Compile Data Set for Download or QSAR
Found 86 with Last Name = 'lukasczyk' and Initial = 'u'
TargetHistamine receptor H3(Macaca mulatta (Rhesus macaque))
Sanofi US

Curated by ChEMBL
LigandPNGBDBM50434389(CHEMBL2387288)copy SMILEScopy InChI
Affinity DataKi:  1.90nMAssay Description:Displacement of [3H]N-alpha-methylhistamine from cloned rhesus monkey histamine H3 receptor transfected in CHO cells after 1 hr by scintillation coun...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2RB75Z5PubMed
TargetHistamine receptor H3(Macaca mulatta (Rhesus macaque))
Sanofi US

Curated by ChEMBL
LigandPNGBDBM50434405(CHEMBL2387306)copy SMILEScopy InChI
Affinity DataKi:  3.40nMAssay Description:Displacement of [3H]N-alpha-methylhistamine from cloned rhesus monkey histamine H3 receptor transfected in CHO cells after 1 hr by scintillation coun...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2RB75Z5PubMed
TargetHistamine receptor H3(Macaca mulatta (Rhesus macaque))
Sanofi US

Curated by ChEMBL
LigandPNGBDBM50434382(CHEMBL2387309)copy SMILEScopy InChI
Affinity DataKi:  3.40nMAssay Description:Displacement of [3H]N-alpha-methylhistamine from cloned rhesus monkey histamine H3 receptor transfected in CHO cells after 1 hr by scintillation coun...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2RB75Z5PubMed
TargetHistamine receptor H3(Macaca mulatta (Rhesus macaque))
Sanofi US

Curated by ChEMBL
LigandPNGBDBM50434401(CHEMBL2387314)copy SMILEScopy InChI
Affinity DataKi:  4.10nMAssay Description:Displacement of [3H]N-alpha-methylhistamine from cloned rhesus monkey histamine H3 receptor transfected in CHO cells after 1 hr by scintillation coun...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2RB75Z5PubMed
TargetHistamine receptor H3(Macaca mulatta (Rhesus macaque))
Sanofi US

Curated by ChEMBL
LigandPNGBDBM50434400(CHEMBL2387315)copy SMILEScopy InChI
Affinity DataKi:  4.60nMAssay Description:Displacement of [3H]N-alpha-methylhistamine from cloned rhesus monkey histamine H3 receptor transfected in CHO cells after 1 hr by scintillation coun...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2RB75Z5PubMed
TargetHistamine receptor H3(Macaca mulatta (Rhesus macaque))
Sanofi US

Curated by ChEMBL
LigandPNGBDBM50434392(CHEMBL2387285)copy SMILEScopy InChI
Affinity DataKi:  6nMAssay Description:Displacement of [3H]N-alpha-methylhistamine from cloned rhesus monkey histamine H3 receptor transfected in CHO cells after 1 hr by scintillation coun...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2RB75Z5PubMed
TargetHistamine receptor H3(Macaca mulatta (Rhesus macaque))
Sanofi US

Curated by ChEMBL
LigandPNGBDBM50434387(CHEMBL2387290)copy SMILEScopy InChI
Affinity DataKi:  7.10nMAssay Description:Displacement of [3H]N-alpha-methylhistamine from cloned rhesus monkey histamine H3 receptor transfected in CHO cells after 1 hr by scintillation coun...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2RB75Z5PubMed
TargetHistamine receptor H3(Macaca mulatta (Rhesus macaque))
Sanofi US

Curated by ChEMBL
LigandPNGBDBM50434388(CHEMBL2387289)copy SMILEScopy InChI
Affinity DataKi:  8.40nMAssay Description:Displacement of [3H]N-alpha-methylhistamine from cloned rhesus monkey histamine H3 receptor transfected in CHO cells after 1 hr by scintillation coun...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2RB75Z5PubMed
TargetHistamine receptor H3(Macaca mulatta (Rhesus macaque))
Sanofi US

Curated by ChEMBL
LigandPNGBDBM50434399(CHEMBL2387316)copy SMILEScopy InChI
Affinity DataKi:  11nMAssay Description:Displacement of [3H]N-alpha-methylhistamine from cloned rhesus monkey histamine H3 receptor transfected in CHO cells after 1 hr by scintillation coun...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2RB75Z5PubMed
TargetHistamine receptor H3(Macaca mulatta (Rhesus macaque))
Sanofi US

