Compile Data Set for Download or QSAR
Found 70 with Last Name = 'gajda' and Initial = 't'
TargetArginase-2, mitochondrial(Homo sapiens (Human))TBA
LigandPNGBDBM50350311(CHEMBL1812661)copy SMILEScopy InChI
Affinity DataKi:  8.5nMAssay Description:Inhibition of human Arg2 at pH 7.5More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WS8XZCPubMed
TargetArginase-1(Homo sapiens (Human))TBA
LigandPNGBDBM50561045(CHEMBL4758805)copy SMILES
Affinity DataKi: <10nMAssay Description:Inhibition of human Arg1 using L-arginine as substrate after 60 mins by spectrophotometric analysisMore data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WS8XZCPubMed
TargetArginase-2, mitochondrial(Homo sapiens (Human))TBA
LigandPNGBDBM50561046(CHEMBL4790798)copy SMILES
Affinity DataKi: <10nMAssay Description:Inhibition of human Arg2 using L-arginine as substrate after 60 mins by spectrophotometric analysisMore data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WS8XZCPubMed
TargetArginase-2, mitochondrial(Homo sapiens (Human))TBA
LigandPNGBDBM50561045(CHEMBL4758805)copy SMILES
Affinity DataKi: <10nMAssay Description:Inhibition of human Arg2 using L-arginine as substrate after 60 mins by spectrophotometric analysisMore data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WS8XZCPubMed
TargetArginase-1(Homo sapiens (Human))TBA
LigandPNGBDBM50561046(CHEMBL4790798)copy SMILES
Affinity DataKi: <10nMAssay Description:Inhibition of human Arg1 using L-arginine as substrate after 60 mins by spectrophotometric analysisMore data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WS8XZCPubMed
TargetArginase-2, mitochondrial(Homo sapiens (Human))TBA
LigandPNGBDBM50561034(CHEMBL4244287)copy SMILES
Affinity DataKi:  30nMAssay Description:Inhibition of human Arg2 at pH 7.5More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WS8XZCPubMed
TargetArginase-2, mitochondrial(Homo sapiens (Human))TBA
LigandPNGBDBM50008099(CHEMBL1234777)copy SMILEScopy InChI
Affinity DataKi:  51nMAssay Description:Inhibition of human Arg2 at pH 7.5More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WS8XZCPubMed
TargetArginase-2, mitochondrial(Homo sapiens (Human))TBA
LigandPNGBDBM50230418(CHEMBL260629 | N(gamma)-hydroxy-L-arginine | N-OME...)copy SMILEScopy InChI
Affinity DataKi:  1.60E+3nMAssay Description:Inhibition of human Arg2 at pH 7.5More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WS8XZCPubMed
TargetArginase-2, mitochondrial(Homo sapiens (Human))TBA
LigandPNGBDBM50561047(CHEMBL4764455)copy SMILES
Affinity DataIC50: 0.100nMAssay Description:Inhibition of human Arg2More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WS8XZCPubMed
TargetArginase-1(Homo sapiens (Human))TBA
LigandPNGBDBM50561047(CHEMBL4764455)copy SMILES
Affinity DataIC50: 0.100nMAssay Description:Inhibition of human Arg1More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WS8XZCPubMed
TargetArginase-1(Homo sapiens (Human))TBA
LigandPNGBDBM50561040(CHEMBL4754637)copy SMILES
Affinity DataIC50: 0.800nMAssay Description:Inhibition of human Arg1 by TOGA assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WS8XZCPubMed
TargetArginase-1(Homo sapiens (Human))TBA
LigandPNGBDBM50561042(CHEMBL4748950)copy SMILES
Affinity DataIC50: 0.800nMAssay Description:Inhibition of human Arg1 by TOGA assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WS8XZCPubMed
TargetArginase-1(Homo sapiens (Human))TBA
LigandPNGBDBM50561049(CHEMBL4793482)copy SMILES
Affinity DataIC50: 1nMAssay Description:Inhibition of human Arg1More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WS8XZCPubMed
TargetArginase-1(Homo sapiens (Human))TBA
LigandPNGBDBM50561052(CHEMBL4755855)copy SMILES
Affinity DataIC50: 1nMAssay Description:Inhibition of human Arg1More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WS8XZCPubMed
TargetArginase-1(Homo sapiens (Human))TBA
LigandPNGBDBM50561053(CHEMBL4750602)copy SMILES
Affinity DataIC50: 1nMAssay Description:Inhibition of human Arg1More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WS8XZCPubMed
TargetArginase-1(Homo sapiens (Human))TBA
LigandPNGBDBM50561051(CHEMBL4749434)copy SMILES
Affinity DataIC50: 1nMAssay Description:Inhibition of human Arg1More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WS8XZCPubMed
TargetArginase-1(Homo sapiens (Human))TBA
