Compile Data Set for Download or QSAR
Found 72 Enz. Inhib. hit(s) with Target = 'Bromodomain-containing protein 9 [134-239]'
TargetBromodomain-containing protein 9 [134-239](Homo sapiens (Human))
GENENTECH, INC.; CONSTELLATION PHARMACEUTICALS, INC.

US Patent
LigandPNGBDBM321411(6-[(E)-but-2-enyl]-4-[3-methoxy-4-(morpholine-4-ca...)copy SMILEScopy InChI
Affinity DataIC50: 3nMAssay Description:His/Flag epitope tagged BRD9134-239 was cloned, expressed, and purified to homogeneity. BRD9 binding and inhibition was assessed by monitoring the en...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2125VRQUS Patent
TargetBromodomain-containing protein 9 [134-239](Homo sapiens (Human))
GENENTECH, INC.; CONSTELLATION PHARMACEUTICALS, INC.

US Patent
LigandPNGBDBM321429((E)-1-(4-(6-(but-2-en-1-yl)-2-methyl-7-oxo-6,7-dih...)copy SMILEScopy InChI
Affinity DataIC50: 3nMAssay Description:His/Flag epitope tagged BRD9134-239 was cloned, expressed, and purified to homogeneity. BRD9 binding and inhibition was assessed by monitoring the en...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2125VRQUS Patent
TargetBromodomain-containing protein 9 [134-239](Homo sapiens (Human))
GENENTECH, INC.; CONSTELLATION PHARMACEUTICALS, INC.

US Patent
LigandPNGBDBM321430(6-[(E)-but-2-enyl]-4-[3-isopropoxy-4-(morpholine-4...)copy SMILEScopy InChI
Affinity DataIC50: 3nMAssay Description:His/Flag epitope tagged BRD9134-239 was cloned, expressed, and purified to homogeneity. BRD9 binding and inhibition was assessed by monitoring the en...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2125VRQUS Patent
TargetBromodomain-containing protein 9 [134-239](Homo sapiens (Human))
GENENTECH, INC.; CONSTELLATION PHARMACEUTICALS, INC.

US Patent
LigandPNGBDBM321438(3-[6-[(E)-but-2-enyl]-2-methyl-7-oxo-1H-pyrrolo[2,...)copy SMILEScopy InChI
Affinity DataIC50: 3nMAssay Description:His/Flag epitope tagged BRD9134-239 was cloned, expressed, and purified to homogeneity. BRD9 binding and inhibition was assessed by monitoring the en...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2125VRQUS Patent
TargetBromodomain-containing protein 9 [134-239](Homo sapiens (Human))
GENENTECH, INC.; CONSTELLATION PHARMACEUTICALS, INC.

US Patent
LigandPNGBDBM321424(6-[(E)-but-2-enyl]-4-[2,5-dimethoxy-4-(morpholine-...)copy SMILEScopy InChI
Affinity DataIC50: 4nMAssay Description:His/Flag epitope tagged BRD9134-239 was cloned, expressed, and purified to homogeneity. BRD9 binding and inhibition was assessed by monitoring the en...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2125VRQUS Patent
TargetBromodomain-containing protein 9 [134-239](Homo sapiens (Human))
GENENTECH, INC.; CONSTELLATION PHARMACEUTICALS, INC.

US Patent
LigandPNGBDBM321432((E)-6-(but-2-en-1-yl)-4-(3-chloro-4-(piperazine-1-...)copy SMILEScopy InChI
Affinity DataIC50: 4nMAssay Description:His/Flag epitope tagged BRD9134-239 was cloned, expressed, and purified to homogeneity. BRD9 binding and inhibition was assessed by monitoring the en...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2125VRQUS Patent
TargetBromodomain-containing protein 9 [134-239](Homo sapiens (Human))
GENENTECH, INC.; CONSTELLATION PHARMACEUTICALS, INC.

US Patent
LigandPNGBDBM321433((E)-4-(4-(3-(3-amino-1H-pyrazol-1-yl)azetidine-1-c...)copy SMILEScopy InChI
Affinity DataIC50: 5nMAssay Description:His/Flag epitope tagged BRD9134-239 was cloned, expressed, and purified to homogeneity. BRD9 binding and inhibition was assessed by monitoring the en...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2125VRQUS Patent
TargetBromodomain-containing protein 9 [134-239](Homo sapiens (Human))
GENENTECH, INC.; CONSTELLATION PHARMACEUTICALS, INC.

