Compile Data Set for Download or QSAR
Found 134 Enz. Inhib. hit(s) with Target = 'Phosphatidylinositol 3-kinase C2 domain-containing subunit gamma'
LigandPNGBDBM50193031(CHEMBL3959351 | US11155556, No. 12)copy SMILEScopy InChI
Affinity DataIC50: 2nMAssay Description:The enzymatic activities against PI3K-α, PI3K-β, PI3K-γ and PI3K-δ were tested in ADAPTA assays. Activity against AURKB and AURKB...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q20868G7US Patent
LigandPNGBDBM50193014(CHEMBL3942643 | US11155556, No. 9)copy SMILEScopy InChI
Affinity DataIC50: 2nMAssay Description:The enzymatic activities against PI3K-α, PI3K-β, PI3K-γ and PI3K-δ were tested in ADAPTA assays. Activity against AURKB and AURKB...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q20868G7US Patent
LigandPNGBDBM50193032(CHEMBL3979343 | US11155556, No. 2)copy SMILEScopy InChI
Affinity DataIC50: 2nMAssay Description:The enzymatic activities against PI3K-α, PI3K-β, PI3K-γ and PI3K-δ were tested in ADAPTA assays. Activity against AURKB and AURKB...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q20868G7US Patent
LigandPNGBDBM50193017(CHEMBL3904942 | US11155556, No. 17)copy SMILEScopy InChI
Affinity DataIC50: 4nMAssay Description:The enzymatic activities against PI3K-α, PI3K-β, PI3K-γ and PI3K-δ were tested in ADAPTA assays. Activity against AURKB and AURKB...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q20868G7US Patent
LigandPNGBDBM50193016(CHEMBL3889977 | US11155556, No. 3)copy SMILEScopy InChI
Affinity DataIC50: 20nMAssay Description:The enzymatic activities against PI3K-α, PI3K-β, PI3K-γ and PI3K-δ were tested in ADAPTA assays. Activity against AURKB and AURKB...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q20868G7US Patent
LigandPNGBDBM50193023(CHEMBL3898901 | US11155556, No. 5)copy SMILEScopy InChI
Affinity DataIC50: 29.3nMAssay Description:The enzymatic activities against PI3K-α, PI3K-β, PI3K-γ and PI3K-δ were tested in ADAPTA assays. Activity against AURKB and AURKB...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q20868G7US Patent
LigandPNGBDBM50193030(CHEMBL3950648 | US11155556, No. 14)copy SMILEScopy InChI
Affinity DataIC50: 30nMAssay Description:The enzymatic activities against PI3K-α, PI3K-β, PI3K-γ and PI3K-δ were tested in ADAPTA assays. Activity against AURKB and AURKB...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q20868G7US Patent
LigandPNGBDBM50193020(CHEMBL3907932 | US11155556, No. 7)copy SMILEScopy InChI
Affinity DataIC50: 39nMAssay Description:The enzymatic activities against PI3K-α, PI3K-β, PI3K-γ and PI3K-δ were tested in ADAPTA assays. Activity against AURKB and AURKB...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q20868G7US Patent
LigandPNGBDBM50193021(CHEMBL3922919 | US11155556, No. 13)copy SMILEScopy InChI
Affinity DataIC50: 41nMAssay Description:The enzymatic activities against PI3K-α, PI3K-β, PI3K-γ and PI3K-δ were tested in ADAPTA assays. Activity against AURKB and AURKB...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q20868G7US Patent
LigandPNGBDBM50337135(4-((5,11-dimethyl-6-oxo-6,11-dihydro-5H-benzo[e]py...)copy SMILEScopy InChI
Affinity DataIC50: 49nMAssay Description:The enzymatic activities against PI3K-α, PI3K-β, PI3K-γ and PI3K-δ were tested in ADAPTA assays. Activity against AURKB and AURKB...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q20868G7US Patent
LigandPNGBDBM50193018(CHEMBL3986648 | US11155556, No. 10)copy SMILEScopy InChI
Affinity DataIC50: 50.7nMAssay Description:The enzymatic activities against PI3K-α, PI3K-β, PI3K-γ and PI3K-δ were tested in ADAPTA assays. Activity against AURKB and AURKB...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q20868G7US Patent
LigandPNGBDBM50512861(CHEMBL4558527)copy SMILEScopy InChI
Affinity DataIC50: 63nMAssay Description:Inhibition of PIK3C2G (unknown origin) assessed as reduction in substrate phosphorylation by FRET Adapta assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24Q7ZVJPubMed
