Compile Data Set for Download or QSAR
Found 303 with Last Name = 'sievers' and Initial = 's'
TargetCasein kinase I isoform delta(Homo sapiens (Human))TBA
LigandPNGBDBM50105742(4-[4-(4-Fluoro-phenyl)-5-(2-methoxy-pyrimidin-4-yl...)copy SMILEScopy InChI
Affinity DataKi:  25nMMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2P84GZFPubMed
TargetCasein kinase I isoform delta(Homo sapiens (Human))TBA
LigandPNGBDBM50284506(4-[5-(4-Fluoro-phenyl)-2-(4-methanesulfonyl-phenyl...)copy SMILEScopy InChI
Affinity DataKi:  39nMMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2P84GZFPubMed
TargetNAD-dependent protein deacetylase sirtuin-1(Homo sapiens (Human))TBA
LigandPNGBDBM50178769((+/-)-6-chloro-2,3,4,9-tetrahydro-1H-carbazole-1-c...)copy SMILEScopy InChI
Affinity DataKi:  114nMAssay Description:Uncompetitive inhibition of His6-tagged SIRT1 (unknown origin) expressed in Escherichia coli BL21 (DE3) assessed as inhibition constant measured ever...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MK6HQZPubMed
TargetNAD-dependent protein deacetylase sirtuin-1(Homo sapiens (Human))TBA
LigandPNGBDBM50576050(CHEMBL4858009)copy SMILES
Affinity DataKi:  285nMAssay Description:Uncompetitive inhibition of His6-tagged SIRT1 (unknown origin) expressed in Escherichia coli BL21 (DE3) assessed as inhibition constant measured ever...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MK6HQZPubMed
TargetNAD-dependent protein deacetylase sirtuin-1(Homo sapiens (Human))TBA
LigandPNGBDBM50576055(CHEMBL4855963)copy SMILES
Affinity DataKi:  400nMAssay Description:Uncompetitive inhibition of His6-tagged SIRT1 (unknown origin) expressed in Escherichia coli BL21 (DE3) assessed as inhibition constant measured ever...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MK6HQZPubMed
TargetCasein kinase I isoform alpha(Homo sapiens (Human))TBA
LigandPNGBDBM50105742(4-[4-(4-Fluoro-phenyl)-5-(2-methoxy-pyrimidin-4-yl...)copy SMILEScopy InChI
Affinity DataKi:  501nMMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2P84GZFPubMed
TargetCasein kinase I isoform alpha(Homo sapiens (Human))TBA
LigandPNGBDBM50284506(4-[5-(4-Fluoro-phenyl)-2-(4-methanesulfonyl-phenyl...)copy SMILEScopy InChI
Affinity DataKi:  650nMMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2P84GZFPubMed
LigandPNGBDBM50547124(CHEMBL242708 | NCI-0001009)copy SMILES
Affinity DataKi:  2.60E+3nMAssay Description:Reversible inhibition of CPM binding to nonacylated N-terminal His6-tagged human TEAD4 (217 to 434 residues) expressed in Escherichia coli BL21-Codon...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QN6BC1PubMed
LigandPNGBDBM50547126(CHEMBL4763473)copy SMILES
Affinity DataKi:  1.04E+4nMAssay Description:Inhibition of CPM binding to N-terminal His6-tagged human TEAD4 (217 to 434 residues) expressed in Escherichia coli BL21-CodonPlus (DE3)-RIPL cells p...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QN6BC1PubMed
TargetActivin receptor type-1(Homo sapiens (Human))TBA
LigandPNGBDBM50261979(5-(6-(4-methoxyphenyl)pyrazolo[1,5-a]pyrimidin-3-y...)copy SMILEScopy InChI
Affinity DataIC50: 32nMMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q20C50VHPubMed
TargetMitogen-activated protein kinase 11(Homo sapiens (Human))TBA
LigandPNGBDBM50284506(4-[5-(4-Fluoro-phenyl)-2-(4-methanesulfonyl-phenyl...)copy SMILEScopy InChI
Affinity DataIC50: 40nMMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2P84GZFPubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))TBA
LigandPNGBDBM50284506(4-[5-(4-Fluoro-phenyl)-2-(4-methanesulfonyl-phenyl...)copy SMILEScopy InChI