Curated by ChEMBL
LigandPNGBDBM50434397(CHEMBL2387318)copy SMILEScopy InChI
Affinity DataKi:  11nMAssay Description:Displacement of [3H]N-alpha-methylhistamine from cloned rhesus monkey histamine H3 receptor transfected in CHO cells after 1 hr by scintillation coun...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2RB75Z5PubMed
TargetHistamine receptor H3(Macaca mulatta (Rhesus macaque))
Sanofi US

Curated by ChEMBL
LigandPNGBDBM50434393(CHEMBL2387284)copy SMILEScopy InChI
Affinity DataKi:  11nMAssay Description:Displacement of [3H]N-alpha-methylhistamine from cloned rhesus monkey histamine H3 receptor transfected in CHO cells after 1 hr by scintillation coun...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2RB75Z5PubMed
TargetHistamine receptor H3(Macaca mulatta (Rhesus macaque))
Sanofi US

Curated by ChEMBL
LigandPNGBDBM50434396(CHEMBL2387319)copy SMILEScopy InChI
Affinity DataKi:  13nMAssay Description:Displacement of [3H]N-alpha-methylhistamine from cloned rhesus monkey histamine H3 receptor transfected in CHO cells after 1 hr by scintillation coun...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2RB75Z5PubMed
TargetHistamine receptor H3(Macaca mulatta (Rhesus macaque))
Sanofi US

Curated by ChEMBL
LigandPNGBDBM50434381(CHEMBL2387310)copy SMILEScopy InChI
Affinity DataKi:  16nMAssay Description:Displacement of [3H]N-alpha-methylhistamine from cloned rhesus monkey histamine H3 receptor transfected in CHO cells after 1 hr by scintillation coun...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2RB75Z5PubMed
TargetHistamine H3 receptor(Rattus norvegicus (rat))
Sanofi US

Curated by ChEMBL
LigandPNGBDBM50435303(CHEMBL2391167)copy SMILEScopy InChI
Affinity DataKi:  17nMAssay Description:Displacement of [3H]N-alpha-methylhistamine from rat histamine H3 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HH6MGFPubMed
TargetHistamine receptor H3(Macaca mulatta (Rhesus macaque))
Sanofi US

Curated by ChEMBL
LigandPNGBDBM50434383(CHEMBL2387307)copy SMILEScopy InChI
Affinity DataKi:  18nMAssay Description:Displacement of [3H]N-alpha-methylhistamine from cloned rhesus monkey histamine H3 receptor transfected in CHO cells after 1 hr by scintillation coun...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2RB75Z5PubMed
TargetHistamine receptor H3(Macaca mulatta (Rhesus macaque))
Sanofi US

Curated by ChEMBL
LigandPNGBDBM50434404(CHEMBL2387311)copy SMILEScopy InChI
Affinity DataKi:  19nMAssay Description:Displacement of [3H]N-alpha-methylhistamine from cloned rhesus monkey histamine H3 receptor transfected in CHO cells after 1 hr by scintillation coun...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2RB75Z5PubMed
TargetHistamine receptor H3(Macaca mulatta (Rhesus macaque))
Sanofi US

Curated by ChEMBL
LigandPNGBDBM50434403(CHEMBL2387312)copy SMILEScopy InChI
Affinity DataKi:  22nMAssay Description:Displacement of [3H]N-alpha-methylhistamine from cloned rhesus monkey histamine H3 receptor transfected in CHO cells after 1 hr by scintillation coun...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2RB75Z5PubMed
TargetHistamine receptor H3(Macaca mulatta (Rhesus macaque))
Sanofi US

Curated by ChEMBL
LigandPNGBDBM50434394(CHEMBL2387283)copy SMILEScopy InChI
Affinity DataKi:  23nMAssay Description:Displacement of [3H]N-alpha-methylhistamine from cloned rhesus monkey histamine H3 receptor transfected in CHO cells after 1 hr by scintillation coun...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2RB75Z5PubMed
TargetHistamine receptor H3(Macaca mulatta (Rhesus macaque))
Sanofi US

Curated by ChEMBL
LigandPNGBDBM50434398(CHEMBL2387317)copy SMILEScopy InChI
Affinity DataKi:  26nMAssay Description:Displacement of [3H]N-alpha-methylhistamine from cloned rhesus monkey histamine H3 receptor transfected in CHO cells after 1 hr by scintillation coun...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2RB75Z5PubMed
TargetHistamine receptor H3(Macaca mulatta (Rhesus macaque))
Sanofi US