LigandPNGBDBM50561041(CHEMBL4791224)copy SMILES
Affinity DataIC50: 1.60nMAssay Description:Inhibition of human Arg1 by TOGA assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WS8XZCPubMed
TargetArginase-1(Homo sapiens (Human))TBA
LigandPNGBDBM50561039(CHEMBL4749355 | US11420984, Example 23)copy SMILES
Affinity DataIC50: 3nMAssay Description:Inhibition of human Arg1 by TOGA assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WS8XZCPubMed
TargetArginase-1(Homo sapiens (Human))TBA
LigandPNGBDBM50561035(CHEMBL4763578)copy SMILES
Affinity DataIC50: 3.20nMAssay Description:Inhibition of human Arg1 by TOGA assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WS8XZCPubMed
TargetArginase-1(Homo sapiens (Human))TBA
LigandPNGBDBM50561036(CHEMBL4778978)copy SMILES
Affinity DataIC50: 6nMAssay Description:Inhibition of human Arg1 by TOGA assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WS8XZCPubMed
TargetArginase-1(Homo sapiens (Human))TBA
LigandPNGBDBM50561037(CHEMBL4762611)copy SMILES
Affinity DataIC50: 8nMAssay Description:Inhibition of human Arg1 by TOGA assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WS8XZCPubMed
TargetArginase-2, mitochondrial(Homo sapiens (Human))TBA
LigandPNGBDBM50561039(CHEMBL4749355 | US11420984, Example 23)copy SMILES
Affinity DataIC50: 10nMAssay Description:Inhibition of human Arg2 by TOGA assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WS8XZCPubMed
TargetArginase-1(Homo sapiens (Human))TBA
LigandPNGBDBM50561038(CHEMBL4752307 | US11420984, Example 7)copy SMILES
Affinity DataIC50: 10nMAssay Description:Inhibition of human Arg1 by TOGA assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WS8XZCPubMed
TargetArginase-2, mitochondrial(Homo sapiens (Human))TBA
LigandPNGBDBM50561038(CHEMBL4752307 | US11420984, Example 7)copy SMILES
Affinity DataIC50: 20nMAssay Description:Inhibition of human Arg2 by TOGA assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WS8XZCPubMed
TargetArginase-1(Homo sapiens (Human))TBA
LigandPNGBDBM50538526(CHEMBL4646697)copy SMILEScopy InChI
Affinity DataIC50: 52nMAssay Description:Inhibition of human Arg1 by TOGA assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WS8XZCPubMed
TargetArginase-1(Homo sapiens (Human))TBA
LigandPNGBDBM50511658(Cb-1158 | INCB-001158 | Incb 001158 | Incb001158 |...)copy SMILEScopy InChI
Affinity DataIC50: 86nMAssay Description:Inhibition of human Arg1More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WS8XZCPubMed
TargetArginase-1(Homo sapiens (Human))TBA
LigandPNGBDBM50538522(CHEMBL4633222)copy SMILEScopy InChI
Affinity DataIC50: 100nMAssay Description:Inhibition of human Arg1More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WS8XZCPubMed
TargetArginase-1(Homo sapiens (Human))TBA
LigandPNGBDBM50538525(CHEMBL4647364)copy SMILEScopy InChI
Affinity DataIC50: 100nMAssay Description:Inhibition of human Arg1More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WS8XZCPubMed
TargetArginase-1(Homo sapiens (Human))TBA
LigandPNGBDBM50561048(CHEMBL4796018)copy SMILES
Affinity DataIC50: 100nMAssay Description:Inhibition of human Arg1More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WS8XZCPubMed
TargetArginase-1(Homo sapiens (Human))TBA
LigandPNGBDBM50538547(CHEMBL4648504)copy SMILEScopy InChI
Affinity DataIC50: 100nMAssay Description:Inhibition of human Arg1More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WS8XZCPubMed
TargetArginase-2, mitochondrial(Homo sapiens (Human))TBA
LigandPNGBDBM50561049(CHEMBL4793482)copy SMILES
Affinity DataIC50: 100nMAssay Description:Inhibition of human Arg2More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WS8XZCPubMed
TargetArginase-1(Homo sapiens (Human))TBA
LigandPNGBDBM50538525(CHEMBL4647364)copy SMILEScopy InChI
Affinity DataIC50: 108nMAssay Description:Inhibition of human Arg1 by TOGA assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WS8XZCPubMed
TargetArginase-2, mitochondrial(Homo sapiens (Human))TBA
LigandPNGBDBM50511658(Cb-1158 | INCB-001158 | Incb 001158 | Incb001158 |...)copy SMILEScopy InChI
Affinity DataIC50: 296nMAssay Description:Inhibition of human Arg2More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WS8XZCPubMed
TargetArginase-1(Homo sapiens (Human))TBA
LigandPNGBDBM50561043(CHEMBL4746323 | US11420984, Example 9)copy SMILES