US Patent
LigandPNGBDBM321412(6-[(E)-but-2-enyl]-4-[3-chloro-4-(morpholine-4-car...)copy SMILEScopy InChI
Affinity DataIC50: 5nMAssay Description:His/Flag epitope tagged BRD9134-239 was cloned, expressed, and purified to homogeneity. BRD9 binding and inhibition was assessed by monitoring the en...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2125VRQUS Patent
TargetBromodomain-containing protein 9 [134-239](Homo sapiens (Human))
GENENTECH, INC.; CONSTELLATION PHARMACEUTICALS, INC.

US Patent
LigandPNGBDBM321431(6-[(E)-but-2-enyl]-4-[3-(cyclopropylmethoxy)-4-(mo...)copy SMILEScopy InChI
Affinity DataIC50: 5nMAssay Description:His/Flag epitope tagged BRD9134-239 was cloned, expressed, and purified to homogeneity. BRD9 binding and inhibition was assessed by monitoring the en...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2125VRQUS Patent
TargetBromodomain-containing protein 9 [134-239](Homo sapiens (Human))
GENENTECH, INC.; CONSTELLATION PHARMACEUTICALS, INC.

US Patent
LigandPNGBDBM321425(3-[6-[(E)-but-2-enyl]-2-methyl-7-oxo-1H-pyrrolo[2,...)copy SMILEScopy InChI
Affinity DataIC50: 6nMAssay Description:His/Flag epitope tagged BRD9134-239 was cloned, expressed, and purified to homogeneity. BRD9 binding and inhibition was assessed by monitoring the en...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2125VRQUS Patent
TargetBromodomain-containing protein 9 [134-239](Homo sapiens (Human))
GENENTECH, INC.; CONSTELLATION PHARMACEUTICALS, INC.

US Patent
LigandPNGBDBM321422(5-[6-[(E)-but-2-enyl]-2-methyl-7-oxo-1H-pyrrolo[2,...)copy SMILEScopy InChI
Affinity DataIC50: 6nMAssay Description:His/Flag epitope tagged BRD9134-239 was cloned, expressed, and purified to homogeneity. BRD9 binding and inhibition was assessed by monitoring the en...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2125VRQUS Patent
TargetBromodomain-containing protein 9 [134-239](Homo sapiens (Human))
GENENTECH, INC.; CONSTELLATION PHARMACEUTICALS, INC.

US Patent
LigandPNGBDBM321437((E)-6-(but-2-en-1-yl)-4-(4-(2-hydroxypropan-2-yl)-...)copy SMILEScopy InChI
Affinity DataIC50: 6nMAssay Description:His/Flag epitope tagged BRD9134-239 was cloned, expressed, and purified to homogeneity. BRD9 binding and inhibition was assessed by monitoring the en...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2125VRQUS Patent
TargetBromodomain-containing protein 9 [134-239](Homo sapiens (Human))
GENENTECH, INC.; CONSTELLATION PHARMACEUTICALS, INC.

US Patent
LigandPNGBDBM321428(1-[4-[6-[(E)-but-2-enyl]-2-methyl-7-oxo-1H-pyrrolo...)copy SMILEScopy InChI
Affinity DataIC50: 8nMAssay Description:His/Flag epitope tagged BRD9134-239 was cloned, expressed, and purified to homogeneity. BRD9 binding and inhibition was assessed by monitoring the en...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2125VRQUS Patent
TargetBromodomain-containing protein 9 [134-239](Homo sapiens (Human))
GENENTECH, INC.; CONSTELLATION PHARMACEUTICALS, INC.

US Patent
LigandPNGBDBM321436(4-[4-[3-(3-aminopyrazol-1-yl)azetidine-1-carbonyl]...)copy SMILEScopy InChI
Affinity DataIC50: 9nMAssay Description:His/Flag epitope tagged BRD9134-239 was cloned, expressed, and purified to homogeneity. BRD9 binding and inhibition was assessed by monitoring the en...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2125VRQUS Patent
TargetBromodomain-containing protein 9 [134-239](Homo sapiens (Human))
GENENTECH, INC.; CONSTELLATION PHARMACEUTICALS, INC.