LigandPNGBDBM50193029(CHEMBL3913941 | US11155556, No. 15)copy SMILEScopy InChI
Affinity DataIC50: 75.9nMAssay Description:The enzymatic activities against PI3K-α, PI3K-β, PI3K-γ and PI3K-δ were tested in ADAPTA assays. Activity against AURKB and AURKB...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q20868G7US Patent
LigandPNGBDBM50193012(CHEMBL3926951 | US11155556, No. 6)copy SMILEScopy InChI
Affinity DataIC50: 96nMAssay Description:The enzymatic activities against PI3K-α, PI3K-β, PI3K-γ and PI3K-δ were tested in ADAPTA assays. Activity against AURKB and AURKB...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q20868G7US Patent
LigandPNGBDBM50193015(CHEMBL3918001 | US11155556, No. 4)copy SMILEScopy InChI
Affinity DataIC50: 123nMAssay Description:The enzymatic activities against PI3K-α, PI3K-β, PI3K-γ and PI3K-δ were tested in ADAPTA assays. Activity against AURKB and AURKB...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q20868G7US Patent
LigandPNGBDBM50193032(CHEMBL3979343 | US11155556, No. 2)copy SMILEScopy InChI
Affinity DataIC50: 231nMAssay Description:The enzymatic activities against PI3K-α, PI3K-β, PI3K-γ and PI3K-δ were tested in ADAPTA assays. Activity against AURKB and AURKB...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q20868G7US Patent
LigandPNGBDBM50048418(CHEMBL3360227)copy SMILEScopy InChI
Affinity DataIC50: 340nMAssay Description:Inhibition of human GDT-fused recombinant PI3K-C2gamma assessed as residual activity by nonradiometric ADP-Glo assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HM5B2DPubMed
LigandPNGBDBM50193027(CHEMBL3935895 | US11155556, No. 8)copy SMILEScopy InChI
Affinity DataIC50: 438nMAssay Description:The enzymatic activities against PI3K-α, PI3K-β, PI3K-γ and PI3K-δ were tested in ADAPTA assays. Activity against AURKB and AURKB...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q20868G7US Patent
LigandPNGBDBM50193025(CHEMBL3932938 | US11155556, No. 18)copy SMILEScopy InChI
Affinity DataIC50: 822nMAssay Description:The enzymatic activities against PI3K-α, PI3K-β, PI3K-γ and PI3K-δ were tested in ADAPTA assays. Activity against AURKB and AURKB...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q20868G7US Patent
LigandPNGBDBM50160075(CHEMBL3786230)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of N-terminal GST-tagged recombinant human full length PI3KC2gamma expressed in baculovirus infected Sf21 insect cells preincubated for 15...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29888W5PubMed
LigandPNGBDBM513328(US11091472, Compound S-1)copy SMILES
Affinity DataIC50: 1.00E+3nMAssay Description:In some embodiments, the subject compounds inhibit a P14-kinase, as determined by a kinase activity assay, e.g., by an assay that determines the leve...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2RF5Z5NUS Patent
LigandPNGBDBM50160074(CHEMBL3785311)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of N-terminal GST-tagged recombinant human full length PI3KC2gamma expressed in baculovirus infected Sf21 insect cells preincubated for 15...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29888W5PubMed
LigandPNGBDBM50193026(CHEMBL3948672 | US11155556, No. 11)copy SMILEScopy InChI
Affinity DataIC50: 2.61E+3nMAssay Description:The enzymatic activities against PI3K-α, PI3K-β, PI3K-γ and PI3K-δ were tested in ADAPTA assays. Activity against AURKB and AURKB...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q20868G7US Patent
LigandPNGBDBM50274638(CHEMBL4126156 | US10858355, Example 4)copy SMILEScopy InChI
Affinity DataIC50: 3.16E+3nMAssay Description:Inhibition of PI3KC2gamma (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27M0BFZPubMed
LigandPNGBDBM50048416(CHEMBL3360219)copy SMILEScopy InChI
Affinity DataIC50: 3.41E+3nMAssay Description:Inhibition of human GDT-fused recombinant PI3K-C2gamma assessed as residual activity by nonradiometric ADP-Glo assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HM5B2DPubMed
LigandPNGBDBM50048417(CHEMBL3360221)copy SMILEScopy InChI
Affinity DataIC50: 3.61E+3nMAssay Description:Inhibition of human GDT-fused recombinant PI3K-C2gamma assessed as residual activity by nonradiometric ADP-Glo assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HM5B2DPubMed
LigandPNGBDBM60631(BDBM50447096 | US9133168, 19b)copy SMILES
Affinity DataIC50: 3.81E+3nMAssay Description:Inhibition of PI3KC2gamma (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2R212VJPubMed
LigandPNGBDBM513435(US11091472, Compound S-231)copy SMILES
Affinity DataIC50: 5.50E+3nMAssay Description:In some embodiments, the subject compounds inhibit a P14-kinase, as determined by a kinase activity assay, e.g., by an assay that determines the leve...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2RF5Z5NUS Patent
LigandPNGBDBM513442(US11091472, Compound S-261)copy SMILES
Affinity DataIC50: 5.50E+3nMAssay Description:In some embodiments, the subject compounds inhibit a P14-kinase, as determined by a kinase activity assay, e.g., by an assay that determines the leve...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2RF5Z5NUS Patent
LigandPNGBDBM513443(US11091472, Compound S-262)copy SMILES
Affinity DataIC50: 5.50E+3nMAssay Description:In some embodiments, the subject compounds inhibit a P14-kinase, as determined by a kinase activity assay, e.g., by an assay that determines the leve...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2RF5Z5NUS Patent
LigandPNGBDBM513444(US11091472, Compound S-263)copy SMILES
Affinity DataIC50: 5.50E+3nMAssay Description:In some embodiments, the subject compounds inhibit a P14-kinase, as determined by a kinase activity assay, e.g., by an assay that determines the leve...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2RF5Z5NUS Patent
LigandPNGBDBM513389(US11091472, Compound S-160)copy SMILES
Affinity DataIC50: 5.50E+3nMAssay Description:In some embodiments, the subject compounds inhibit a P14-kinase, as determined by a kinase activity assay, e.g., by an assay that determines the leve...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2RF5Z5NUS Patent
LigandPNGBDBM50197067(CHEMBL3913746)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of PI3KC2gamma (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PG1TPXPubMed
LigandPNGBDBM50121212(CHEMBL3622372)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of PI3KC2gamma (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PG1TPXPubMed
LigandPNGBDBM50048419(CHEMBL3360231)copy SMILEScopy InChI
Affinity DataIC50: 2.32E+4nMAssay Description:Inhibition of human GDT-fused recombinant PI3K-C2gamma assessed as residual activity by nonradiometric ADP-Glo assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HM5B2DPubMed
LigandPNGBDBM513422(US11091472, Compound S-215)copy SMILES
Affinity DataIC50: 5.50E+4nMAssay Description:In some embodiments, the subject compounds inhibit a P14-kinase, as determined by a kinase activity assay, e.g., by an assay that determines the leve...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2RF5Z5NUS Patent
LigandPNGBDBM513423(US11091472, Compound S-216)copy SMILES
Affinity DataIC50: 5.50E+4nMAssay Description:In some embodiments, the subject compounds inhibit a P14-kinase, as determined by a kinase activity assay, e.g., by an assay that determines the leve...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2RF5Z5NUS Patent
LigandPNGBDBM513353(US11091472, Compound S-100)copy SMILES
Affinity DataIC50: 5.50E+4nMAssay Description:In some embodiments, the subject compounds inhibit a P14-kinase, as determined by a kinase activity assay, e.g., by an assay that determines the leve...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2RF5Z5NUS Patent
LigandPNGBDBM513445(US11091472, Compound S-265)copy SMILES
