Found 1 Enz. Inhib. hit(s) with Target = 'Bromodomain-containing protein 9 [134-239]' and Ligand = 'BDBM310898' TargetBromodomain-containing protein 9 [134-239](Homo sapiens (Human))
Genentech, Inc.; Constellation Pharmaceuticals Inc.
US Patent
Genentech, Inc.; Constellation Pharmaceuticals Inc.
US Patent
Affinity DataIC50: 53nMAssay Description:His/Flag epitope tagged BRD9134-239 was cloned, expressed, and purified to homogeneity. BRD9 binding and inhibition was assessed by monitoring the en...More data for this Ligand-Target Pair
3D Structure (crystal)