Curated by ChEMBL
LigandPNGBDBM50434386(CHEMBL2387291)copy SMILEScopy InChI
Affinity DataKi:  29nMAssay Description:Displacement of [3H]N-alpha-methylhistamine from cloned rhesus monkey histamine H3 receptor transfected in CHO cells after 1 hr by scintillation coun...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2RB75Z5PubMed
TargetHistamine H3 receptor(Rattus norvegicus (rat))
Sanofi US

Curated by ChEMBL
LigandPNGBDBM50434382(CHEMBL2387309)copy SMILEScopy InChI
Affinity DataKi:  33nMAssay Description:Displacement of [3H]N-alpha-methylhistamine from cloned rat histamine H3 receptor transfected in CHO cells after 1 hr by scintillation counting analy...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2RB75Z5PubMed
TargetHistamine receptor H3(Macaca mulatta (Rhesus macaque))
Sanofi US

Curated by ChEMBL
LigandPNGBDBM50434395(CHEMBL2387282)copy SMILEScopy InChI
Affinity DataKi:  34nMAssay Description:Displacement of [3H]N-alpha-methylhistamine from cloned rhesus monkey histamine H3 receptor transfected in CHO cells after 1 hr by scintillation coun...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2RB75Z5PubMed
TargetHistamine receptor H3(Macaca mulatta (Rhesus macaque))
Sanofi US

Curated by ChEMBL
LigandPNGBDBM50434391(CHEMBL2387286)copy SMILEScopy InChI
Affinity DataKi:  36nMAssay Description:Displacement of [3H]N-alpha-methylhistamine from cloned rhesus monkey histamine H3 receptor transfected in CHO cells after 1 hr by scintillation coun...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2RB75Z5PubMed
TargetHistamine H3 receptor(Rattus norvegicus (rat))
Sanofi US

Curated by ChEMBL
LigandPNGBDBM50434381(CHEMBL2387310)copy SMILEScopy InChI
Affinity DataKi:  40nMAssay Description:Displacement of [3H]N-alpha-methylhistamine from cloned rat histamine H3 receptor transfected in CHO cells after 1 hr by scintillation counting analy...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2RB75Z5PubMed
TargetHistamine receptor H3(Macaca mulatta (Rhesus macaque))
Sanofi US

Curated by ChEMBL
LigandPNGBDBM50434402(CHEMBL2387313)copy SMILEScopy InChI
Affinity DataKi:  43nMAssay Description:Displacement of [3H]N-alpha-methylhistamine from cloned rhesus monkey histamine H3 receptor transfected in CHO cells after 1 hr by scintillation coun...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2RB75Z5PubMed
TargetHistamine receptor H3(Macaca mulatta (Rhesus macaque))
Sanofi US

Curated by ChEMBL
LigandPNGBDBM50434385(CHEMBL2387292)copy SMILEScopy InChI
Affinity DataKi:  47nMAssay Description:Displacement of [3H]N-alpha-methylhistamine from cloned rhesus monkey histamine H3 receptor transfected in CHO cells after 1 hr by scintillation coun...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2RB75Z5PubMed
TargetHistamine H3 receptor(Rattus norvegicus (rat))
Sanofi US

Curated by ChEMBL
LigandPNGBDBM50435304(CHEMBL2391166)copy SMILEScopy InChI
Affinity DataKi:  55nMAssay Description:Displacement of [3H]N-alpha-methylhistamine from rat histamine H3 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HH6MGFPubMed
TargetHistamine receptor H3(Macaca mulatta (Rhesus macaque))
Sanofi US

Curated by ChEMBL
LigandPNGBDBM50434390(CHEMBL2387287)copy SMILEScopy InChI
Affinity DataKi:  90nMAssay Description:Displacement of [3H]N-alpha-methylhistamine from cloned rhesus monkey histamine H3 receptor transfected in CHO cells after 1 hr by scintillation coun...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2RB75Z5PubMed
TargetHistamine receptor H3(Macaca mulatta (Rhesus macaque))
Sanofi US

Curated by ChEMBL
LigandPNGBDBM50434384(CHEMBL2387293)copy SMILEScopy InChI
Affinity DataKi:  115nMAssay Description:Displacement of [3H]N-alpha-methylhistamine from cloned rhesus monkey histamine H3 receptor transfected in CHO cells after 1 hr by scintillation coun...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2RB75Z5PubMed
TargetHistamine H3 receptor(Rattus norvegicus (rat))
Sanofi US

