Compile Data Set for Download or QSAR
Found 223 with Last Name = 'ostenfeld' and Initial = 't'
Targethek293 luciferase(Human immunodeficiency virus type 1 group M subtyp...)TBA
LigandPNGBDBM578497(US11479539, Compound 16)copy SMILES
Affinity DataEC50:  660nMAssay Description:Purpose of the AssayThe purpose of this assay is to identify small molecule inhibitors of Keap1, preventing Keap1 binding to Nrf2, and thus activatin...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2GQ720PUS Patent
Targethek293 luciferase(Human immunodeficiency virus type 1 group M subtyp...)TBA
LigandPNGBDBM578498(US11479539, Compound 17)copy SMILES
Affinity DataEC50:  309nMAssay Description:Purpose of the AssayThe purpose of this assay is to identify small molecule inhibitors of Keap1, preventing Keap1 binding to Nrf2, and thus activatin...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2GQ720PUS Patent
Targethek293 luciferase(Human immunodeficiency virus type 1 group M subtyp...)TBA
LigandPNGBDBM578499(US11479539, Compound 18)copy SMILES
Affinity DataEC50:  265nMAssay Description:Purpose of the AssayThe purpose of this assay is to identify small molecule inhibitors of Keap1, preventing Keap1 binding to Nrf2, and thus activatin...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2GQ720PUS Patent
Targethek293 luciferase(Human immunodeficiency virus type 1 group M subtyp...)TBA
LigandPNGBDBM578500(US11479539, Compound 19)copy SMILES
Affinity DataEC50:  1.24E+3nMAssay Description:Purpose of the AssayThe purpose of this assay is to identify small molecule inhibitors of Keap1, preventing Keap1 binding to Nrf2, and thus activatin...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2GQ720PUS Patent
Targethek293 luciferase(Human immunodeficiency virus type 1 group M subtyp...)TBA
LigandPNGBDBM578501(US11479539, Compound 20)copy SMILES
Affinity DataEC50:  126nMAssay Description:Purpose of the AssayThe purpose of this assay is to identify small molecule inhibitors of Keap1, preventing Keap1 binding to Nrf2, and thus activatin...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2GQ720PUS Patent
Targethek293 luciferase(Human immunodeficiency virus type 1 group M subtyp...)TBA
LigandPNGBDBM578502(US11479539, Compound 21)copy SMILES
Affinity DataEC50:  452nMAssay Description:Purpose of the AssayThe purpose of this assay is to identify small molecule inhibitors of Keap1, preventing Keap1 binding to Nrf2, and thus activatin...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2GQ720PUS Patent
Targethek293 luciferase(Human immunodeficiency virus type 1 group M subtyp...)TBA
LigandPNGBDBM578503(US11479539, Compound 22)copy SMILES
Affinity DataEC50:  45nMAssay Description:Purpose of the AssayThe purpose of this assay is to identify small molecule inhibitors of Keap1, preventing Keap1 binding to Nrf2, and thus activatin...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2GQ720PUS Patent
Targethek293 luciferase(Human immunodeficiency virus type 1 group M subtyp...)TBA
LigandPNGBDBM50502729(CHEMBL4593124 | US11479539, Compound 23)copy SMILEScopy InChI
Affinity DataEC50:  56nMAssay Description:Purpose of the AssayThe purpose of this assay is to identify small molecule inhibitors of Keap1, preventing Keap1 binding to Nrf2, and thus activatin...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2GQ720PUS Patent
Targethek293 luciferase(Human immunodeficiency virus type 1 group M subtyp...)TBA
LigandPNGBDBM578505(US11479539, Compound 24)copy SMILES
Affinity DataEC50: >1.00E+4nMAssay Description:Purpose of the AssayThe purpose of this assay is to identify small molecule inhibitors of Keap1, preventing Keap1 binding to Nrf2, and thus activatin...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2GQ720PUS Patent
Targethek293 luciferase(Human immunodeficiency virus type 1 group M subtyp...)TBA
LigandPNGBDBM578506(US11479539, Compound 25)copy SMILES
Affinity DataEC50:  70nMAssay Description:Purpose of the AssayThe purpose of this assay is to identify small molecule inhibitors of Keap1, preventing Keap1 binding to Nrf2, and thus activatin...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2GQ720PUS Patent
Targethek293 luciferase(Human immunodeficiency virus type 1 group M subtyp...)TBA
