Compile Data Set for Download or QSAR
Found 35 Enz. Inhib. hit(s) with Target = 'Segment polarity protein dishevelled homolog DVL-1'
TargetSegment polarity protein dishevelled homolog DVL-1(Homo sapiens (Human))
St. Jude Children's Research Hospital

Curated by ChEMBL
LigandPNGBDBM50373848(CHEMBL255779)copy SMILEScopy InChI
Affinity DataIC50: 4.90E+4nMAssay Description:Antagonist activity at human Dvl1 assessed as inhibition of interaction between Dvl1 PDZ domain and Fz7 PDZ domain by alphaScreen assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25D8SPTPubMed
TargetSegment polarity protein dishevelled homolog DVL-1(Homo sapiens (Human))
St. Jude Children's Research Hospital

Curated by ChEMBL
LigandPNGBDBM50373845(CHEMBL402939)copy SMILEScopy InChI
Affinity DataIC50: 7.80E+4nMAssay Description:Antagonist activity at human Dvl1 assessed as inhibition of interaction between Dvl1 PDZ domain and Fz7 PDZ domain by alphaScreen assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25D8SPTPubMed
TargetSegment polarity protein dishevelled homolog DVL-1(Homo sapiens (Human))
St. Jude Children's Research Hospital

Curated by ChEMBL
LigandPNGBDBM50373844(CHEMBL272948)copy SMILEScopy InChI
Affinity DataIC50: 9.70E+4nMAssay Description:Antagonist activity at human Dvl1 assessed as inhibition of interaction between Dvl1 PDZ domain and Fz7 PDZ domain by alphaScreen assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25D8SPTPubMed
TargetSegment polarity protein dishevelled homolog DVL-1(Homo sapiens (Human))
St. Jude Children's Research Hospital

Curated by ChEMBL
LigandPNGBDBM50373847(CHEMBL256605)copy SMILEScopy InChI
Affinity DataIC50: 1.57E+5nMAssay Description:Antagonist activity at human Dvl1 assessed as inhibition of interaction between Dvl1 PDZ domain and Fz7 PDZ domain by alphaScreen assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25D8SPTPubMed
TargetSegment polarity protein dishevelled homolog DVL-1(Homo sapiens (Human))
St. Jude Children's Research Hospital

Curated by ChEMBL
LigandPNGBDBM50373851(CHEMBL256431)copy SMILEScopy InChI
Affinity DataIC50: 1.59E+5nMAssay Description:Antagonist activity at human Dvl1 assessed as inhibition of interaction between Dvl1 PDZ domain and Fz7 PDZ domain by alphaScreen assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25D8SPTPubMed
TargetSegment polarity protein dishevelled homolog DVL-1(Homo sapiens (Human))
St. Jude Children's Research Hospital

Curated by ChEMBL
LigandPNGBDBM50373846(CHEMBL401537)copy SMILEScopy InChI
Affinity DataIC50: 1.97E+5nMAssay Description:Antagonist activity at human Dvl1 assessed as inhibition of interaction between Dvl1 PDZ domain and Fz7 PDZ domain by alphaScreen assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25D8SPTPubMed
TargetSegment polarity protein dishevelled homolog DVL-1(Homo sapiens (Human))
St. Jude Children's Research Hospital

Curated by ChEMBL
LigandPNGBDBM50373850(CHEMBL404331)copy SMILEScopy InChI
Affinity DataIC50: 5.00E+5nMAssay Description:Antagonist activity at human Dvl1 assessed as inhibition of interaction between Dvl1 PDZ domain and Fz7 PDZ domain by alphaScreen assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25D8SPTPubMed
TargetSegment polarity protein dishevelled homolog DVL-1(Homo sapiens (Human))
St. Jude Children's Research Hospital

Curated by ChEMBL
LigandPNGBDBM50373843(CHEMBL410400)copy SMILEScopy InChI
Affinity DataIC50: 5.00E+5nMAssay Description:Antagonist activity at human Dvl1 assessed as inhibition of interaction between Dvl1 PDZ domain and Fz7 PDZ domain by alphaScreen assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25D8SPTPubMed
TargetSegment polarity protein dishevelled homolog DVL-1(Homo sapiens (Human))
St. Jude Children's Research Hospital