Affinity DataIC50: 5.50E+4nMAssay Description:In some embodiments, the subject compounds inhibit a P14-kinase, as determined by a kinase activity assay, e.g., by an assay that determines the leve...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2RF5Z5NUS Patent
LigandPNGBDBM513440(US11091472, Compound S-259)copy SMILES
Affinity DataIC50: 5.50E+4nMAssay Description:In some embodiments, the subject compounds inhibit a P14-kinase, as determined by a kinase activity assay, e.g., by an assay that determines the leve...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2RF5Z5NUS Patent
LigandPNGBDBM513431(US11091472, Compound S-227)copy SMILES
Affinity DataIC50: 5.50E+4nMAssay Description:In some embodiments, the subject compounds inhibit a P14-kinase, as determined by a kinase activity assay, e.g., by an assay that determines the leve...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2RF5Z5NUS Patent
LigandPNGBDBM513439(US11091472, Compound S-258 | US11091472, Compound ...)copy SMILES
Affinity DataIC50: 2.00E+5nMAssay Description:In some embodiments, the subject compounds inhibit a P14-kinase, as determined by a kinase activity assay, e.g., by an assay that determines the leve...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2RF5Z5NUS Patent
LigandPNGBDBM513421(US11091472, Compound S-214)copy SMILES
Affinity DataIC50: 2.00E+5nMAssay Description:In some embodiments, the subject compounds inhibit a P14-kinase, as determined by a kinase activity assay, e.g., by an assay that determines the leve...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2RF5Z5NUS Patent
LigandPNGBDBM513403(US11091472, Compound S-193)copy SMILES
Affinity DataIC50: 2.00E+5nMAssay Description:In some embodiments, the subject compounds inhibit a P14-kinase, as determined by a kinase activity assay, e.g., by an assay that determines the leve...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2RF5Z5NUS Patent
LigandPNGBDBM513395(US11091472, Compound S-170)copy SMILES
Affinity DataIC50: 2.00E+5nMAssay Description:In some embodiments, the subject compounds inhibit a P14-kinase, as determined by a kinase activity assay, e.g., by an assay that determines the leve...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2RF5Z5NUS Patent
LigandPNGBDBM513394(US11091472, Compound S-169)copy SMILES
Affinity DataIC50: 2.00E+5nMAssay Description:In some embodiments, the subject compounds inhibit a P14-kinase, as determined by a kinase activity assay, e.g., by an assay that determines the leve...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2RF5Z5NUS Patent
LigandPNGBDBM513369(US11091472, Compound S-131)copy SMILES
Affinity DataIC50: 2.00E+5nMAssay Description:In some embodiments, the subject compounds inhibit a P14-kinase, as determined by a kinase activity assay, e.g., by an assay that determines the leve...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2RF5Z5NUS Patent
LigandPNGBDBM513368(US11091472, Compound S-129)copy SMILES
Affinity DataIC50: 2.00E+5nMAssay Description:In some embodiments, the subject compounds inhibit a P14-kinase, as determined by a kinase activity assay, e.g., by an assay that determines the leve...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2RF5Z5NUS Patent
LigandPNGBDBM513366(US11091472, Compound S-127)copy SMILES
Affinity DataIC50: 2.00E+5nMAssay Description:In some embodiments, the subject compounds inhibit a P14-kinase, as determined by a kinase activity assay, e.g., by an assay that determines the leve...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2RF5Z5NUS Patent
LigandPNGBDBM513367(US11091472, Compound S-128)copy SMILES
Affinity DataIC50: 2.00E+5nMAssay Description:In some embodiments, the subject compounds inhibit a P14-kinase, as determined by a kinase activity assay, e.g., by an assay that determines the leve...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2RF5Z5NUS Patent
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