Compile Data Set for Download or QSAR
Found 7 Enz. Inhib. hit(s) with Target = 'Cytohesin-2'
TargetCytohesin-2(Homo sapiens (Human))
UMR 5247

Curated by ChEMBL
LigandPNGBDBM50441975(CHEMBL2440216)copy SMILEScopy InChI
Affinity DataKi:  5.40E+5nMAssay Description:Inhibition of human Arno Sec7 domain-mediated nucleotide exchange in delta17 Arf1 (17 to 181) by BODIPY-GTP based time resolved fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2251KMFPubMed
TargetCytohesin-2(Homo sapiens (Human))
UMR 5247

Curated by ChEMBL
LigandPNGBDBM50441972(CHEMBL2440207)copy SMILEScopy InChI
Affinity DataKi:  9.80E+5nMAssay Description:Inhibition of human Arno Sec7 domain-mediated nucleotide exchange in delta17 Arf1 (17 to 181) by BODIPY-GTP based time resolved fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2251KMFPubMed
TargetCytohesin-2(Homo sapiens (Human))
UMR 5247

Curated by ChEMBL
LigandPNGBDBM50441973(CHEMBL2440218)copy SMILEScopy InChI
Affinity DataKi:  1.61E+6nMAssay Description:Inhibition of human Arno Sec7 domain-mediated nucleotide exchange in delta17 Arf1 (17 to 181) by BODIPY-GTP based time resolved fluorescence assayMore data for this Ligand-Target Pair
TargetCytohesin-2(Homo sapiens (Human))
UMR 5247

Curated by ChEMBL
LigandPNGBDBM50441976(CHEMBL2440213)copy SMILEScopy InChI
Affinity DataKi:  1.91E+6nMAssay Description:Inhibition of human Arno Sec7 domain-mediated nucleotide exchange in delta17 Arf1 (17 to 181) by BODIPY-GTP based time resolved fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2251KMFPubMed
TargetCytohesin-2(Homo sapiens (Human))
UMR 5247

Curated by ChEMBL
LigandPNGBDBM50441977(CHEMBL2440208)copy SMILEScopy InChI
Affinity DataKi:  3.72E+6nMAssay Description:Inhibition of human Arno Sec7 domain-mediated nucleotide exchange in delta17 Arf1 (17 to 181) by BODIPY-GTP based time resolved fluorescence assayMore data for this Ligand-Target Pair
TargetCytohesin-2(Homo sapiens (Human))
UMR 5247

Curated by ChEMBL
LigandPNGBDBM50441974(CHEMBL236358)copy SMILEScopy InChI
Affinity DataKi:  5.12E+6nMAssay Description:Inhibition of human Arno Sec7 domain-mediated nucleotide exchange in delta17 Arf1 (17 to 181) by BODIPY-GTP based time resolved fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2251KMFPubMed
TargetCytohesin-2(Homo sapiens (Human))
UMR 5247

Curated by ChEMBL
LigandPNGBDBM50441977(CHEMBL2440208)copy SMILEScopy InChI
Affinity DataKd:  5.00E+5nMAssay Description:Binding affinity to human Arno Sec7 domain immobilized on CAP sensor chip after 15 mins by 1H 1D-NMR-700 MHz spectra analysisMore data for this Ligand-Target Pair