curated by ChEMBL
LigandPNGBDBM50442425(CHEMBL2443086)copy SMILEScopy InChI
Affinity DataIC50: 41nMAssay Description:Antagonist activity at human TRPM8 expressed in CHO cells assessed as inhibition of icilin-induced 45Ca2+ uptake incubated for 10 mins prior to icili...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TH8P5SPubMed
TargetTransient receptor potential cation channel subfamily M member 8(Homo sapiens (Human))
Glenmark Pharmaceuticals Ltd.

Curated by ChEMBL
LigandPNGBDBM50442410(CHEMBL2443074)copy SMILEScopy InChI
Affinity DataIC50: 45nMAssay Description:Antagonist activity at human TRPM8 expressed in CHO cells assessed as inhibition of icilin-induced 45Ca2+ uptake incubated for 10 mins prior to icili...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TH8P5SPubMed
TargetTransient receptor potential cation channel subfamily M member 8(Homo sapiens (Human))
Glenmark Pharmaceuticals Ltd.

Curated by ChEMBL
LigandPNGBDBM50442407(CHEMBL2443060)copy SMILEScopy InChI
Affinity DataIC50: 46nMAssay Description:Antagonist activity at human TRPM8 expressed in CHO cells assessed as inhibition of icilin-induced 45Ca2+ uptake incubated for 10 mins prior to icili...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TH8P5SPubMed
TargetMonocarboxylate transporter 1(Homo sapiens (Human))TBA
LigandPNGBDBM214698(US9296728, 21)copy SMILEScopy InChI
Affinity DataIC50: 48nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
TargetTransient receptor potential cation channel subfamily M member 8(Homo sapiens (Human))
Glenmark Pharmaceuticals Ltd.

Curated by ChEMBL
LigandPNGBDBM50442427(CHEMBL2443084)copy SMILEScopy InChI
Affinity DataIC50: 49nMAssay Description:Antagonist activity at human TRPM8 expressed in CHO cells assessed as inhibition of icilin-induced 45Ca2+ uptake incubated for 10 mins prior to icili...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TH8P5SPubMed
TargetMonocarboxylate transporter 4(Homo sapiens (Human))TBA
LigandPNGBDBM214698(US9296728, 21)copy SMILEScopy InChI
Affinity DataIC50: 53nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
TargetMonocarboxylate transporter 4(Homo sapiens (Human))TBA
LigandPNGBDBM50608633(CHEMBL3582501)copy SMILES
Affinity DataIC50: 58nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
TargetTransient receptor potential cation channel subfamily M member 8(Homo sapiens (Human))
Glenmark Pharmaceuticals Ltd.

Curated by ChEMBL
LigandPNGBDBM50442405(CHEMBL2443062)copy SMILEScopy InChI
Affinity DataIC50: 60nMAssay Description:Antagonist activity at human TRPM8 expressed in CHO cells assessed as inhibition of icilin-induced 45Ca2+ uptake incubated for 10 mins prior to icili...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TH8P5SPubMed
TargetMonocarboxylate transporter 1(Rattus norvegicus (Rat))TBA
LigandPNGBDBM50608639(CHEMBL4793546)copy SMILES
Affinity DataIC50: 66nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
TargetTransient receptor potential cation channel subfamily M member 8(Homo sapiens (Human))
Glenmark Pharmaceuticals Ltd.

Curated by ChEMBL
LigandPNGBDBM50442411(CHEMBL2443073)copy SMILEScopy InChI
Affinity DataIC50: 66nMAssay Description:Antagonist activity at human TRPM8 expressed in CHO cells assessed as inhibition of icilin-induced 45Ca2+ uptake incubated for 10 mins prior to icili...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TH8P5SPubMed
TargetDisintegrin and metalloproteinase domain-containing protein 17(Homo sapiens (Human))
Sun Pharma Advanced Research Company Ltd

Curated by ChEMBL
LigandPNGBDBM50355462(CHEMBL1835559)copy SMILEScopy InChI
Affinity DataIC50: 70nMAssay Description:Inhibition of TACE in human whole blood assessed as reduction of of LPS-induced TNFalpha production pretreated 15 mins before LPS challenge measured ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JQ11FFPubMed
TargetDisintegrin and metalloproteinase domain-containing protein 17(Homo sapiens (Human))
Sun Pharma Advanced Research Company Ltd

Curated by ChEMBL
LigandPNGBDBM50355463(CHEMBL1835560)copy SMILEScopy InChI
Affinity DataIC50: 74nMAssay Description:Inhibition of TACE in human whole blood assessed as reduction of of LPS-induced TNFalpha production pretreated 15 mins before LPS challenge measured ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JQ11FFPubMed
TargetDisintegrin and metalloproteinase domain-containing protein 17(Homo sapiens (Human))
Sun Pharma Advanced Research Company Ltd