Curated by ChEMBL
LigandPNGBDBM50434383(CHEMBL2387307)copy SMILEScopy InChI
Affinity DataKi:  135nMAssay Description:Displacement of [3H]N-alpha-methylhistamine from cloned rat histamine H3 receptor transfected in CHO cells after 1 hr by scintillation counting analy...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2RB75Z5PubMed
TargetHistamine H1 receptor(Homo sapiens (Human))
Sanofi US

Curated by ChEMBL
LigandPNGBDBM50435303(CHEMBL2391167)copy SMILEScopy InChI
Affinity DataKi: >9.30E+3nMAssay Description:Binding affinity to human histamine H1 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HH6MGFPubMed
TargetHistamine H1 receptor(Homo sapiens (Human))
Sanofi US

Curated by ChEMBL
LigandPNGBDBM50435304(CHEMBL2391166)copy SMILEScopy InChI
Affinity DataKi: >9.30E+3nMAssay Description:Binding affinity to human histamine H1 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HH6MGFPubMed
TargetGlucagon-like peptide 1 receptor(Homo sapiens (Human))
Sanofi-Aventis Deutschland GmbH

Curated by ChEMBL
LigandPNGBDBM50275569(CHEMBL4130148)copy SMILEScopy InChI
Affinity DataIC50: 26nMAssay Description:Displacement of [125I]GLP-1 from human GLP1R expressed in HEK293 cell membranes after 180 mins by microbeta counting methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NP26XRPubMed
TargetGlucagon-like peptide 1 receptor(Homo sapiens (Human))
Sanofi-Aventis Deutschland GmbH

Curated by ChEMBL
LigandPNGBDBM50275578(CHEMBL4128112)copy SMILEScopy InChI
Affinity DataIC50: 1.13E+3nMAssay Description:Displacement of [125I]GLP-1 from human GLP1R expressed in HEK293 cell membranes after 180 mins by microbeta counting methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NP26XRPubMed
TargetGlucagon-like peptide 1 receptor(Homo sapiens (Human))
Sanofi-Aventis Deutschland GmbH

Curated by ChEMBL
LigandPNGBDBM50275545(CHEMBL4126953)copy SMILEScopy InChI
Affinity DataEC50:  0.00220nMAssay Description:Agonist activity at human GLP1R expressed in HEK293 cells assessed as cAMP accumulation after 30 mins by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NP26XRPubMed
TargetGlucagon-like peptide 1 receptor(Homo sapiens (Human))
Sanofi-Aventis Deutschland GmbH

Curated by ChEMBL
LigandPNGBDBM50275546(CHEMBL4130044)copy SMILEScopy InChI
Affinity DataEC50:  0.0525nMAssay Description:Agonist activity at human GLP1R expressed in HEK293 cells assessed as cAMP accumulation after 30 mins by HTRF assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NP26XRPubMed
TargetGlucagon receptor(Homo sapiens (Human))
Sanofi-Aventis Deutschland GmbH

Curated by ChEMBL
LigandPNGBDBM50275564(CHEMBL4128125)copy SMILEScopy InChI
Affinity DataEC50:  0.000700nMAssay Description:Agonist activity at human glucagon receptor expressed in HEK293 cells assessed as cAMP accumulation after 30 mins by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NP26XRPubMed
TargetGlucagon-like peptide 1 receptor(Homo sapiens (Human))
Sanofi-Aventis Deutschland GmbH

Curated by ChEMBL
LigandPNGBDBM50266693(CHEBI:5391 | Glucagen Hypokit | Glucagon | Glucago...)copy SMILEScopy InChI
Affinity DataEC50:  0.0439nMAssay Description:Agonist activity at human GLP1R expressed in HEK293 cells assessed as cAMP accumulation after 30 mins by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NP26XRPubMed
TargetGlucagon-like peptide 1 receptor(Homo sapiens (Human))
Sanofi-Aventis Deutschland GmbH

Curated by ChEMBL
LigandPNGBDBM50275565(CHEMBL4125912)copy SMILEScopy InChI
Affinity DataEC50:  0.00640nMAssay Description:Agonist activity at human GLP1R expressed in HEK293 cells assessed as cAMP accumulation after 30 mins by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NP26XRPubMed
TargetGlucagon-like peptide 1 receptor(Macaca fascicularis)
Sanofi-Aventis Deutschland GmbH

Curated by ChEMBL
LigandPNGBDBM50275566(CHEMBL4128276)copy SMILEScopy InChI
Affinity DataEC50:  0.00110nMAssay Description:Agonist activity at monkey GLP1R expressed in HEK293 cells assessed as cAMP accumulation after 30 mins by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NP26XRPubMed
TargetGastric inhibitory polypeptide receptor(Homo sapiens (Human))
Sanofi-Aventis Deutschland GmbH