LigandPNGBDBM578507(3-(5-fluoro-3- (trifluoromethyl)py- ridin-2-yl)-3-...)copy SMILES
Affinity DataEC50:  24nMAssay Description:Purpose of the AssayThe purpose of this assay is to identify small molecule inhibitors of Keap1, preventing Keap1 binding to Nrf2, and thus activatin...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2GQ720PUS Patent
Targethek293 luciferase(Human immunodeficiency virus type 1 group M subtyp...)TBA
LigandPNGBDBM578508(3-(5- fluoropyridin-2- yl)-3-methoxy- 5,5-dimethyl...)copy SMILES
Affinity DataEC50:  180nMAssay Description:Purpose of the AssayThe purpose of this assay is to identify small molecule inhibitors of Keap1, preventing Keap1 binding to Nrf2, and thus activatin...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2GQ720PUS Patent
Targethek293 luciferase(Human immunodeficiency virus type 1 group M subtyp...)TBA
LigandPNGBDBM578509(3-(3,5- difluoropyridin-2- yl)-3-methoxy- 5,5-dime...)copy SMILES
Affinity DataEC50:  36nMAssay Description:Purpose of the AssayThe purpose of this assay is to identify small molecule inhibitors of Keap1, preventing Keap1 binding to Nrf2, and thus activatin...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2GQ720PUS Patent
Targethek293 luciferase(Human immunodeficiency virus type 1 group M subtyp...)TBA
LigandPNGBDBM578510(3-(2,6- dimethylpyridin- 3-yl)-3-methoxy- 5,5-dime...)copy SMILES
Affinity DataEC50:  91nMAssay Description:Purpose of the AssayThe purpose of this assay is to identify small molecule inhibitors of Keap1, preventing Keap1 binding to Nrf2, and thus activatin...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2GQ720PUS Patent
Targethek293 luciferase(Human immunodeficiency virus type 1 group M subtyp...)TBA
LigandPNGBDBM578511(3-methoxy-5,5- dimethyl-3-(6- methylpyrazin-2- yl)...)copy SMILES
Affinity DataEC50:  458nMAssay Description:Purpose of the AssayThe purpose of this assay is to identify small molecule inhibitors of Keap1, preventing Keap1 binding to Nrf2, and thus activatin...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2GQ720PUS Patent
Targethek293 luciferase(Human immunodeficiency virus type 1 group M subtyp...)TBA
LigandPNGBDBM578512(3-(5-fluoro-3- methylpyridin-2- yl)-3-methoxy- 5,5...)copy SMILES
Affinity DataEC50:  19nMAssay Description:Purpose of the AssayThe purpose of this assay is to identify small molecule inhibitors of Keap1, preventing Keap1 binding to Nrf2, and thus activatin...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2GQ720PUS Patent
Targethek293 luciferase(Human immunodeficiency virus type 1 group M subtyp...)TBA
LigandPNGBDBM578513(3-(5- chloropyridin-2- yl)-3-methoxy- 5,5-dimethyl...)copy SMILES
Affinity DataEC50:  55nMAssay Description:Purpose of the AssayThe purpose of this assay is to identify small molecule inhibitors of Keap1, preventing Keap1 binding to Nrf2, and thus activatin...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2GQ720PUS Patent
Targethek293 luciferase(Human immunodeficiency virus type 1 group M subtyp...)TBA
LigandPNGBDBM578514(3-methoxy-5,5- dimethyl-6-oxo- 3-(4-(tri- fluorome...)copy SMILES
Affinity DataEC50:  383nMAssay Description:Purpose of the AssayThe purpose of this assay is to identify small molecule inhibitors of Keap1, preventing Keap1 binding to Nrf2, and thus activatin...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2GQ720PUS Patent
Targethek293 luciferase(Human immunodeficiency virus type 1 group M subtyp...)TBA
LigandPNGBDBM578515(3-methoxy-5,5- dimethyl-3-(3- methylthiophen- 2-yl...)copy SMILES
Affinity DataEC50:  12nMAssay Description:Purpose of the AssayThe purpose of this assay is to identify small molecule inhibitors of Keap1, preventing Keap1 binding to Nrf2, and thus activatin...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2GQ720PUS Patent
Targethek293 luciferase(Human immunodeficiency virus type 1 group M subtyp...)TBA
LigandPNGBDBM578516(3-ethoxy-5,5- dimethyl-6-oxo- 3-(3- (trifluorometh...)copy SMILES
Affinity DataEC50:  39nMAssay Description:Purpose of the AssayThe purpose of this assay is to identify small molecule inhibitors of Keap1, preventing Keap1 binding to Nrf2, and thus activatin...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2GQ720PUS Patent
Targethek293 luciferase(Human immunodeficiency virus type 1 group M subtyp...)TBA
