Compile Data Set for Download or QSAR
Found 12 Enz. Inhib. hit(s) with Target = 'Arginase-1' and Ligand = 'BDBM50008099'
TargetArginase-1(Rattus norvegicus)TBA
LigandPNGBDBM50008099(CHEMBL1234777)copy SMILEScopy InChI
Affinity DataIC50: 800nMAssay Description:Inhibition of rat Arg1 at pH 7.4More data for this Ligand-Target Pair
TargetArginase-1(Rattus norvegicus)TBA
LigandPNGBDBM50008099(CHEMBL1234777)copy SMILEScopy InChI
Affinity DataIC50: 800nMMore data for this Ligand-Target Pair
TargetArginase-1(Homo sapiens (Human))TBA
LigandPNGBDBM50008099(CHEMBL1234777)copy SMILEScopy InChI
Affinity DataIC50: 1.36E+3nMAssay Description:Inhibition of human recombinant arginase 1 expressed in Escherichia coli BL21 (DE3) assessed as reduction in urea production using L-arginine as subs...More data for this Ligand-Target Pair
TargetArginase-1(Rattus norvegicus)TBA
LigandPNGBDBM50008099(CHEMBL1234777)copy SMILEScopy InChI
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibition of rat liver arginaseMore data for this Ligand-Target Pair
TargetArginase-1(Bos taurus)TBA
LigandPNGBDBM50008099(CHEMBL1234777)copy SMILEScopy InChI
Affinity DataIC50: 2.70E+3nMAssay Description:Inhibition of recombinant bovine liver ARGI using L-arginine as substrate incubated for 60 mins by spectroscopic analysisMore data for this Ligand-Target Pair
TargetArginase-1(Homo sapiens (Human))TBA
LigandPNGBDBM50008099(CHEMBL1234777)copy SMILEScopy InChI
Affinity DataIC50: 6.00E+3nMAssay Description:Inhibition of recombinant human liver ARGI using L-arginine as substrate incubated for 60 mins by spectroscopic analysisMore data for this Ligand-Target Pair
TargetArginase-1(Homo sapiens (Human))TBA
LigandPNGBDBM50008099(CHEMBL1234777)copy SMILEScopy InChI
Affinity DataKd:  517nMAssay Description:Binding affinity to human Arg1 at pH 8.5More data for this Ligand-Target Pair
TargetArginase-1(Homo sapiens (Human))TBA
LigandPNGBDBM50008099(CHEMBL1234777)copy SMILEScopy InChI
Affinity DataKd:  47nMAssay Description:Binding affinity to arginase 1 (unknown origin)More data for this Ligand-Target Pair