Affinity DataIC50: 320nMAssay Description:Inhibition of human Arg1 by TOGA assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WS8XZCPubMed
TargetArginase-2, mitochondrial(Homo sapiens (Human))TBA
LigandPNGBDBM50561043(CHEMBL4746323 | US11420984, Example 9)copy SMILES
Affinity DataIC50: 330nMAssay Description:Inhibition of human Arg2 by TOGA assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WS8XZCPubMed
TargetArginase-1(Homo sapiens (Human))TBA
LigandPNGBDBM50561044(CHEMBL4743587 | US11420984, Example 20)copy SMILES
Affinity DataIC50: 340nMAssay Description:Inhibition of human Arg1 by TOGA assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WS8XZCPubMed
TargetArginase-2, mitochondrial(Homo sapiens (Human))TBA
LigandPNGBDBM50561053(CHEMBL4750602)copy SMILES
Affinity DataIC50: 500nMAssay Description:Inhibition of human Arg2More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WS8XZCPubMed
TargetArginase-2, mitochondrial(Homo sapiens (Human))TBA
LigandPNGBDBM50561052(CHEMBL4755855)copy SMILES
Affinity DataIC50: 500nMAssay Description:Inhibition of human Arg2More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WS8XZCPubMed
TargetArginase-2, mitochondrial(Homo sapiens (Human))TBA
LigandPNGBDBM50561051(CHEMBL4749434)copy SMILES
Affinity DataIC50: 500nMAssay Description:Inhibition of human Arg2More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WS8XZCPubMed
TargetArginase-2, mitochondrial(Homo sapiens (Human))TBA
LigandPNGBDBM50561044(CHEMBL4743587 | US11420984, Example 20)copy SMILES
Affinity DataIC50: 520nMAssay Description:Inhibition of human Arg2 by TOGA assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WS8XZCPubMed
TargetArginase-1(Rattus norvegicus)TBA
LigandPNGBDBM50008099(CHEMBL1234777)copy SMILEScopy InChI
Affinity DataIC50: 800nMAssay Description:Inhibition of rat Arg1 at pH 7.4More data for this Ligand-Target Pair
TargetArginase-1(Rattus norvegicus)TBA
LigandPNGBDBM50350311(CHEMBL1812661)copy SMILEScopy InChI
Affinity DataIC50: 800nMAssay Description:Inhibition of rat Arg1 at pH 7.4More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WS8XZCPubMed
TargetArginase-1(Homo sapiens (Human))TBA
LigandPNGBDBM50561050(CHEMBL4748105)copy SMILES
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of human Arg1More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WS8XZCPubMed
TargetArginase-2, mitochondrial(Homo sapiens (Human))TBA
LigandPNGBDBM50561050(CHEMBL4748105)copy SMILES
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of human Arg2More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WS8XZCPubMed
TargetArginase-1(Homo sapiens (Human))TBA
LigandPNGBDBM50561038(CHEMBL4752307 | US11420984, Example 7)copy SMILES
Affinity DataIC50: 4.30E+3nMAssay Description:Inhibition of human Arg1More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WS8XZCPubMed
TargetArginase-1(Rattus norvegicus)TBA
LigandPNGBDBM50561034(CHEMBL4244287)copy SMILES
Affinity DataIC50: 5.00E+3nMAssay Description:Inhibition of rat Arg1 at pH 7.4More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WS8XZCPubMed
TargetArginase-2, mitochondrial(Homo sapiens (Human))TBA
LigandPNGBDBM50561050(CHEMBL4748105)copy SMILES
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human Arg2 by cell based assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WS8XZCPubMed
TargetArginase-1(Homo sapiens (Human))TBA
LigandPNGBDBM50561050(CHEMBL4748105)copy SMILES
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human Arg1 by cell based assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WS8XZCPubMed
TargetArginase-1(Rattus norvegicus)TBA
LigandPNGBDBM50230418(CHEMBL260629 | N(gamma)-hydroxy-L-arginine | N-OME...)copy SMILEScopy InChI
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibition of rat Arg1 at pH 7.4More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WS8XZCPubMedMMDB
TargetHistone deacetylase(Homo sapiens (Human))
Wroclaw University of Technology

Curated by ChEMBL
LigandPNGBDBM50138810(CHEMBL3752558)copy SMILEScopy InChI
Affinity DataIC50: 2.90E+5nMAssay Description:Inhibition of HDAC in human LoVo/DX cells using Boc-Lys(Ac)-AMC as substrate assessed as release of AMC pre-incubated for 15 mins followed by substra...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2D220G2PubMed
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