Compile Data Set for Download or QSAR
Found 141 with Last Name = 'nielsen' and Initial = 'te'
TargetDNA gyrase subunit A/B(Staphylococcus aureus)TBA
LigandPNGBDBM50596272(CHEMBL5199813)copy SMILES
Affinity DataIC50: 190nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2X06C35PubMed
TargetDNA gyrase subunit A/B(Escherichia coli (strain K12))TBA
LigandPNGBDBM21690(1-cyclopropyl-6-fluoro-4-oxo-7-(piperazin-1-yl)-1,...)copy SMILEScopy InChI
Affinity DataIC50: 230nMMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2X06C35PubMedDrugBank
TargetDNA gyrase subunit A/B(Staphylococcus aureus)TBA
LigandPNGBDBM50596278(CHEMBL5178214)copy SMILES
Affinity DataIC50: 280nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2X06C35PubMed
TargetDNA gyrase subunit A/B(Staphylococcus aureus)TBA
LigandPNGBDBM50596263(CHEMBL5207657)copy SMILES
Affinity DataIC50: 280nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2X06C35PubMed
TargetDNA gyrase subunit A/B(Staphylococcus aureus)TBA
LigandPNGBDBM50393503(CHEMBL2158050)copy SMILEScopy InChI
Affinity DataIC50: 340nMMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2X06C35PubMed
TargetDNA gyrase subunit A/B(Staphylococcus aureus)TBA
LigandPNGBDBM50596275(CHEMBL5176348)copy SMILES
Affinity DataIC50: 370nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2X06C35PubMed
TargetDNA gyrase subunit A/B(Staphylococcus aureus)TBA
LigandPNGBDBM50596261(CHEMBL5176134)copy SMILES
Affinity DataIC50: 370nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2X06C35PubMed
TargetDNA gyrase subunit A/B(Staphylococcus aureus)TBA
LigandPNGBDBM50596271(CHEMBL5176046)copy SMILES
Affinity DataIC50: 460nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2X06C35PubMed
TargetDNA gyrase subunit A/B(Staphylococcus aureus)TBA
LigandPNGBDBM50596264(CHEMBL5206355)copy SMILES
Affinity DataIC50: 480nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2X06C35PubMed
TargetDNA gyrase subunit A/B(Staphylococcus aureus)TBA
LigandPNGBDBM50596274(CHEMBL5204986)copy SMILES
Affinity DataIC50: 540nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2X06C35PubMed
TargetDNA gyrase subunit A/B(Staphylococcus aureus)TBA
LigandPNGBDBM50596262(CHEMBL5176331)copy SMILES
Affinity DataIC50: 680nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2X06C35PubMed
TargetDNA topoisomerase 4 subunit A/B(Staphylococcus aureus)TBA
LigandPNGBDBM50596262(CHEMBL5176331)copy SMILES
Affinity DataIC50: 1.81E+3nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2X06C35PubMed
TargetHTH-type quorum-sensing regulator RhlR(Pseudomonas aeruginosa (strain ATCC 15692 / PAO1 /...)
Nanyang Technological University

Curated by ChEMBL
LigandPNGBDBM50470115(CHEMBL4098007)copy SMILEScopy InChI
Affinity DataIC50: 2.03E+3nMAssay Description:Inhibition of quorum sensing regulator protein RhlR in Pseudomonas aeruginosa PAO1 harboring reporter plasmid rhlA-gfp assessed as reduction in rhlA ...More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2125WC6PubMed
TargetDNA topoisomerase 4 subunit A/B(Staphylococcus aureus)TBA
LigandPNGBDBM50596278(CHEMBL5178214)copy SMILES
Affinity DataIC50: 2.41E+3nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2X06C35PubMed
TargetDNA topoisomerase 4 subunit A/B(Staphylococcus aureus)TBA
LigandPNGBDBM50596264(CHEMBL5206355)copy SMILES
Affinity DataIC50: 2.47E+3nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2X06C35PubMed
TargetDNA topoisomerase 4 subunit A/B(Staphylococcus aureus)TBA
LigandPNGBDBM50596272(CHEMBL5199813)copy SMILES
Affinity DataIC50: 3.36E+3nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2X06C35PubMed
TargetDNA topoisomerase 4 subunit A/B(Staphylococcus aureus)TBA
LigandPNGBDBM50596275(CHEMBL5176348)copy SMILES
Affinity DataIC50: 3.82E+3nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2X06C35PubMed
TargetDNA gyrase subunit A/B(Staphylococcus aureus)TBA
LigandPNGBDBM21690(1-cyclopropyl-6-fluoro-4-oxo-7-(piperazin-1-yl)-1,...)copy SMILEScopy InChI
Affinity DataIC50: 3.84E+3nMMore data for this Ligand-Target Pair
TargetDNA gyrase subunit A/B(Escherichia coli (strain K12))TBA
LigandPNGBDBM50393503(CHEMBL2158050)copy SMILEScopy InChI
Affinity DataIC50: 3.90E+3nMMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2X06C35PubMed
TargetDNA gyrase subunit A/B(Escherichia coli (strain K12))TBA
LigandPNGBDBM50596261(CHEMBL5176134)copy SMILES
Affinity DataIC50: 5.40E+3nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2X06C35PubMed
TargetDNA gyrase subunit A/B(Escherichia coli (strain K12))TBA
LigandPNGBDBM50596278(CHEMBL5178214)copy SMILES
Affinity DataIC50: 6.46E+3nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2X06C35PubMed
TargetDNA topoisomerase 4 subunit A/B(Staphylococcus aureus)TBA
LigandPNGBDBM50596261(CHEMBL5176134)copy SMILES
Affinity DataIC50: 7.64E+3nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2X06C35PubMed
TargetDNA topoisomerase 4 subunit A/B(Staphylococcus aureus)TBA
LigandPNGBDBM50393503(CHEMBL2158050)copy SMILEScopy InChI
Affinity DataIC50: 8.80E+3nMMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2X06C35PubMed
TargetDNA topoisomerase 4 subunit A/B(Staphylococcus aureus)TBA
LigandPNGBDBM21690(1-cyclopropyl-6-fluoro-4-oxo-7-(piperazin-1-yl)-1,...)copy SMILEScopy InChI
Affinity DataIC50: 9.16E+3nMMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2X06C35PubMed
TargetDNA topoisomerase 4 subunit A/B(Staphylococcus aureus)TBA
LigandPNGBDBM50596263(CHEMBL5207657)copy SMILES
Affinity DataIC50: 9.92E+3nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2X06C35PubMed
TargetDNA topoisomerase 4 subunit A/B(Staphylococcus aureus)TBA
LigandPNGBDBM50596271(CHEMBL5176046)copy SMILES
Affinity DataIC50: 1.02E+4nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2X06C35PubMed
TargetDNA topoisomerase 4 subunit A/B(Staphylococcus aureus)TBA
LigandPNGBDBM50596274(CHEMBL5204986)copy SMILES
Affinity DataIC50: 1.26E+4nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2X06C35PubMed
TargetDNA gyrase subunit A/B(Escherichia coli (strain K12))TBA
LigandPNGBDBM50596269(CHEMBL5183842)copy SMILES
Affinity DataIC50: 1.84E+4nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2X06C35PubMed
TargetHTH-type quorum-sensing regulator RhlR(Pseudomonas aeruginosa (strain ATCC 15692 / PAO1 /...)
Nanyang Technological University

Curated by ChEMBL
LigandPNGBDBM50240785((E)-1-Allyldisulfanyl-3-(prop-2-ene-1-sulfinyl)-pr...)copy SMILEScopy InChI
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of quorum sensing regulator protein RhlR in Pseudomonas aeruginosa PAO1 harboring reporter plasmid rhlA-gfp assessed as reduction in rhlA ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2125WC6PubMed
TargetDNA gyrase subunit A/B(Staphylococcus aureus)TBA
LigandPNGBDBM50596269(CHEMBL5183842)copy SMILES
Affinity DataIC50: 3.00E+5nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2X06C35PubMed
TargetElastase(Pseudomonas aeruginosa)
Technical University of Denmark

Curated by ChEMBL
LigandPNGBDBM50498101(CHEMBL3403862)copy SMILEScopy InChI
Affinity DataIC50: 3.81E+5nMAssay Description:Antagonist activity at lasB in Pseudomonas aeruginosa harboring lasB-gfp gene assessed as inhibition of 3-oxo-C6-HSL-induced quorum sensing by green ...More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2F192P6PubMed
TargetElastase(Pseudomonas aeruginosa)
Technical University of Denmark

Curated by ChEMBL
LigandPNGBDBM50498105(CHEMBL3403858)copy SMILEScopy InChI
Affinity DataIC50: 4.25E+5nMAssay Description:Antagonist activity at lasB in Pseudomonas aeruginosa harboring lasB-gfp gene assessed as inhibition of 3-oxo-C6-HSL-induced quorum sensing by green ...More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2F192P6PubMed
TargetElastase(Pseudomonas aeruginosa)
Technical University of Denmark

Curated by ChEMBL
LigandPNGBDBM50498098(CHEMBL3403859)copy SMILEScopy InChI
Affinity DataIC50: 4.99E+5nMAssay Description:Antagonist activity at lasB in Pseudomonas aeruginosa harboring lasB-gfp gene assessed as inhibition of 3-oxo-C6-HSL-induced quorum sensing by green ...More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2F192P6PubMed
TargetElastase(Pseudomonas aeruginosa)
Technical University of Denmark

Curated by ChEMBL
LigandPNGBDBM50498104(CHEMBL3403865)copy SMILEScopy InChI
Affinity DataIC50: 5.82E+5nMAssay Description:Antagonist activity at lasB in Pseudomonas aeruginosa harboring lasB-gfp gene assessed as inhibition of 3-oxo-C6-HSL-induced quorum sensing by green ...More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2F192P6PubMed
TargetElastase(Pseudomonas aeruginosa)
Technical University of Denmark

Curated by ChEMBL
LigandPNGBDBM50498097(CHEMBL3403860)copy SMILEScopy InChI
Affinity DataIC50: 6.10E+5nMAssay Description:Antagonist activity at lasB in Pseudomonas aeruginosa harboring lasB-gfp gene assessed as inhibition of 3-oxo-C6-HSL-induced quorum sensing by green ...More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2F192P6PubMed
TargetElastase(Pseudomonas aeruginosa)
Technical University of Denmark

Curated by ChEMBL
LigandPNGBDBM50498102(CHEMBL3403856)copy SMILEScopy InChI
Affinity DataIC50: 6.78E+5nMAssay Description:Antagonist activity at lasB in Pseudomonas aeruginosa harboring lasB-gfp gene assessed as inhibition of 3-oxo-C6-HSL-induced quorum sensing by green ...More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2F192P6PubMed
TargetElastase(Pseudomonas aeruginosa)
Technical University of Denmark

Curated by ChEMBL
LigandPNGBDBM50498100(CHEMBL3403864)copy SMILEScopy InChI
Affinity DataIC50: 6.92E+5nMAssay Description:Antagonist activity at lasB in Pseudomonas aeruginosa harboring lasB-gfp gene assessed as inhibition of 3-oxo-C6-HSL-induced quorum sensing by green ...More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2F192P6PubMed
TargetElastase(Pseudomonas aeruginosa)
Technical University of Denmark

Curated by ChEMBL
LigandPNGBDBM50498103(CHEMBL3403861)copy SMILEScopy InChI
Affinity DataIC50: 8.89E+5nMAssay Description:Antagonist activity at lasB in Pseudomonas aeruginosa harboring lasB-gfp gene assessed as inhibition of 3-oxo-C6-HSL-induced quorum sensing by green ...More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2F192P6PubMed
TargetElastase(Pseudomonas aeruginosa)
Technical University of Denmark

Curated by ChEMBL
LigandPNGBDBM50498099(CHEMBL3403868)copy SMILEScopy InChI
Affinity DataIC50: 1.10E+6nMAssay Description:Antagonist activity at lasB in Pseudomonas aeruginosa harboring lasB-gfp gene assessed as inhibition of 3-oxo-C6-HSL-induced quorum sensing by green ...More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2F192P6PubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
CECB, Department of Chemistry, University of Copenhagen , Universitetsparken 5, 2100 Copenhagen, Denmark.

Curated by ChEMBL
LigandPNGBDBM50250214(CHEMBL4100598)copy SMILEScopy InChI
Affinity DataEC50:  2.30nMAssay Description:Agonist activity at EYFP-fused human MC4R expressed in HEK293 cells after 16 to 20 hrs by CRE-driven reporter assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VQ3535PubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
CECB, Department of Chemistry, University of Copenhagen , Universitetsparken 5, 2100 Copenhagen, Denmark.

Curated by ChEMBL
LigandPNGBDBM50029747((4S)-4-{[(1S)-1-{[(1S)-1-{[(1S)-1-{[(1S)-1-[({[(2S...)copy SMILEScopy InChI
Affinity DataEC50:  24nMAssay Description:Agonist activity at EYFP-fused human MC4R expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by luminescent enzymatic ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VQ3535PubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
CECB, Department of Chemistry, University of Copenhagen , Universitetsparken 5, 2100 Copenhagen, Denmark.

Curated by ChEMBL
LigandPNGBDBM50250212(CHEMBL4089119)copy SMILEScopy InChI
Affinity DataEC50:  185nMAssay Description:Agonist activity at EYFP-fused human MC4R expressed in HEK293 cells after 16 to 20 hrs by CRE-driven reporter assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VQ3535PubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
CECB, Department of Chemistry, University of Copenhagen , Universitetsparken 5, 2100 Copenhagen, Denmark.

Curated by ChEMBL
LigandPNGBDBM50250213(CHEMBL4104927)copy SMILEScopy InChI
Affinity DataEC50:  11nMAssay Description:Agonist activity at EYFP-fused human MC4R expressed in HEK293 cells after 16 to 20 hrs by CRE-driven reporter assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VQ3535PubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
CECB, Department of Chemistry, University of Copenhagen , Universitetsparken 5, 2100 Copenhagen, Denmark.

Curated by ChEMBL
LigandPNGBDBM50250211(CHEMBL4100221)copy SMILEScopy InChI
Affinity DataEC50: >3.00E+3nMAssay Description:Agonist activity at EYFP-fused human MC4R expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by luminescent enzymatic ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VQ3535PubMed
TargetMelanocortin receptor 5(Homo sapiens (Human))
CECB, Department of Chemistry, University of Copenhagen , Universitetsparken 5, 2100 Copenhagen, Denmark.

Curated by ChEMBL
LigandPNGBDBM50029747((4S)-4-{[(1S)-1-{[(1S)-1-{[(1S)-1-{[(1S)-1-[({[(2S...)copy SMILEScopy InChI
Affinity DataEC50:  35nMAssay Description:Agonist activity at EYFP-fused human MC5R expressed in HEK293 cells after 16 to 20 hrs by CRE-driven reporter assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VQ3535PubMed
TargetMelanocortin receptor 5(Homo sapiens (Human))
CECB, Department of Chemistry, University of Copenhagen , Universitetsparken 5, 2100 Copenhagen, Denmark.

Curated by ChEMBL
LigandPNGBDBM50250205(CHEMBL4067491)copy SMILEScopy InChI
Affinity DataEC50:  110nMAssay Description:Agonist activity at EYFP-fused human MC5R expressed in HEK293 cells after 16 to 20 hrs by CRE-driven reporter assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VQ3535PubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
CECB, Department of Chemistry, University of Copenhagen , Universitetsparken 5, 2100 Copenhagen, Denmark.

Curated by ChEMBL
LigandPNGBDBM50250206(CHEMBL4060816)copy SMILEScopy InChI
Affinity DataEC50:  9.20nMAssay Description:Agonist activity at EYFP-fused human MC4R expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by luminescent enzymatic ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VQ3535PubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
CECB, Department of Chemistry, University of Copenhagen , Universitetsparken 5, 2100 Copenhagen, Denmark.

Curated by ChEMBL
LigandPNGBDBM50250207(CHEMBL4082585)copy SMILEScopy InChI
Affinity DataEC50:  64nMAssay Description:Agonist activity at EYFP-fused human MC4R expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by luminescent enzymatic ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VQ3535PubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
CECB, Department of Chemistry, University of Copenhagen , Universitetsparken 5, 2100 Copenhagen, Denmark.

Curated by ChEMBL
LigandPNGBDBM50250208(CHEMBL4062443)copy SMILEScopy InChI
Affinity DataEC50:  792nMAssay Description:Agonist activity at EYFP-fused human MC4R expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by luminescent enzymatic ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VQ3535PubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
CECB, Department of Chemistry, University of Copenhagen , Universitetsparken 5, 2100 Copenhagen, Denmark.

Curated by ChEMBL
LigandPNGBDBM50250209(CHEMBL4090425)copy SMILEScopy InChI
Affinity DataEC50:  124nMAssay Description:Agonist activity at EYFP-fused human MC4R expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by luminescent enzymatic ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VQ3535PubMed
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