LigandPNGBDBM578517(3-methoxy-5,5- dimethyl-3-(4- methylthiazol-2- yl)...)copy SMILES
Affinity DataEC50:  96nMAssay Description:Purpose of the AssayThe purpose of this assay is to identify small molecule inhibitors of Keap1, preventing Keap1 binding to Nrf2, and thus activatin...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2GQ720PUS Patent
Targethek293 luciferase(Human immunodeficiency virus type 1 group M subtyp...)TBA
LigandPNGBDBM578518(3-ethoxy-3-(5- fluoropyridin-2- yl)-5,5-dimethyl- ...)copy SMILES
Affinity DataEC50:  86nMAssay Description:Purpose of the AssayThe purpose of this assay is to identify small molecule inhibitors of Keap1, preventing Keap1 binding to Nrf2, and thus activatin...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2GQ720PUS Patent
Targethek293 luciferase(Human immunodeficiency virus type 1 group M subtyp...)TBA
LigandPNGBDBM578519((S)-3-methoxy- 5,5-dimethyl-3- (5-methylthiazol- 4...)copy SMILES
Affinity DataEC50:  132nMAssay Description:Purpose of the AssayThe purpose of this assay is to identify small molecule inhibitors of Keap1, preventing Keap1 binding to Nrf2, and thus activatin...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2GQ720PUS Patent
Targethek293 luciferase(Human immunodeficiency virus type 1 group M subtyp...)TBA
LigandPNGBDBM578520(3-methoxy-5,5- dimethyl-6-oxo- 3-(thiazol-2- yl)cy...)copy SMILES
Affinity DataEC50:  125nMAssay Description:Purpose of the AssayThe purpose of this assay is to identify small molecule inhibitors of Keap1, preventing Keap1 binding to Nrf2, and thus activatin...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2GQ720PUS Patent
Targethek293 luciferase(Human immunodeficiency virus type 1 group M subtyp...)TBA
LigandPNGBDBM578521((S)-3-methoxy- 5,5-dimethyl-3- (5-methylthiazol- 2...)copy SMILES
Affinity DataEC50:  38nMAssay Description:Purpose of the AssayThe purpose of this assay is to identify small molecule inhibitors of Keap1, preventing Keap1 binding to Nrf2, and thus activatin...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2GQ720PUS Patent
Targethek293 luciferase(Human immunodeficiency virus type 1 group M subtyp...)TBA
LigandPNGBDBM578522(3-methoxy-5,5- dimethyl-6-oxo- 3-(3- (trifluoromet...)copy SMILES
Affinity DataEC50:  11nMAssay Description:Purpose of the AssayThe purpose of this assay is to identify small molecule inhibitors of Keap1, preventing Keap1 binding to Nrf2, and thus activatin...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2GQ720PUS Patent
Targethek293 luciferase(Human immunodeficiency virus type 1 group M subtyp...)TBA
LigandPNGBDBM50502734(CHEMBL4442320 | US11479539, Compound 42)copy SMILEScopy InChI
Affinity DataEC50:  33nMAssay Description:Purpose of the AssayThe purpose of this assay is to identify small molecule inhibitors of Keap1, preventing Keap1 binding to Nrf2, and thus activatin...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2GQ720PUS Patent
Targethek293 luciferase(Human immunodeficiency virus type 1 group M subtyp...)TBA
LigandPNGBDBM578524(3-methoxy-5,5- dimethyl-3-(4- methylthiazol-5- yl)...)copy SMILES
Affinity DataEC50:  129nMAssay Description:Purpose of the AssayThe purpose of this assay is to identify small molecule inhibitors of Keap1, preventing Keap1 binding to Nrf2, and thus activatin...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2GQ720PUS Patent
Targethek293 luciferase(Human immunodeficiency virus type 1 group M subtyp...)TBA
LigandPNGBDBM578509(3-(3,5- difluoropyridin-2- yl)-3-methoxy- 5,5-dime...)copy SMILES
Affinity DataEC50:  37nMAssay Description:Purpose of the AssayThe purpose of this assay is to identify small molecule inhibitors of Keap1, preventing Keap1 binding to Nrf2, and thus activatin...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2GQ720PUS Patent
Targethek293 luciferase(Human immunodeficiency virus type 1 group M subtyp...)TBA
LigandPNGBDBM578526(3-(5-chloro-3- (difluoromethyl)py- ridin-2-yl)-3- ...)copy SMILES
Affinity DataEC50:  28nMAssay Description:Purpose of the AssayThe purpose of this assay is to identify small molecule inhibitors of Keap1, preventing Keap1 binding to Nrf2, and thus activatin...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2GQ720PUS Patent
Targethek293 luciferase(Human immunodeficiency virus type 1 group M subtyp...)TBA
LigandPNGBDBM578527(3-(2,4- dimethylthiazol- 5-yl)-3-methoxy- 5,5-dime...)copy SMILES
Affinity DataEC50:  304nMAssay Description:Purpose of the AssayThe purpose of this assay is to identify small molecule inhibitors of Keap1, preventing Keap1 binding to Nrf2, and thus activatin...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2GQ720PUS Patent
Targethek293 luciferase(Human immunodeficiency virus type 1 group M subtyp...)TBA
LigandPNGBDBM50502728(CHEMBL4542755 | US11479539, Compound 174)copy SMILEScopy InChI
Affinity DataEC50:  8nMAssay Description:Purpose of the AssayThe purpose of this assay is to identify small molecule inhibitors of Keap1, preventing Keap1 binding to Nrf2, and thus activatin...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2GQ720PUS Patent
Targethek293 luciferase(Human immunodeficiency virus type 1 group M subtyp...)TBA
LigandPNGBDBM50502727(CHEMBL4584154 | US11479539, Compound 48)copy SMILEScopy InChI
Affinity DataEC50:  6nMAssay Description:Purpose of the AssayThe purpose of this assay is to identify small molecule inhibitors of Keap1, preventing Keap1 binding to Nrf2, and thus activatin...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2GQ720PUS Patent
Targethek293 luciferase(Human immunodeficiency virus type 1 group M subtyp...)TBA
LigandPNGBDBM578530(US11479539, Compound 126 | US11479539, Compound 49)copy SMILES
Affinity DataEC50:  138nMAssay Description:Purpose of the AssayThe purpose of this assay is to identify small molecule inhibitors of Keap1, preventing Keap1 binding to Nrf2, and thus activatin...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2GQ720PUS Patent
Targethek293 luciferase(Human immunodeficiency virus type 1 group M subtyp...)TBA
LigandPNGBDBM578531(7-methoxy-7-(6- (2- methylpyrimidin- 5-yl)pyridin-...)copy SMILES
Affinity DataEC50:  30nMAssay Description:Purpose of the AssayThe purpose of this assay is to identify small molecule inhibitors of Keap1, preventing Keap1 binding to Nrf2, and thus activatin...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2GQ720PUS Patent
Targethek293 luciferase(Human immunodeficiency virus type 1 group M subtyp...)TBA
LigandPNGBDBM578532(7-methoxy-4- oxo-7-(6- (pyrimidin-5- yl)pyridin-2-...)copy SMILES
Affinity DataEC50:  48nMAssay Description:Purpose of the AssayThe purpose of this assay is to identify small molecule inhibitors of Keap1, preventing Keap1 binding to Nrf2, and thus activatin...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2GQ720PUS Patent
Targethek293 luciferase(Human immunodeficiency virus type 1 group M subtyp...)TBA
LigandPNGBDBM578533(7-(6-(3,5- dimethylisoxazol- 4-yl)pyridin-2- yl)-7...)copy SMILES
Affinity DataEC50:  74nMAssay Description:Purpose of the AssayThe purpose of this assay is to identify small molecule inhibitors of Keap1, preventing Keap1 binding to Nrf2, and thus activatin...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2GQ720PUS Patent
Targethek293 luciferase(Human immunodeficiency virus type 1 group M subtyp...)TBA
LigandPNGBDBM578534(7-methoxy-7-(6- (1-methyl-1H- pyrazol-5- yl)pyridi...)copy SMILES
Affinity DataEC50:  133nMAssay Description:Purpose of the AssayThe purpose of this assay is to identify small molecule inhibitors of Keap1, preventing Keap1 binding to Nrf2, and thus activatin...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2GQ720PUS Patent
Targethek293 luciferase(Human immunodeficiency virus type 1 group M subtyp...)TBA
LigandPNGBDBM578535(US11479539, Compound 131 | US11479539, Compound 54)copy SMILES
Affinity DataEC50:  363nMAssay Description:Purpose of the AssayThe purpose of this assay is to identify small molecule inhibitors of Keap1, preventing Keap1 binding to Nrf2, and thus activatin...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2GQ720PUS Patent
Targethek293 luciferase(Human immunodeficiency virus type 1 group M subtyp...)TBA
LigandPNGBDBM50502726(CHEMBL4583328 | US11479539, Compound 55)copy SMILEScopy InChI
Affinity DataEC50:  14nMAssay Description:Purpose of the AssayThe purpose of this assay is to identify small molecule inhibitors of Keap1, preventing Keap1 binding to Nrf2, and thus activatin...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2GQ720PUS Patent
Targethek293 luciferase(Human immunodeficiency virus type 1 group M subtyp...)TBA
LigandPNGBDBM578491(US11479539, Compound 10)copy SMILES
Affinity DataEC50: >3.00E+4nMAssay Description:Purpose of the AssayThe purpose of this assay is to identify small molecule inhibitors of Keap1, preventing Keap1 binding to Nrf2, and thus activatin...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2GQ720PUS Patent
Targethek293 luciferase(Human immunodeficiency virus type 1 group M subtyp...)TBA
LigandPNGBDBM578492(US11479539, Compound 11)copy SMILES
Affinity DataEC50:  85nMAssay Description:Purpose of the AssayThe purpose of this assay is to identify small molecule inhibitors of Keap1, preventing Keap1 binding to Nrf2, and thus activatin...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2GQ720PUS Patent
Targethek293 luciferase(Human immunodeficiency virus type 1 group M subtyp...)TBA
LigandPNGBDBM578493(US11479539, Compound 12)copy SMILES
Affinity DataEC50:  119nMAssay Description:Purpose of the AssayThe purpose of this assay is to identify small molecule inhibitors of Keap1, preventing Keap1 binding to Nrf2, and thus activatin...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2GQ720PUS Patent
Targethek293 luciferase(Human immunodeficiency virus type 1 group M subtyp...)TBA
LigandPNGBDBM578494(US11479539, Compound 13)copy SMILES
Affinity DataEC50:  1.00E+4nMAssay Description:Purpose of the AssayThe purpose of this assay is to identify small molecule inhibitors of Keap1, preventing Keap1 binding to Nrf2, and thus activatin...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2GQ720PUS Patent
Targethek293 luciferase(Human immunodeficiency virus type 1 group M subtyp...)TBA
LigandPNGBDBM578495(US11479539, Compound 107 | US11479539, Compound 11...)copy SMILES
Affinity DataEC50:  12nMAssay Description:Purpose of the AssayThe purpose of this assay is to identify small molecule inhibitors of Keap1, preventing Keap1 binding to Nrf2, and thus activatin...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2GQ720PUS Patent
Targethek293 luciferase(Human immunodeficiency virus type 1 group M subtyp...)TBA
LigandPNGBDBM50502724(CHEMBL4463989 | US11479539, Compound 122)copy SMILEScopy InChI
Affinity DataEC50:  24nMAssay Description:Purpose of the AssayThe purpose of this assay is to identify small molecule inhibitors of Keap1, preventing Keap1 binding to Nrf2, and thus activatin...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2GQ720PUS Patent
Targethek293 luciferase(Human immunodeficiency virus type 1 group M subtyp...)TBA
LigandPNGBDBM578537(7-methoxy-4- oxo-7-(pyridin- 2- yl)spiro[2.5]oct- ...)copy SMILES
Affinity DataEC50:  179nMAssay Description:Purpose of the AssayThe purpose of this assay is to identify small molecule inhibitors of Keap1, preventing Keap1 binding to Nrf2, and thus activatin...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2GQ720PUS Patent
Targethek293 luciferase(Human immunodeficiency virus type 1 group M subtyp...)TBA
LigandPNGBDBM578538(7-methoxy-4- oxo-7-[3- (trifluoromethyl) pyridin-2...)copy SMILES
Affinity DataEC50:  47nMAssay Description:Purpose of the AssayThe purpose of this assay is to identify small molecule inhibitors of Keap1, preventing Keap1 binding to Nrf2, and thus activatin...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2GQ720PUS Patent
Targethek293 luciferase(Human immunodeficiency virus type 1 group M subtyp...)TBA
LigandPNGBDBM578539(7-methoxy-4-7- (4-methyl-1,3- thiazol-2-yl)-4- oxo...)copy SMILES
Affinity DataEC50:  261nMAssay Description:Purpose of the AssayThe purpose of this assay is to identify small molecule inhibitors of Keap1, preventing Keap1 binding to Nrf2, and thus activatin...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2GQ720PUS Patent
Targethek293 luciferase(Human immunodeficiency virus type 1 group M subtyp...)TBA
LigandPNGBDBM578540(7-(3,5- difluoropyridin- 2-yl)-7- methoxy-4- oxosp...)copy SMILES
Affinity DataEC50:  153nMAssay Description:Purpose of the AssayThe purpose of this assay is to identify small molecule inhibitors of Keap1, preventing Keap1 binding to Nrf2, and thus activatin...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2GQ720PUS Patent
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