Curated by ChEMBL
LigandPNGBDBM50275567(CHEMBL4128194)copy SMILEScopy InChI
Affinity DataEC50:  0.189nMAssay Description:Agonist activity at human GIP receptor expressed in HEK293 cells assessed as cAMP accumulation after 30 mins by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NP26XRPubMed
TargetGlucagon receptor(Homo sapiens (Human))
Sanofi-Aventis Deutschland GmbH

Curated by ChEMBL
LigandPNGBDBM50275567(CHEMBL4128194)copy SMILEScopy InChI
Affinity DataEC50:  0.00160nMAssay Description:Agonist activity at human glucagon receptor expressed in HEK293 cells assessed as cAMP accumulation after 30 mins by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NP26XRPubMed
TargetGlucagon receptor(Homo sapiens (Human))
Sanofi-Aventis Deutschland GmbH

Curated by ChEMBL
LigandPNGBDBM50275568(CHEMBL4126738)copy SMILEScopy InChI
Affinity DataEC50:  0.0276nMAssay Description:Agonist activity at human glucagon receptor expressed in HEK293 cells assessed as cAMP accumulation after 30 mins by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NP26XRPubMed
TargetGastric inhibitory polypeptide receptor(Homo sapiens (Human))
Sanofi-Aventis Deutschland GmbH

Curated by ChEMBL
LigandPNGBDBM50275569(CHEMBL4130148)copy SMILEScopy InChI
Affinity DataEC50:  114nMAssay Description:Agonist activity at human GIP receptor expressed in HEK293 cells assessed as cAMP accumulation after 30 mins by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NP26XRPubMed
TargetGastric inhibitory polypeptide receptor(Homo sapiens (Human))
Sanofi-Aventis Deutschland GmbH

Curated by ChEMBL
LigandPNGBDBM50275578(CHEMBL4128112)copy SMILEScopy InChI
Affinity DataEC50: >1.00E+5nMAssay Description:Agonist activity at human GIP receptor expressed in HEK293 cells assessed as cAMP accumulation after 30 mins by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NP26XRPubMed
TargetGastric inhibitory polypeptide receptor(Homo sapiens (Human))
Sanofi-Aventis Deutschland GmbH

Curated by ChEMBL
LigandPNGBDBM50275568(CHEMBL4126738)copy SMILEScopy InChI
Affinity DataEC50:  2.03nMAssay Description:Agonist activity at human GIP receptor expressed in HEK293 cells assessed as cAMP accumulation after 30 mins by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NP26XRPubMed
TargetGlucagon-like peptide 1 receptor(Macaca fascicularis)
Sanofi-Aventis Deutschland GmbH

Curated by ChEMBL
LigandPNGBDBM50266693(CHEBI:5391 | Glucagen Hypokit | Glucagon | Glucago...)copy SMILEScopy InChI
Affinity DataEC50:  0.0310nMAssay Description:Agonist activity at monkey GLP1R expressed in HEK293 cells assessed as cAMP accumulation after 30 mins by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NP26XRPubMed
TargetGlucagon-like peptide 1 receptor(Macaca fascicularis)
Sanofi-Aventis Deutschland GmbH

Curated by ChEMBL
LigandPNGBDBM50275565(CHEMBL4125912)copy SMILEScopy InChI
Affinity DataEC50:  0.00410nMAssay Description:Agonist activity at monkey GLP1R expressed in HEK293 cells assessed as cAMP accumulation after 30 mins by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NP26XRPubMed
TargetGlucagon-like peptide 1 receptor(Macaca fascicularis)
Sanofi-Aventis Deutschland GmbH

Curated by ChEMBL
LigandPNGBDBM50275568(CHEMBL4126738)copy SMILEScopy InChI
Affinity DataEC50:  0.00220nMAssay Description:Agonist activity at monkey GLP1R expressed in HEK293 cells assessed as cAMP accumulation after 30 mins by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NP26XRPubMed
TargetGastric inhibitory polypeptide receptor(Homo sapiens (Human))
Sanofi-Aventis Deutschland GmbH

Curated by ChEMBL
LigandPNGBDBM50275546(CHEMBL4130044)copy SMILEScopy InChI
Affinity DataEC50:  177nMAssay Description:Agonist activity at human GIP receptor expressed in HEK293 cells assessed as cAMP accumulation after 30 mins by HTRF assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NP26XRPubMed
Displayed 1 to 50 (of 86 total ) | Next | Last >>
Jump to: