Affinity DataKi: 0.0460nMAssay Description:Binding affinity to pig brain tubulinMore data for this Ligand-Target Pair
Affinity DataKi: 0.0585nMAssay Description:Binding affinity to pig brain tubulinMore data for this Ligand-Target Pair
Affinity DataKi: 0.0637nMAssay Description:Binding affinity to pig brain tubulinMore data for this Ligand-Target Pair
Affinity DataKi: 0.122nMAssay Description:Binding affinity to pig brain tubulinMore data for this Ligand-Target Pair
Affinity DataKi: 0.127nMAssay Description:Binding affinity to pig brain tubulinMore data for this Ligand-Target Pair
Affinity DataKi: 0.131nMAssay Description:Binding affinity to pig brain tubulinMore data for this Ligand-Target Pair
Affinity DataKi: 0.143nMAssay Description:Binding affinity to pig brain tubulinMore data for this Ligand-Target Pair
Affinity DataKi: 0.183nMAssay Description:Binding affinity to pig brain tubulinMore data for this Ligand-Target Pair
Affinity DataKi: 0.198nMAssay Description:Binding affinity to pig brain tubulinMore data for this Ligand-Target Pair
Affinity DataKi: 0.280nMAssay Description:Binding affinity to pig brain tubulinMore data for this Ligand-Target Pair
Affinity DataKi: 0.367nMAssay Description:Binding affinity to pig brain tubulinMore data for this Ligand-Target Pair
Affinity DataKi: 1.60nMAssay Description:Binding affinity to pig brain tubulinMore data for this Ligand-Target Pair
Affinity DataKi: 9.50E+4nMAssay Description:Non-competitive inhibition of human placental insulin receptor expressed in CHO cell membrane assessed as decrease in insulin-stimulated A2 phosphory...More data for this Ligand-Target Pair
Affinity DataIC50: 4nMAssay Description:Inhibition of human recombinant pp60c-src expressed in baculovirus infected Sf9 insect cells using poly(Glu,Tyr) 4:1 as substrate after 15 minsMore data for this Ligand-Target Pair
Affinity DataIC50: 6.5nMAssay Description:Inhibition of human c-SRC expressed in mouse NIH/3T3 cells assessed as inhibition of cell growth in presence of 0.5% FCSMore data for this Ligand-Target Pair
Affinity DataIC50: 13nMAssay Description:Inhibition of human c-SRC expressed in mouse NIH/3T3 cells assessed as inhibition of cell growth in presence of 1.5% FCS by BrdU incorporation assayMore data for this Ligand-Target Pair
Affinity DataIC50: 60nMAssay Description:Inhibition of Src autophosphorylation in mouse GL261 cellsMore data for this Ligand-Target Pair
TargetBreakpoint cluster region protein/Tyrosine-protein kinase ABL1(Homo sapiens (Human))
Athenex Inc.
Curated by ChEMBL
Athenex Inc.
Curated by ChEMBL
Affinity DataIC50: 100nMAssay Description:Inhibition of BCR/ABL (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 100nMAssay Description:Inhibition of LYN (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 110nMAssay Description:Inhibition of human c-SRC expressed in mouse NIH/3T3 cells assessed as reduction in BrdU incorporation after 24 hrs by ELISAMore data for this Ligand-Target Pair
Affinity DataIC50: 118nMAssay Description:Inhibition of human c-SRC expressed in mouse NIH/3T3 cells assessed as inhibition of cell growth in presence of 1.5% FCS by BrdU incorporation assayMore data for this Ligand-Target Pair
Affinity DataIC50: 269nMAssay Description:Inhibition of human c-SRC expressed in mouse NIH/3T3 cells assessed as inhibition of cell growth in presence of 1.5% FCS by BrdU incorporation assayMore data for this Ligand-Target Pair
Affinity DataIC50: 349nMAssay Description:Inhibition of human c-SRC expressed in mouse NIH/3T3 cells assessed as inhibition of cell growth in presence of 1.5% FCS by BrdU incorporation assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.49E+3nMAssay Description:Binding affinity to pig brain tubulin polymerization measured every 1 mins of 60 mins by fluorescence assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.52E+3nMAssay Description:Binding affinity to pig brain tubulin polymerization measured every 1 mins of 60 mins by fluorescence assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.62E+3nMAssay Description:Binding affinity to pig brain tubulin polymerization measured every 1 mins of 60 mins by fluorescence assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.70E+3nMAssay Description:Binding affinity to pig brain tubulin polymerization measured every 1 mins of 60 mins by fluorescence assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.99E+3nMAssay Description:Binding affinity to pig brain tubulin polymerization measured every 1 mins of 60 mins by fluorescence assayMore data for this Ligand-Target Pair
Affinity DataIC50: 2.98E+3nMAssay Description:Binding affinity to pig brain tubulin polymerization measured every 1 mins of 60 mins by fluorescence assayMore data for this Ligand-Target Pair
Affinity DataIC50: 4.60E+3nMAssay Description:Binding affinity to pig brain tubulin polymerization measured every 1 mins of 60 mins by fluorescence assayMore data for this Ligand-Target Pair
Affinity DataIC50: 6.49E+3nMAssay Description:Binding affinity to pig brain tubulin polymerization measured every 1 mins of 60 mins by fluorescence assayMore data for this Ligand-Target Pair
Affinity DataIC50: 7.85E+3nMAssay Description:Binding affinity to pig brain tubulin polymerization measured every 1 mins of 60 mins by fluorescence assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human placental insulin receptor expressed in CHO cells assessed as decrease in insulin-stimulated [3H]-2-deoxyglucose uptake preincuba...More data for this Ligand-Target Pair
Affinity DataIC50: 1.60E+4nMAssay Description:Inhibition of full length human recombinant pp60c-src using RR-SRC as substrateMore data for this Ligand-Target Pair
Affinity DataIC50: 3.80E+4nMAssay Description:Inhibition of full length human recombinant pp60c-src using RR-SRC as substrateMore data for this Ligand-Target Pair
Affinity DataIC50: 6.70E+4nMAssay Description:Inhibition of Src (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 6.70E+4nMAssay Description:Inhibition of Src (unknown origin)More data for this Ligand-Target Pair