Affinity DataIC50: 40nMMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2P84GZFPubMed
TargetMitogen-activated protein kinase 11(Homo sapiens (Human))TBA
LigandPNGBDBM50105742(4-[4-(4-Fluoro-phenyl)-5-(2-methoxy-pyrimidin-4-yl...)copy SMILEScopy InChI
Affinity DataIC50: 44nMMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2P84GZFPubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))TBA
LigandPNGBDBM50105742(4-[4-(4-Fluoro-phenyl)-5-(2-methoxy-pyrimidin-4-yl...)copy SMILEScopy InChI
Affinity DataIC50: 44nMMore data for this Ligand-Target Pair
TargetNAD-dependent protein deacetylase sirtuin-1(Homo sapiens (Human))TBA
LigandPNGBDBM50178769((+/-)-6-chloro-2,3,4,9-tetrahydro-1H-carbazole-1-c...)copy SMILEScopy InChI
Affinity DataIC50: 48nMAssay Description:Inhibition of His6-tagged SIRT1 (unknown origin) expressed in Escherichia coli BL21 (DE3) preincubated for 15 mins followed by NAD+ addition and meas...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MK6HQZPubMed
LigandPNGBDBM50547124(CHEMBL242708 | NCI-0001009)copy SMILES
Affinity DataIC50: 70nMAssay Description:Binding affinity to nonacylated N-terminal His6-tagged human TEAD4 (217 to 434 residues) expressed in Escherichia coli BL21-CodonPlus (DE3)-RIPL cell...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QN6BC1PubMed
LigandPNGBDBM50547134(CHEMBL4787565)copy SMILES
Affinity DataIC50: 100nMAssay Description:Inhibition of FITC-labeled palmitate tracer binding to N-terminal His6-tagged human TEAD4 (217 to 434 residues) expressed in Escherichia coli BL21-Co...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QN6BC1PubMed
TargetCasein kinase I isoform delta(Homo sapiens (Human))TBA
LigandPNGBDBM50588635(CHEMBL5186013)copy SMILES
Affinity DataIC50: 120nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FX7FFTPubMed
TargetDNA-dependent protein kinase catalytic subunit(Homo sapiens (Human))TBA
LigandPNGBDBM50004566(9-Chloro-2-furan-2-yl-[1,2,4]triazolo[1,5-c]quinaz...)copy SMILEScopy InChI
Affinity DataIC50: 140nMMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FX7FFTPubMed
TargetNAD-dependent protein deacetylase sirtuin-1(Homo sapiens (Human))TBA
LigandPNGBDBM50576050(CHEMBL4858009)copy SMILES
Affinity DataIC50: 150nMAssay Description:Inhibition of His6-tagged SIRT1 (unknown origin) expressed in Escherichia coli BL21 (DE3) preincubated for 15 mins followed by NAD+ addition and meas...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MK6HQZPubMed
LigandPNGBDBM50547124(CHEMBL242708 | NCI-0001009)copy SMILES
Affinity DataIC50: 200nMAssay Description:Inhibition of FITC-labeled palmitate tracer binding to N-terminal His6-tagged human TEAD4 (217 to 434 residues) expressed in Escherichia coli BL21-Co...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QN6BC1PubMed
LigandPNGBDBM50547135(CHEMBL4776143)copy SMILES
Affinity DataIC50: 200nMAssay Description:Inhibition of FITC-labeled palmitate tracer binding to N-terminal His6-tagged human TEAD4 (217 to 434 residues) expressed in Escherichia coli BL21-Co...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QN6BC1PubMed
LigandPNGBDBM50547136(CHEMBL4757924)copy SMILES
Affinity DataIC50: 200nMAssay Description:Inhibition of FITC-labeled palmitate tracer binding to N-terminal His6-tagged human TEAD4 (217 to 434 residues) expressed in Escherichia coli BL21-Co...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QN6BC1PubMed
LigandPNGBDBM50547146(CHEMBL4745853)copy SMILES
Affinity DataIC50: 200nMAssay Description:Inhibition of FITC-labeled palmitate tracer binding to N-terminal His6-tagged human TEAD4 (217 to 434 residues) expressed in Escherichia coli BL21-Co...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QN6BC1PubMed
LigandPNGBDBM50547142(CHEMBL4757369)copy SMILES
Affinity DataIC50: 200nMAssay Description:Inhibition of FITC-labeled palmitate tracer binding to N-terminal His6-tagged human TEAD4 (217 to 434 residues) expressed in Escherichia coli BL21-Co...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QN6BC1PubMed
LigandPNGBDBM50547154(CHEMBL4745831)copy SMILES
Affinity DataIC50: 200nMAssay Description:Inhibition of FITC-labeled palmitate tracer binding to N-terminal His6-tagged human TEAD4 (217 to 434 residues) expressed in Escherichia coli BL21-Co...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QN6BC1PubMed
TargetCasein kinase I isoform alpha(Homo sapiens (Human))TBA
LigandPNGBDBM50588635(CHEMBL5186013)copy SMILES
Affinity DataIC50: 220nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FX7FFTPubMed
TargetNAD-dependent protein deacetylase sirtuin-1(Homo sapiens (Human))TBA
LigandPNGBDBM50576055(CHEMBL4855963)copy SMILES
Affinity DataIC50: 220nMAssay Description:Inhibition of His6-tagged SIRT1 (unknown origin) expressed in Escherichia coli BL21 (DE3) preincubated for 15 mins followed by NAD+ addition and meas...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MK6HQZPubMed
TargetNAD-dependent protein deacetylase sirtuin-1(Homo sapiens (Human))TBA
LigandPNGBDBM50576055(CHEMBL4855963)copy SMILES
Affinity DataIC50: 220nMAssay Description:Inhibition of His6-tagged SIRT1 (unknown origin) expressed in Escherichia coli BL21 (DE3) preincubated for 15 mins followed by NAD+ addition and meas...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MK6HQZPubMed
TargetNAD-dependent protein deacetylase sirtuin-1(Homo sapiens (Human))TBA
LigandPNGBDBM50576049(CHEMBL4876032)copy SMILES
Affinity DataIC50: 230nMAssay Description:Inhibition of His6-tagged SIRT1 (unknown origin) expressed in Escherichia coli BL21 (DE3) preincubated for 15 mins followed by NAD+ addition and meas...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MK6HQZPubMed
TargetCasein kinase I isoform delta(Homo sapiens (Human))TBA
LigandPNGBDBM50004566(9-Chloro-2-furan-2-yl-[1,2,4]triazolo[1,5-c]quinaz...)copy SMILEScopy InChI
Affinity DataIC50: 240nMMore data for this Ligand-Target Pair
LigandPNGBDBM50547143(CHEMBL4789889)copy SMILES
Affinity DataIC50: 300nMAssay Description:Inhibition of FITC-labeled palmitate tracer binding to N-terminal His6-tagged human TEAD4 (217 to 434 residues) expressed in Escherichia coli BL21-Co...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QN6BC1PubMed
LigandPNGBDBM50547152(CHEMBL4750726)copy SMILES
Affinity DataIC50: 300nMAssay Description:Inhibition of FITC-labeled palmitate tracer binding to N-terminal His6-tagged human TEAD4 (217 to 434 residues) expressed in Escherichia coli BL21-Co...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QN6BC1PubMed
LigandPNGBDBM50547148(CHEMBL4797833)copy SMILES
Affinity DataIC50: 300nMAssay Description:Inhibition of FITC-labeled palmitate tracer binding to N-terminal His6-tagged human TEAD4 (217 to 434 residues) expressed in Escherichia coli BL21-Co...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QN6BC1PubMed
LigandPNGBDBM50547155(CHEMBL4744235)copy SMILES
Affinity DataIC50: 300nMAssay Description:Inhibition of FITC-labeled palmitate tracer binding to N-terminal His6-tagged human TEAD4 (217 to 434 residues) expressed in Escherichia coli BL21-Co...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QN6BC1PubMed
LigandPNGBDBM50547156(CHEMBL4783341)copy SMILES