US Patent
LigandPNGBDBM321418(6-allyl-4-[2,5-dimethoxy-4-(morpholine-4-carbonyl)...)copy SMILEScopy InChI
Affinity DataIC50: 9nMAssay Description:His/Flag epitope tagged BRD9134-239 was cloned, expressed, and purified to homogeneity. BRD9 binding and inhibition was assessed by monitoring the en...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2125VRQUS Patent
TargetBromodomain-containing protein 9 [134-239](Homo sapiens (Human))
GENENTECH, INC.; CONSTELLATION PHARMACEUTICALS, INC.

US Patent
LigandPNGBDBM321414(6-[(E)-but-2-enyl]-4-[3-chloro-4-(4-methylpiperazi...)copy SMILEScopy InChI
Affinity DataIC50: 9nMAssay Description:His/Flag epitope tagged BRD9134-239 was cloned, expressed, and purified to homogeneity. BRD9 binding and inhibition was assessed by monitoring the en...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2125VRQUS Patent
TargetBromodomain-containing protein 9 [134-239](Homo sapiens (Human))
GENENTECH, INC.; CONSTELLATION PHARMACEUTICALS, INC.

US Patent
LigandPNGBDBM321409(6-[(E)-but-2-enyl]-4-[3-chloro-4-(pyrrolidine-1-ca...)copy SMILEScopy InChI
Affinity DataIC50: 10nMAssay Description:His/Flag epitope tagged BRD9134-239 was cloned, expressed, and purified to homogeneity. BRD9 binding and inhibition was assessed by monitoring the en...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2125VRQUS Patent
TargetBromodomain-containing protein 9 [134-239](Homo sapiens (Human))
GENENTECH, INC.; CONSTELLATION PHARMACEUTICALS, INC.

US Patent
LigandPNGBDBM321415(6-[(E)-but-2-enyl]-2-methyl-4-[3-methyl-4-(morphol...)copy SMILEScopy InChI
Affinity DataIC50: 11nMAssay Description:His/Flag epitope tagged BRD9134-239 was cloned, expressed, and purified to homogeneity. BRD9 binding and inhibition was assessed by monitoring the en...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2125VRQUS Patent
TargetBromodomain-containing protein 9 [134-239](Homo sapiens (Human))
GENENTECH, INC.; CONSTELLATION PHARMACEUTICALS, INC.

US Patent
LigandPNGBDBM321417(6-allyl-4-[3-chloro-4-(morpholine-4-carbonyl)pheny...)copy SMILEScopy InChI
Affinity DataIC50: 12nMAssay Description:His/Flag epitope tagged BRD9134-239 was cloned, expressed, and purified to homogeneity. BRD9 binding and inhibition was assessed by monitoring the en...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2125VRQUS Patent
TargetBromodomain-containing protein 9 [134-239](Homo sapiens (Human))
GENENTECH, INC.; CONSTELLATION PHARMACEUTICALS, INC.

US Patent
LigandPNGBDBM321407(6-[(E)-but-2-enyl]-2-methyl-4-[4-(morpholine-4-car...)copy SMILEScopy InChI
Affinity DataIC50: 13nMAssay Description:His/Flag epitope tagged BRD9134-239 was cloned, expressed, and purified to homogeneity. BRD9 binding and inhibition was assessed by monitoring the en...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2125VRQUS Patent
TargetBromodomain-containing protein 9 [134-239](Homo sapiens (Human))
GENENTECH, INC.; CONSTELLATION PHARMACEUTICALS, INC.

US Patent
LigandPNGBDBM321408(6-[(E)-but-2-enyl]-2-methyl-4-[4-(pyrrolidine-1-ca...)copy SMILEScopy InChI
Affinity DataIC50: 13nMAssay Description:His/Flag epitope tagged BRD9134-239 was cloned, expressed, and purified to homogeneity. BRD9 binding and inhibition was assessed by monitoring the en...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2125VRQUS Patent
TargetBromodomain-containing protein 9 [134-239](Homo sapiens (Human))
GENENTECH, INC.; CONSTELLATION PHARMACEUTICALS, INC.

US Patent
LigandPNGBDBM321389(6-[(E)-but-2-enyl]-4-[3-chloro-4-(morpholine-4-car...)copy SMILEScopy InChI
Affinity DataIC50: 13nMAssay Description:His/Flag epitope tagged BRD9134-239 was cloned, expressed, and purified to homogeneity. BRD9 binding and inhibition was assessed by monitoring the en...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2125VRQUS Patent
TargetBromodomain-containing protein 9 [134-239](Homo sapiens (Human))
GENENTECH, INC.; CONSTELLATION PHARMACEUTICALS, INC.

US Patent
LigandPNGBDBM321383(6-but-2-enyl-4-[4-(morpholine-4-carbonyl)phenyl]-1...)copy SMILEScopy InChI
Affinity DataIC50: 13nMAssay Description:His/Flag epitope tagged BRD9134-239 was cloned, expressed, and purified to homogeneity. BRD9 binding and inhibition was assessed by monitoring the en...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2125VRQUS Patent
TargetBromodomain-containing protein 9 [134-239](Homo sapiens (Human))
GENENTECH, INC.; CONSTELLATION PHARMACEUTICALS, INC.

US Patent
LigandPNGBDBM321402(6-[(E)-but-2-enyl]-4-[4-(1-hydroxy-1-methyl-ethyl)...)copy SMILEScopy InChI
Affinity DataIC50: 17nMAssay Description:His/Flag epitope tagged BRD9134-239 was cloned, expressed, and purified to homogeneity. BRD9 binding and inhibition was assessed by monitoring the en...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2125VRQUS Patent
TargetBromodomain-containing protein 9 [134-239](Homo sapiens (Human))
GENENTECH, INC.; CONSTELLATION PHARMACEUTICALS, INC.

US Patent
LigandPNGBDBM321439(6-butyl-4-[2,5-dimethoxy-4-(morpholine-4-carbonyl)...)copy SMILEScopy InChI
Affinity DataIC50: 17nMAssay Description:His/Flag epitope tagged BRD9134-239 was cloned, expressed, and purified to homogeneity. BRD9 binding and inhibition was assessed by monitoring the en...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2125VRQUS Patent
TargetBromodomain-containing protein 9 [134-239](Homo sapiens (Human))
GENENTECH, INC.; CONSTELLATION PHARMACEUTICALS, INC.

US Patent
LigandPNGBDBM321400(6-[(E)-but-2-enyl]-4-[4-(1-hydroxy-1-methyl-ethyl)...)copy SMILEScopy InChI
Affinity DataIC50: 20nMAssay Description:His/Flag epitope tagged BRD9134-239 was cloned, expressed, and purified to homogeneity. BRD9 binding and inhibition was assessed by monitoring the en...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2125VRQUS Patent
TargetBromodomain-containing protein 9 [134-239](Homo sapiens (Human))
GENENTECH, INC.; CONSTELLATION PHARMACEUTICALS, INC.

US Patent
LigandPNGBDBM310899(4-[4-(1-hydroxy-1-methyl-ethyl)phenyl]-6-methyl-1H...)copy SMILEScopy InChI
Affinity DataIC50: 21nMAssay Description:His/Flag epitope tagged BRD9134-239 was cloned, expressed, and purified to homogeneity. BRD9 binding and inhibition was assessed by monitoring the en...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2V98B5WUS Patent
TargetBromodomain-containing protein 9 [134-239](Homo sapiens (Human))
GENENTECH, INC.; CONSTELLATION PHARMACEUTICALS, INC.

US Patent
LigandPNGBDBM321381(N-[4-(6-but-2-enyl-7-oxo-1H-pyrrolo[2,3-c]pyridin-...)copy SMILEScopy InChI
Affinity DataIC50: 22nMAssay Description:His/Flag epitope tagged BRD9134-239 was cloned, expressed, and purified to homogeneity. BRD9 binding and inhibition was assessed by monitoring the en...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2125VRQUS Patent
TargetBromodomain-containing protein 9 [134-239](Homo sapiens (Human))
GENENTECH, INC.; CONSTELLATION PHARMACEUTICALS, INC.

US Patent
LigandPNGBDBM321420(6-[(E)-but-2-enyl]-4-[4-chloro-5-(morpholine-4-car...)copy SMILEScopy InChI
Affinity DataIC50: 22nMAssay Description:His/Flag epitope tagged BRD9134-239 was cloned, expressed, and purified to homogeneity. BRD9 binding and inhibition was assessed by monitoring the en...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2125VRQUS Patent
TargetBromodomain-containing protein 9 [134-239](Homo sapiens (Human))
GENENTECH, INC.; CONSTELLATION PHARMACEUTICALS, INC.

US Patent
LigandPNGBDBM321396(3-[6-[(E)-but-2-enyl]-7-oxo-1H-pyrrolo[2,3-c]pyrid...)copy SMILEScopy InChI
Affinity DataIC50: 23nMAssay Description:His/Flag epitope tagged BRD9134-239 was cloned, expressed, and purified to homogeneity. BRD9 binding and inhibition was assessed by monitoring the en...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2125VRQUS Patent
TargetBromodomain-containing protein 9 [134-239](Homo sapiens (Human))
GENENTECH, INC.; CONSTELLATION PHARMACEUTICALS, INC.

US Patent
LigandPNGBDBM310892(N-(2-methoxyethyl)-4-(6-methyl-7-oxo-1H-pyrrolo[2,...)copy SMILEScopy InChI
Affinity DataIC50: 24nMAssay Description:His/Flag epitope tagged BRD9134-239 was cloned, expressed, and purified to homogeneity. BRD9 binding and inhibition was assessed by monitoring the en...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2V98B5WUS Patent
TargetBromodomain-containing protein 9 [134-239](Homo sapiens (Human))
GENENTECH, INC.; CONSTELLATION PHARMACEUTICALS, INC.

US Patent
LigandPNGBDBM310896(7-(6-methyl-7-oxo-1H-pyrrolo[2,3-c]pyridin-4-yl)-1...)copy SMILEScopy InChI
Affinity DataIC50: 25nMAssay Description:His/Flag epitope tagged BRD9134-239 was cloned, expressed, and purified to homogeneity. BRD9 binding and inhibition was assessed by monitoring the en...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2V98B5WUS Patent
TargetBromodomain-containing protein 9 [134-239](Homo sapiens (Human))
GENENTECH, INC.; CONSTELLATION PHARMACEUTICALS, INC.

US Patent
LigandPNGBDBM321398(3-[6-[(E)-but-2-enyl]-7-oxo-1H-pyrrolo[2,3-c]pyrid...)copy SMILEScopy InChI
Affinity DataIC50: 27nMAssay Description:His/Flag epitope tagged BRD9134-239 was cloned, expressed, and purified to homogeneity. BRD9 binding and inhibition was assessed by monitoring the en...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2125VRQUS Patent
TargetBromodomain-containing protein 9 [134-239](Homo sapiens (Human))
GENENTECH, INC.; CONSTELLATION PHARMACEUTICALS, INC.

US Patent
LigandPNGBDBM321392(3-[6-[(E)-but-2-enyl]-7-oxo-1H-pyrrolo[2,3-c]pyrid...)copy SMILEScopy InChI
Affinity DataIC50: 28nMAssay Description:His/Flag epitope tagged BRD9134-239 was cloned, expressed, and purified to homogeneity. BRD9 binding and inhibition was assessed by monitoring the en...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2125VRQUS Patent
TargetBromodomain-containing protein 9 [134-239](Homo sapiens (Human))
GENENTECH, INC.; CONSTELLATION PHARMACEUTICALS, INC.

US Patent
LigandPNGBDBM321395(3-[6-[(E)-but-2-enyl]-7-oxo-1H-pyrrolo[2,3-c]pyrid...)copy SMILEScopy InChI
Affinity DataIC50: 28nMAssay Description:His/Flag epitope tagged BRD9134-239 was cloned, expressed, and purified to homogeneity. BRD9 binding and inhibition was assessed by monitoring the en...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2125VRQUS Patent
TargetBromodomain-containing protein 9 [134-239](Homo sapiens (Human))
GENENTECH, INC.; CONSTELLATION PHARMACEUTICALS, INC.

US Patent
LigandPNGBDBM321377(4-(6-but-2-enyl-7-oxo-1H-pyrrolo[2,3-c]pyridin-4-y...)copy SMILEScopy InChI
Affinity DataIC50: 29nMAssay Description:His/Flag epitope tagged BRD9134-239 was cloned, expressed, and purified to homogeneity. BRD9 binding and inhibition was assessed by monitoring the en...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2125VRQUS Patent
TargetBromodomain-containing protein 9 [134-239](Homo sapiens (Human))
GENENTECH, INC.; CONSTELLATION PHARMACEUTICALS, INC.

US Patent
LigandPNGBDBM310895(3-methyl-7-(6-methyl-7-oxo-1H-pyrrolo[2,3-c]pyridi...)copy SMILES
Affinity DataIC50: 31nMAssay Description:His/Flag epitope tagged BRD9134-239 was cloned, expressed, and purified to homogeneity. BRD9 binding and inhibition was assessed by monitoring the en...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2V98B5WUS Patent
TargetBromodomain-containing protein 9 [134-239](Homo sapiens (Human))
GENENTECH, INC.; CONSTELLATION PHARMACEUTICALS, INC.

US Patent
LigandPNGBDBM321413(6-[(E)-but-2-enyl]-4-[5-chloro-6-(morpholine-4-car...)copy SMILEScopy InChI
Affinity DataIC50: 32nMAssay Description:His/Flag epitope tagged BRD9134-239 was cloned, expressed, and purified to homogeneity. BRD9 binding and inhibition was assessed by monitoring the en...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2125VRQUS Patent
TargetBromodomain-containing protein 9 [134-239](Homo sapiens (Human))
GENENTECH, INC.; CONSTELLATION PHARMACEUTICALS, INC.

US Patent
LigandPNGBDBM321410(6-[(E)-but-2-enyl]-4-[2,3-difluoro-4-(morpholine-4...)copy SMILEScopy InChI
Affinity DataIC50: 34nMAssay Description:His/Flag epitope tagged BRD9134-239 was cloned, expressed, and purified to homogeneity. BRD9 binding and inhibition was assessed by monitoring the en...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2125VRQUS Patent
TargetBromodomain-containing protein 9 [134-239](Homo sapiens (Human))
GENENTECH, INC.; CONSTELLATION PHARMACEUTICALS, INC.

US Patent
LigandPNGBDBM321397(3-[6-[(E)-but-2-enyl]-7-oxo-1H-pyrrolo[2,3-c]pyrid...)copy SMILEScopy InChI
Affinity DataIC50: 35nMAssay Description:His/Flag epitope tagged BRD9134-239 was cloned, expressed, and purified to homogeneity. BRD9 binding and inhibition was assessed by monitoring the en...More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2125VRQUS Patent
TargetBromodomain-containing protein 9 [134-239](Homo sapiens (Human))
GENENTECH, INC.; CONSTELLATION PHARMACEUTICALS, INC.

US Patent
LigandPNGBDBM321393(3-[6-[(E)-but-2-enyl]-7-oxo-1H-pyrrolo[2,3-c]pyrid...)copy SMILEScopy InChI
Affinity DataIC50: 35nMAssay Description:His/Flag epitope tagged BRD9134-239 was cloned, expressed, and purified to homogeneity. BRD9 binding and inhibition was assessed by monitoring the en...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2125VRQUS Patent
TargetBromodomain-containing protein 9 [134-239](Homo sapiens (Human))
GENENTECH, INC.; CONSTELLATION PHARMACEUTICALS, INC.

US Patent
LigandPNGBDBM321394(6-[(E)-but-2-enyl]-4-[2-methoxy-5-(pyrrolidine-1-c...)copy SMILEScopy InChI
Affinity DataIC50: 39nMAssay Description:His/Flag epitope tagged BRD9134-239 was cloned, expressed, and purified to homogeneity. BRD9 binding and inhibition was assessed by monitoring the en...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2125VRQUS Patent
TargetBromodomain-containing protein 9 [134-239](Homo sapiens (Human))
GENENTECH, INC.; CONSTELLATION PHARMACEUTICALS, INC.

US Patent
LigandPNGBDBM321378(6-but-2-enyl-4-[3-(pyrrolidine-1-carbonyl)phenyl]-...)copy SMILEScopy InChI
Affinity DataIC50: 39nMAssay Description:His/Flag epitope tagged BRD9134-239 was cloned, expressed, and purified to homogeneity. BRD9 binding and inhibition was assessed by monitoring the en...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2125VRQUS Patent
TargetBromodomain-containing protein 9 [134-239](Homo sapiens (Human))
GENENTECH, INC.; CONSTELLATION PHARMACEUTICALS, INC.

US Patent
LigandPNGBDBM321426(6-but-2-enyl-4-[3-methoxy-5-(4-methylpiperazine-1-...)copy SMILEScopy InChI
Affinity DataIC50: 39nMAssay Description:His/Flag epitope tagged BRD9134-239 was cloned, expressed, and purified to homogeneity. BRD9 binding and inhibition was assessed by monitoring the en...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2125VRQUS Patent
TargetBromodomain-containing protein 9 [134-239](Homo sapiens (Human))
GENENTECH, INC.; CONSTELLATION PHARMACEUTICALS, INC.

US Patent
LigandPNGBDBM321403(6-butyl-4-(4-(2-hydroxypropan-2-yl)phenyl)-1H-pyrr...)copy SMILEScopy InChI
Affinity DataIC50: 43nMAssay Description:His/Flag epitope tagged BRD9134-239 was cloned, expressed, and purified to homogeneity. BRD9 binding and inhibition was assessed by monitoring the en...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2125VRQUS Patent
TargetBromodomain-containing protein 9 [134-239](Homo sapiens (Human))
GENENTECH, INC.; CONSTELLATION PHARMACEUTICALS, INC.

US Patent
LigandPNGBDBM321388(3-(6-butyl-7-oxo-1H-pyrrolo[2,3-c]pyridin-4-yl)-4-...)copy SMILEScopy InChI
Affinity DataIC50: 46nMAssay Description:His/Flag epitope tagged BRD9134-239 was cloned, expressed, and purified to homogeneity. BRD9 binding and inhibition was assessed by monitoring the en...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2125VRQUS Patent
TargetBromodomain-containing protein 9 [134-239](Homo sapiens (Human))
GENENTECH, INC.; CONSTELLATION PHARMACEUTICALS, INC.

US Patent
LigandPNGBDBM321390(6-[(E)-but-2-enyl]-4-[3-chloro-4-(pyrrolidine-1-ca...)copy SMILEScopy InChI
Affinity DataIC50: 46nMAssay Description:His/Flag epitope tagged BRD9134-239 was cloned, expressed, and purified to homogeneity. BRD9 binding and inhibition was assessed by monitoring the en...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2125VRQUS Patent
TargetBromodomain-containing protein 9 [134-239](Homo sapiens (Human))
GENENTECH, INC.; CONSTELLATION PHARMACEUTICALS, INC.

US Patent
LigandPNGBDBM321419(6-[(E)-but-2-enyl]-4-[3-methoxy-5-(morpholine-4-ca...)copy SMILEScopy InChI
Affinity DataIC50: 46nMAssay Description:His/Flag epitope tagged BRD9134-239 was cloned, expressed, and purified to homogeneity. BRD9 binding and inhibition was assessed by monitoring the en...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2125VRQUS Patent
TargetBromodomain-containing protein 9 [134-239](Homo sapiens (Human))
GENENTECH, INC.; CONSTELLATION PHARMACEUTICALS, INC.

US Patent
LigandPNGBDBM310898(N,N-dimethyl-3-(6-methyl-7-oxo-1H-pyrrolo[2,3-c]py...)copy SMILEScopy InChI
Affinity DataIC50: 53nMAssay Description:His/Flag epitope tagged BRD9134-239 was cloned, expressed, and purified to homogeneity. BRD9 binding and inhibition was assessed by monitoring the en...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetBromodomain-containing protein 9 [134-239](Homo sapiens (Human))
GENENTECH, INC.; CONSTELLATION PHARMACEUTICALS, INC.

US Patent
LigandPNGBDBM310902(6-methyl-4-[4-(1-methyl-4-piperidyl)phenyl]-1H-pyr...)copy SMILEScopy InChI
Affinity DataIC50: 53nMAssay Description:His/Flag epitope tagged BRD9134-239 was cloned, expressed, and purified to homogeneity. BRD9 binding and inhibition was assessed by monitoring the en...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2V98B5WUS Patent
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