Curated by ChEMBL
LigandPNGBDBM50355458(CHEMBL1835555)copy SMILEScopy InChI
Affinity DataIC50: 80nMAssay Description:Inhibition of TACE in human whole blood assessed as reduction of of LPS-induced TNFalpha production pretreated 15 mins before LPS challenge measured ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JQ11FFPubMed
TargetMonocarboxylate transporter 4(Homo sapiens (Human))TBA
LigandPNGBDBM50092070(CHEMBL3582421 | US9296728, 15)copy SMILEScopy InChI
Affinity DataIC50: 85nMMore data for this Ligand-Target Pair
In DepthDetails
TargetTransient receptor potential cation channel subfamily M member 8(Homo sapiens (Human))
Glenmark Pharmaceuticals Ltd.

Curated by ChEMBL
LigandPNGBDBM50442412(CHEMBL2443072)copy SMILEScopy InChI
Affinity DataIC50: 90nMAssay Description:Antagonist activity at human TRPM8 expressed in CHO cells assessed as inhibition of icilin-induced 45Ca2+ uptake incubated for 10 mins prior to icili...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TH8P5SPubMed
TargetTransient receptor potential cation channel subfamily M member 8(Homo sapiens (Human))
Glenmark Pharmaceuticals Ltd.

Curated by ChEMBL
LigandPNGBDBM50442409(CHEMBL2443078)copy SMILEScopy InChI
Affinity DataIC50: 94nMAssay Description:Antagonist activity at human TRPM8 expressed in CHO cells assessed as inhibition of icilin-induced 45Ca2+ uptake incubated for 10 mins prior to icili...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TH8P5SPubMed
TargetTransient receptor potential cation channel subfamily M member 8(Homo sapiens (Human))
Glenmark Pharmaceuticals Ltd.

Curated by ChEMBL
LigandPNGBDBM50442428(CHEMBL2443083)copy SMILEScopy InChI
Affinity DataIC50: 97nMAssay Description:Antagonist activity at human TRPM8 expressed in CHO cells assessed as inhibition of icilin-induced 45Ca2+ uptake incubated for 10 mins prior to icili...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TH8P5SPubMed
TargetMonocarboxylate transporter 1(Rattus norvegicus (Rat))TBA
LigandPNGBDBM50608637(CHEMBL5280660)copy SMILES
Affinity DataIC50: 97nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
TargetTransient receptor potential cation channel subfamily M member 8(Homo sapiens (Human))
Glenmark Pharmaceuticals Ltd.

Curated by ChEMBL
LigandPNGBDBM50442413(CHEMBL2443071)copy SMILEScopy InChI
Affinity DataIC50: 107nMAssay Description:Antagonist activity at human TRPM8 expressed in CHO cells assessed as inhibition of icilin-induced 45Ca2+ uptake incubated for 10 mins prior to icili...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TH8P5SPubMed
TargetTransient receptor potential cation channel subfamily M member 8(Homo sapiens (Human))
Glenmark Pharmaceuticals Ltd.

Curated by ChEMBL
LigandPNGBDBM50442414(CHEMBL2443070)copy SMILEScopy InChI
Affinity DataIC50: 111nMAssay Description:Antagonist activity at human TRPM8 expressed in CHO cells assessed as inhibition of icilin-induced 45Ca2+ uptake incubated for 10 mins prior to icili...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TH8P5SPubMed
TargetTransient receptor potential cation channel subfamily M member 8(Homo sapiens (Human))
Glenmark Pharmaceuticals Ltd.

Curated by ChEMBL
LigandPNGBDBM50442419(CHEMBL2443066)copy SMILEScopy InChI
Affinity DataIC50: 113nMAssay Description:Antagonist activity at human TRPM8 expressed in CHO cells assessed as inhibition of icilin-induced 45Ca2+ uptake incubated for 10 mins prior to icili...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TH8P5SPubMed
TargetDisintegrin and metalloproteinase domain-containing protein 17(Homo sapiens (Human))
Sun Pharma Advanced Research Company Ltd

Curated by ChEMBL
LigandPNGBDBM50355460(CHEMBL1835557)copy SMILEScopy InChI
Affinity DataIC50: 126nMAssay Description:Inhibition of TACE in human whole blood assessed as reduction of of LPS-induced TNFalpha production pretreated 15 mins before LPS challenge measured ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JQ11FFPubMed
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