Affinity DataIC50: 300nMAssay Description:Inhibition of FITC-labeled palmitate tracer binding to N-terminal His6-tagged human TEAD4 (217 to 434 residues) expressed in Escherichia coli BL21-Co...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QN6BC1PubMed
LigandPNGBDBM50547130(CHEMBL1701986)copy SMILES
Affinity DataIC50: 300nMAssay Description:Inhibition of FITC-labeled palmitate tracer binding to N-terminal His6-tagged human TEAD4 (217 to 434 residues) expressed in Escherichia coli BL21-Co...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QN6BC1PubMed
TargetCasein kinase I isoform epsilon(Homo sapiens (Human))TBA
LigandPNGBDBM50588635(CHEMBL5186013)copy SMILES
Affinity DataIC50: 380nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FX7FFTPubMed
LigandPNGBDBM50547131(CHEMBL4800702)copy SMILES
Affinity DataIC50: 400nMAssay Description:Inhibition of FITC-labeled palmitate tracer binding to N-terminal His6-tagged human TEAD4 (217 to 434 residues) expressed in Escherichia coli BL21-Co...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QN6BC1PubMed
LigandPNGBDBM50547145(CHEMBL4750624)copy SMILES
Affinity DataIC50: 400nMAssay Description:Inhibition of FITC-labeled palmitate tracer binding to N-terminal His6-tagged human TEAD4 (217 to 434 residues) expressed in Escherichia coli BL21-Co...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QN6BC1PubMed
TargetCasein kinase I isoform delta(Homo sapiens (Human))TBA
LigandPNGBDBM50588636(CHEMBL5182545)copy SMILES
Affinity DataIC50: 430nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FX7FFTPubMed
TargetNAD-dependent protein deacetylase sirtuin-1(Homo sapiens (Human))TBA
LigandPNGBDBM50576056(CHEMBL4846832)copy SMILES
Affinity DataIC50: 430nMAssay Description:Inhibition of His6-tagged SIRT1 (unknown origin) expressed in Escherichia coli BL21 (DE3) preincubated for 15 mins followed by NAD+ addition and meas...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MK6HQZPubMed
TargetNAD-dependent protein deacetylase sirtuin-1(Homo sapiens (Human))TBA
LigandPNGBDBM50576063(CHEMBL4847946)copy SMILES
Affinity DataIC50: 470nMAssay Description:Inhibition of His6-tagged SIRT1 (unknown origin) expressed in Escherichia coli BL21 (DE3) preincubated for 15 mins followed by NAD+ addition and meas...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MK6HQZPubMed
TargetNAD-dependent protein deacetylase sirtuin-1(Homo sapiens (Human))TBA
LigandPNGBDBM50576068(CHEMBL4871919)copy SMILES
Affinity DataIC50: 490nMAssay Description:Inhibition of His6-tagged SIRT1 (unknown origin) expressed in Escherichia coli BL21 (DE3) preincubated for 15 mins followed by NAD+ addition and meas...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MK6HQZPubMed
TargetCasein kinase I isoform epsilon(Homo sapiens (Human))TBA
LigandPNGBDBM50004566(9-Chloro-2-furan-2-yl-[1,2,4]triazolo[1,5-c]quinaz...)copy SMILEScopy InChI
Affinity DataIC50: 490nMMore data for this Ligand-Target Pair
TargetNAD-dependent protein deacetylase sirtuin-2(Homo sapiens (Human))TBA
LigandPNGBDBM50178769((+/-)-6-chloro-2,3,4,9-tetrahydro-1H-carbazole-1-c...)copy SMILEScopy InChI
Affinity DataIC50: 500nMAssay Description:Inhibition of His6-tagged/TEV fused SIRT2 (unknown origin) expressed in Escherichia coli BL21 (DE3) preincubated for 15 mins followed by NAD+ additio...More data for this Ligand-Target Pair
LigandPNGBDBM50547133(CHEMBL4757939)copy SMILES
Affinity DataIC50: 500nMAssay Description:Inhibition of FITC-labeled palmitate tracer binding to N-terminal His6-tagged human TEAD4 (217 to 434 residues) expressed in Escherichia coli BL21-Co...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QN6BC1PubMed
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