Compile Data Set for Download or QSAR
Found 375 with Last Name = 'morita' and Initial = 'y'
TargetCoagulation factor X(Homo sapiens (Human))
Astellas Pharma Inc

Curated by ChEMBL
LigandPNGBDBM50358251(CHEMBL1922344)copy SMILEScopy InChI
Affinity DataKi:  20nMAssay Description:Inhibition of human factor 10A using chromogenic substrate S2222 by dixon plot analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2D50ND9PubMed
TargetCoagulation factor X(Homo sapiens (Human))
Astellas Pharma Inc

Curated by ChEMBL
LigandPNGBDBM50358252(CHEMBL1922235)copy SMILEScopy InChI
Affinity DataKi:  31nMAssay Description:Inhibition of human factor 10A using chromogenic substrate S2222 by dixon plot analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2D50ND9PubMed
TargetProstacyclin receptor(Homo sapiens (Human))
Toray Industries, Inc.

Curated by ChEMBL
LigandPNGBDBM50167257(CHEMBL3798917)copy SMILEScopy InChI
Affinity DataKi:  400nMAssay Description:Binding affinity to human IP receptorMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PV6N9MPubMed
TargetPlasma kallikrein(Homo sapiens (Human))
Astellas Pharma Inc

Curated by ChEMBL
LigandPNGBDBM50358252(CHEMBL1922235)copy SMILEScopy InChI
Affinity DataKi:  1.10E+4nMAssay Description:Inhibition of human plasma kallikrein using chromogenic substrate S2302 by dixon plot analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2D50ND9PubMed
TargetPlasma kallikrein(Homo sapiens (Human))
Astellas Pharma Inc

Curated by ChEMBL
LigandPNGBDBM50358251(CHEMBL1922344)copy SMILEScopy InChI
Affinity DataKi:  1.70E+4nMAssay Description:Inhibition of human plasma kallikrein using chromogenic substrate S2302 by dixon plot analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2D50ND9PubMed
TargetProstaglandin E2 receptor EP3 subtype(Homo sapiens (Human))
Toray Industries, Inc.

Curated by ChEMBL
LigandPNGBDBM50167257(CHEMBL3798917)copy SMILEScopy InChI
Affinity DataKi: >5.00E+4nMAssay Description:Binding affinity to human EP3 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PV6N9MPubMed
TargetProstaglandin E2 receptor EP4 subtype(Homo sapiens (Human))
Toray Industries, Inc.

Curated by ChEMBL
LigandPNGBDBM50167257(CHEMBL3798917)copy SMILEScopy InChI
Affinity DataKi: >5.00E+4nMAssay Description:Binding affinity to human EP4 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PV6N9MPubMed
TargetProstaglandin F2-alpha receptor(Homo sapiens (Human))
Toray Industries, Inc.

Curated by ChEMBL
LigandPNGBDBM50167257(CHEMBL3798917)copy SMILEScopy InChI
Affinity DataKi: >5.00E+4nMAssay Description:Binding affinity to human FP receptorMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PV6N9MPubMed
TargetProstaglandin E2 receptor EP2 subtype(Homo sapiens (Human))
Toray Industries, Inc.

Curated by ChEMBL
LigandPNGBDBM50167257(CHEMBL3798917)copy SMILEScopy InChI
Affinity DataKi: >5.00E+4nMAssay Description:Binding affinity to human EP2 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PV6N9MPubMed
TargetThromboxane A2 receptor(Homo sapiens (Human))
Toray Industries, Inc.

Curated by ChEMBL
LigandPNGBDBM50167257(CHEMBL3798917)copy SMILEScopy InChI
Affinity DataKi: >5.00E+4nMAssay Description:Binding affinity to human TP receptorMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PV6N9MPubMed
TargetProthrombin(Homo sapiens (Human))
Astellas Pharma Inc

Curated by ChEMBL
LigandPNGBDBM50358252(CHEMBL1922235)copy SMILEScopy InChI
Affinity DataKi: >1.00E+5nMAssay Description:Inhibition of human thrombin using chromogenic substrate S2238 by dixon plot analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2D50ND9PubMed
TargetProthrombin(Homo sapiens (Human))
Astellas Pharma Inc

Curated by ChEMBL
LigandPNGBDBM50358251(CHEMBL1922344)copy SMILEScopy InChI
Affinity DataKi: >1.00E+5nMAssay Description:Inhibition of human thrombin using chromogenic substrate S2238 by dixon plot analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2D50ND9PubMed
TargetcGMP-specific 3',5'-cyclic phosphodiesterase(Canis lupus familiaris)
Tanabe Seiyaku Co., Ltd.

Curated by ChEMBL
LigandPNGBDBM50130021(7-(2-Methyl-pyridin-4-ylmethyl)-8-oxo-2-(pyridin-2...)copy SMILEScopy InChI
Affinity DataIC50: 0.220nMAssay Description:Inhibitory activity against phosphodiesterase 5 (PDE5) isolated from canine lungMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2WQ04B2PubMed
TargetcGMP-specific 3',5'-cyclic phosphodiesterase(Canis lupus familiaris)
Tanabe Seiyaku Co., Ltd.

Curated by ChEMBL
LigandPNGBDBM50100673(CHEMBL538498 | methyl 2-(4-aminophenyl)-4-(4-bromo...)copy SMILEScopy InChI
Affinity DataIC50: 0.220nMAssay Description:Inhibitory activity against canine lung Phosphodiesterase 5 (PDE5)More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2QR4XT5PubMed
TargetcGMP-specific 3',5'-cyclic phosphodiesterase(Canis lupus familiaris)
Tanabe Seiyaku Co., Ltd.

Curated by ChEMBL
LigandPNGBDBM50130017(2-(2-Methyl-pyridin-4-ylmethyl)-1-oxo-8-(pyrimidin...)copy SMILEScopy InChI
Affinity DataIC50: 0.230nMAssay Description:Inhibitory activity against phosphodiesterase 5 (PDE5) isolated from canine lungMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2WQ04B2PubMed
TargetcGMP-specific 3',5'-cyclic phosphodiesterase(Canis lupus familiaris)
Tanabe Seiyaku Co., Ltd.

Curated by ChEMBL
LigandPNGBDBM50130025(7-(2-Methyl-pyridin-4-ylmethyl)-8-oxo-2-(pyrazin-2...)copy SMILEScopy InChI
Affinity DataIC50: 0.290nMAssay Description:Inhibitory activity against phosphodiesterase 5 (PDE5) isolated from canine lungMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2WQ04B2PubMed
TargetcGMP-specific 3',5'-cyclic phosphodiesterase(Canis lupus familiaris)
Tanabe Seiyaku Co., Ltd.

Curated by ChEMBL
LigandPNGBDBM50130020(2-(2-Methyl-pyridin-4-ylmethyl)-1-oxo-8-(pyridin-2...)copy SMILEScopy InChI
Affinity DataIC50: 0.310nMAssay Description:Inhibitory activity against phosphodiesterase 5 (PDE5) isolated from canine lungMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2WQ04B2PubMed
TargetcGMP-specific 3',5'-cyclic phosphodiesterase(Canis lupus familiaris)
Tanabe Seiyaku Co., Ltd.

Curated by ChEMBL
LigandPNGBDBM50130027(8-Oxo-2-(pyridin-2-ylmethoxy)-7-pyridin-4-ylmethyl...)copy SMILEScopy InChI
Affinity DataIC50: 0.380nMAssay Description:Inhibitory activity against phosphodiesterase 5 (PDE5) isolated from canine lungMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2WQ04B2PubMed
TargetcGMP-specific 3',5'-cyclic phosphodiesterase(Canis lupus familiaris)
Tanabe Seiyaku Co., Ltd.

Curated by ChEMBL
LigandPNGBDBM50100674(CHEMBL541818 | methyl 2-(4-aminophenyl)-4-(3,5-dim...)copy SMILEScopy InChI
Affinity DataIC50: 0.390nMAssay Description:Inhibitory activity against canine lung Phosphodiesterase 5 (PDE5)More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2QR4XT5PubMed
TargetExtracellular calcium-sensing receptor(Rattus norvegicus)
Mitsubishi Tanabe Pharma Corporation

Curated by ChEMBL
LigandPNGBDBM50272596(CHEMBL4126450)copy SMILEScopy InChI
Affinity DataIC50: 0.470nMAssay Description:Agonist activity at CaSR in rat parathyroid cells assessed as inhibition of PTH (1 to 84 residues) production in presence of Cacl2 by ELISAMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DF6TP0PubMed
TargetcGMP-specific 3',5'-cyclic phosphodiesterase(Canis lupus familiaris)
Tanabe Seiyaku Co., Ltd.

Curated by ChEMBL
LigandPNGBDBM50130028(7-(4-Amino-phenyl)-8-oxo-2-(pyridin-2-ylmethoxy)-5...)copy SMILEScopy InChI
Affinity DataIC50: 0.510nMAssay Description:Inhibitory activity against phosphodiesterase 5 (PDE5) isolated from canine lungMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2WQ04B2PubMed
TargetcGMP-specific 3',5'-cyclic phosphodiesterase(Canis lupus familiaris)
Tanabe Seiyaku Co., Ltd.

Curated by ChEMBL
LigandPNGBDBM50130024(2-(2-Methyl-pyridin-4-ylmethyl)-1-oxo-8-(2-pyridin...)copy SMILEScopy InChI
Affinity DataIC50: 0.520nMAssay Description:Inhibitory activity against phosphodiesterase 5 (PDE5) isolated from canine lungMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2WQ04B2PubMed
TargetExtracellular calcium-sensing receptor(Rattus norvegicus)
Mitsubishi Tanabe Pharma Corporation

Curated by ChEMBL
LigandPNGBDBM50272602(CHEMBL4126877)copy SMILEScopy InChI
Affinity DataIC50: 0.910nMAssay Description:Agonist activity at CaSR in rat parathyroid cells assessed as inhibition of PTH (1 to 84 residues) production in presence of Cacl2 by ELISAMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DF6TP0PubMed
TargetcGMP-specific 3',5'-cyclic phosphodiesterase(Canis lupus familiaris)
Tanabe Seiyaku Co., Ltd.

Curated by ChEMBL
LigandPNGBDBM50100662(CHEMBL553371 | CHEMBL77971 | methyl 2-(4-aminophen...)copy SMILEScopy InChI
Affinity DataIC50: 1nMAssay Description:Inhibitory activity against canine lung Phosphodiesterase 5 (PDE5)More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2QR4XT5PubMed
TargetcGMP-specific 3',5'-cyclic phosphodiesterase(Canis lupus familiaris)
Tanabe Seiyaku Co., Ltd.

Curated by ChEMBL
LigandPNGBDBM50100662(CHEMBL553371 | CHEMBL77971 | methyl 2-(4-aminophen...)copy SMILEScopy InChI
Affinity DataIC50: 1nMAssay Description:Inhibitory activity against phosphodiesterase 5 (PDE5) isolated from canine lungMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2WQ04B2PubMed
TargetcGMP-specific 3',5'-cyclic phosphodiesterase(Canis lupus familiaris)
Tanabe Seiyaku Co., Ltd.

Curated by ChEMBL
LigandPNGBDBM14390(5-[2-ethoxy-5-(4-methyl-1-piperazinylsulfonyl)phen...)copy SMILEScopy InChI
Affinity DataIC50: 1nMAssay Description:Inhibitory activity against phosphodiesterase 5 (PDE5) isolated from canine lungMore data for this Ligand-Target Pair
TargetcGMP-specific 3',5'-cyclic phosphodiesterase(Canis lupus familiaris)
Tanabe Seiyaku Co., Ltd.

Curated by ChEMBL
LigandPNGBDBM50100659(CHEMBL544289 | methyl 2-(4-aminophenyl)-1-oxo-7-(3...)copy SMILEScopy InChI
Affinity DataIC50: 1.10nMAssay Description:Inhibitory activity against canine lung Phosphodiesterase 5 (PDE5)More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2QR4XT5PubMed
TargetcGMP-specific 3',5'-cyclic phosphodiesterase(Canis lupus familiaris)
Tanabe Seiyaku Co., Ltd.

Curated by ChEMBL
LigandPNGBDBM50130029(7-(2-Methyl-pyridin-4-ylmethyl)-8-oxo-2-(2-pyridin...)copy SMILEScopy InChI
Affinity DataIC50: 1.20nMAssay Description:Inhibitory activity against phosphodiesterase 5 (PDE5) isolated from canine lungMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2WQ04B2PubMed
TargetcGMP-specific 3',5'-cyclic phosphodiesterase(Canis lupus familiaris)
Tanabe Seiyaku Co., Ltd.

Curated by ChEMBL
LigandPNGBDBM50100656(2-(4-Amino-phenyl)-7-benzyloxy-1-oxo-4-(3,4,5-trim...)copy SMILEScopy InChI
Affinity DataIC50: 1.20nMAssay Description:Inhibitory activity against canine lung Phosphodiesterase 5 (PDE5)More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2QR4XT5PubMed
TargetAndrogen receptor(Homo sapiens (Human))
National Institute of Health Sciences

Curated by ChEMBL
LigandPNGBDBM50459869(CHEMBL4227715)copy SMILEScopy InChI
Affinity DataIC50: 1.40nMAssay Description:Binding affinity to androgen receptor (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VT1VR7PubMed
TargetExtracellular calcium-sensing receptor(Rattus norvegicus)
Mitsubishi Tanabe Pharma Corporation

Curated by ChEMBL
LigandPNGBDBM50272605(CHEMBL4128542)copy SMILEScopy InChI
Affinity DataIC50: 1.40nMAssay Description:Agonist activity at CaSR in rat parathyroid cells assessed as inhibition of PTH (1 to 84 residues) production in presence of Cacl2 by ELISAMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DF6TP0PubMed
TargetAndrogen receptor(Homo sapiens (Human))
National Institute of Health Sciences

Curated by ChEMBL
LigandPNGBDBM50459874(CHEMBL4226259)copy SMILEScopy InChI
Affinity DataIC50: 1.40nMAssay Description:Binding affinity to androgen receptor (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VT1VR7PubMed
TargetcGMP-specific 3',5'-cyclic phosphodiesterase(Canis lupus familiaris)
Tanabe Seiyaku Co., Ltd.

Curated by ChEMBL
LigandPNGBDBM50366818(CHEMBL1202833)copy SMILEScopy InChI
Affinity DataIC50: 1.80nMAssay Description:Inhibitory activity against phosphodiesterase 5 (PDE5) isolated from canine lungMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2WQ04B2PubMed
TargetcGMP-specific 3',5'-cyclic phosphodiesterase(Canis lupus familiaris)
Tanabe Seiyaku Co., Ltd.

Curated by ChEMBL
LigandPNGBDBM50130026(7-(2-Methyl-pyridin-4-ylmethyl)-8-oxo-2-(pyrimidin...)copy SMILEScopy InChI
Affinity DataIC50: 1.90nMAssay Description:Inhibitory activity against phosphodiesterase 5 (PDE5) isolated from canine lungMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2WQ04B2PubMed
TargetExtracellular calcium-sensing receptor(Rattus norvegicus)
Mitsubishi Tanabe Pharma Corporation

Curated by ChEMBL
LigandPNGBDBM50272606(CHEMBL4125917)copy SMILEScopy InChI
Affinity DataIC50: 2.10nMAssay Description:Agonist activity at CaSR in rat parathyroid cells assessed as inhibition of PTH (1 to 84 residues) production in presence of Cacl2 by ELISAMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DF6TP0PubMed
TargetcGMP-specific 3',5'-cyclic phosphodiesterase(Canis lupus familiaris)
Tanabe Seiyaku Co., Ltd.

Curated by ChEMBL
LigandPNGBDBM50130019(8-Oxo-2-(pyridin-2-ylmethoxy)-7-pyridin-3-ylmethyl...)copy SMILEScopy InChI
Affinity DataIC50: 2.30nMAssay Description:Inhibitory activity against phosphodiesterase 5 (PDE5) isolated from canine lungMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2WQ04B2PubMed
TargetcGMP-specific 3',5'-cyclic phosphodiesterase(Canis lupus familiaris)
Tanabe Seiyaku Co., Ltd.

Curated by ChEMBL
LigandPNGBDBM50130016(8-(2-Hydroxy-ethylamino)-2-(2-methyl-pyridin-4-ylm...)copy SMILEScopy InChI
Affinity DataIC50: 2.60nMAssay Description:Inhibitory activity against phosphodiesterase 5 (PDE5) isolated from canine lungMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2WQ04B2PubMed
TargetcGMP-specific 3',5'-cyclic phosphodiesterase(Canis lupus familiaris)
Tanabe Seiyaku Co., Ltd.

Curated by ChEMBL
LigandPNGBDBM50100670(CHEMBL553786 | methyl 2-(4-aminophenyl)-1-oxo-7-(4...)copy SMILEScopy InChI
Affinity DataIC50: 3.10nMAssay Description:Inhibitory activity against canine lung Phosphodiesterase 5 (PDE5)More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2QR4XT5PubMed
TargetcGMP-specific 3',5'-cyclic phosphodiesterase(Canis lupus familiaris)
Tanabe Seiyaku Co., Ltd.

Curated by ChEMBL
LigandPNGBDBM14390(5-[2-ethoxy-5-(4-methyl-1-piperazinylsulfonyl)phen...)copy SMILEScopy InChI
Affinity DataIC50: 3.90nMAssay Description:Inhibitory activity against canine lung Phosphodiesterase 5 (PDE5)More data for this Ligand-Target Pair
TargetExtracellular calcium-sensing receptor(Rattus norvegicus)
Mitsubishi Tanabe Pharma Corporation

Curated by ChEMBL
LigandPNGBDBM50272607(CHEMBL4126057)copy SMILEScopy InChI
Affinity DataIC50: 4.30nMAssay Description:Agonist activity at CaSR in rat parathyroid cells assessed as inhibition of PTH (1 to 84 residues) production in presence of Cacl2 by ELISAMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DF6TP0PubMed
TargetP04972/P11541/P16586/P22571/P23439/Q95142(Bos taurus)
Tanabe Seiyaku Co., Ltd.

Curated by ChEMBL
LigandPNGBDBM50130020(2-(2-Methyl-pyridin-4-ylmethyl)-1-oxo-8-(pyridin-2...)copy SMILEScopy InChI
Affinity DataIC50: 4.40nMAssay Description:Inhibitory activity against Phosphodiesterase 6 isolated from bovine retinaMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2WQ04B2PubMed
TargetcGMP-specific 3',5'-cyclic phosphodiesterase(Canis lupus familiaris)
Tanabe Seiyaku Co., Ltd.

Curated by ChEMBL
LigandPNGBDBM50100664(2-(4-Amino-phenyl)-1-oxo-7-(2-pyridin-2-yl-ethoxy)...)copy SMILEScopy InChI
Affinity DataIC50: 5nMAssay Description:Inhibitory activity against canine lung Phosphodiesterase 5 (PDE5)More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2QR4XT5PubMed
TargetP04972/P11541/P16586/P22571/P23439/Q95142(Bos taurus)
Tanabe Seiyaku Co., Ltd.

Curated by ChEMBL
LigandPNGBDBM50130025(7-(2-Methyl-pyridin-4-ylmethyl)-8-oxo-2-(pyrazin-2...)copy SMILEScopy InChI
Affinity DataIC50: 7.70nMAssay Description:Inhibitory activity against Phosphodiesterase 6 isolated from bovine retinaMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2WQ04B2PubMed
TargetExtracellular calcium-sensing receptor(Rattus norvegicus)
Mitsubishi Tanabe Pharma Corporation

Curated by ChEMBL
LigandPNGBDBM50272604(CHEMBL4129011)copy SMILEScopy InChI
Affinity DataIC50: 7.80nMAssay Description:Agonist activity at CaSR in rat parathyroid cells assessed as inhibition of PTH (1 to 84 residues) production in presence of Cacl2 by ELISAMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DF6TP0PubMed
TargetExtracellular calcium-sensing receptor(Rattus norvegicus)
Mitsubishi Tanabe Pharma Corporation

Curated by ChEMBL
LigandPNGBDBM50261663(CHEMBL4079960)copy SMILEScopy InChI
Affinity DataIC50: 8nMAssay Description:Agonist activity at CaSR in rat parathyroid cells assessed as inhibition of PTH (1 to 84 residues) production in presence of Cacl2 by ELISAMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DF6TP0PubMed
TargetCoagulation factor X(Homo sapiens (Human))
Astellas Pharma Inc

Curated by ChEMBL
LigandPNGBDBM50209900(3-(({7-[amino(imino)methyl]-2-naphthyl}methyl)-{1-...)copy SMILEScopy InChI
Affinity DataIC50: 8.10nMAssay Description:Inhibition of human factor 10aMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27H1J90PubMed
TargetcGMP-specific 3',5'-cyclic phosphodiesterase(Canis lupus familiaris)
Tanabe Seiyaku Co., Ltd.

Curated by ChEMBL
LigandPNGBDBM50100663(CHEMBL542878 | methyl 2-(4-aminophenyl)-4-(3-hydro...)copy SMILEScopy InChI
Affinity DataIC50: 8.5nMAssay Description:Inhibitory activity against canine lung Phosphodiesterase 5 (PDE5)More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2QR4XT5PubMed
TargetP04972/P11541/P16586/P22571/P23439/Q95142(Bos taurus)
Tanabe Seiyaku Co., Ltd.

Curated by ChEMBL
LigandPNGBDBM50130021(7-(2-Methyl-pyridin-4-ylmethyl)-8-oxo-2-(pyridin-2...)copy SMILEScopy InChI
Affinity DataIC50: 8.60nMAssay Description:Inhibitory activity against Phosphodiesterase 6 isolated from bovine retinaMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2WQ04B2PubMed
TargetExtracellular calcium-sensing receptor(Rattus norvegicus)
Mitsubishi Tanabe Pharma Corporation

Curated by ChEMBL
LigandPNGBDBM50272608(CHEMBL4125688)copy SMILEScopy InChI
Affinity DataIC50: 9.70nMAssay Description:Agonist activity at CaSR in rat parathyroid cells assessed as inhibition of PTH (1 to 84 residues) production in presence of Cacl2 by ELISAMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DF6TP0PubMed
TargetCoagulation factor X(Homo sapiens (Human))
Astellas Pharma Inc

Curated by ChEMBL
LigandPNGBDBM50209891(CHEMBL390266 | [(((E)-3-{3-[amino(imino)methyl]phe...)copy SMILEScopy InChI
Affinity DataIC50: 10nMAssay Description:Inhibition of human factor 10aMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27H1J90PubMed
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