Curated by ChEMBL
LigandPNGBDBM50231890(2-((2-carboxyethyl)carbamoyl)-6-methyl-3-phenethyl...)copy SMILEScopy InChI
Affinity DataIC50: 5.00E+5nMAssay Description:Antagonist activity at human Dvl1 assessed as inhibition of interaction between Dvl1 PDZ domain and Fz7 PDZ domain by alphaScreen assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25D8SPTPubMed
TargetSegment polarity protein dishevelled homolog DVL-1(Homo sapiens (Human))
St. Jude Children's Research Hospital

Curated by ChEMBL
LigandPNGBDBM50373849(CHEMBL255988)copy SMILEScopy InChI
Affinity DataIC50: 5.00E+5nMAssay Description:Antagonist activity at human Dvl1 assessed as inhibition of interaction between Dvl1 PDZ domain and Fz7 PDZ domain by alphaScreen assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25D8SPTPubMed
TargetSegment polarity protein dishevelled homolog DVL-1(Homo sapiens (Human))
St. Jude Children's Research Hospital

Curated by ChEMBL
LigandPNGBDBM50177709(CHEMBL3814864)copy SMILEScopy InChI
Affinity DataKd:  1.30nMAssay Description:Binding affinity to His-tagged Dvl-1 PDZ domain (247 to 337 residues) (unknown origin) expressed in Escherichia coli BL21 (DE3) assessed as dissociat...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2N58P84PubMed
TargetSegment polarity protein dishevelled homolog DVL-1(Homo sapiens (Human))
St. Jude Children's Research Hospital

Curated by ChEMBL
LigandPNGBDBM50177677(CHEMBL3814692)copy SMILEScopy InChI
Affinity DataKd:  5.80nMAssay Description:Binding affinity to His-tagged Dvl-1 PDZ domain (247 to 337 residues) (unknown origin) expressed in Escherichia coli BL21 (DE3) assessed as dissociat...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2N58P84PubMed
TargetSegment polarity protein dishevelled homolog DVL-1(Homo sapiens (Human))
St. Jude Children's Research Hospital

Curated by ChEMBL
LigandPNGBDBM50177714(CHEMBL3813775)copy SMILEScopy InChI
Affinity DataKd:  6.20nMAssay Description:Binding affinity to His-tagged Dvl-1 PDZ domain (247 to 337 residues) (unknown origin) expressed in Escherichia coli BL21 (DE3) assessed as dissociat...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2N58P84PubMed
TargetSegment polarity protein dishevelled homolog DVL-1(Homo sapiens (Human))
St. Jude Children's Research Hospital

Curated by ChEMBL
LigandPNGBDBM50177676(CHEMBL3814041)copy SMILEScopy InChI
Affinity DataKd:  2.5nMAssay Description:Binding affinity to His-tagged Dvl-1 PDZ domain (247 to 337 residues) (unknown origin) expressed in Escherichia coli BL21 (DE3) assessed as dissociat...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2N58P84PubMed
TargetSegment polarity protein dishevelled homolog DVL-1(Homo sapiens (Human))
St. Jude Children's Research Hospital

Curated by ChEMBL
LigandPNGBDBM50177677(CHEMBL3814692)copy SMILEScopy InChI
Affinity DataKd:  1.12E+4nMAssay Description:Binding affinity to His-tagged Dvl-1 PDZ domain (247 to 337 residues) (unknown origin) expressed in Escherichia coli BL21 (DE3) by SPR analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2N58P84PubMed
TargetSegment polarity protein dishevelled homolog DVL-1(Homo sapiens (Human))
St. Jude Children's Research Hospital

Curated by ChEMBL
LigandPNGBDBM50177709(CHEMBL3814864)copy SMILEScopy InChI
Affinity DataKd:  6.84E+4nMAssay Description:Binding affinity to His-tagged Dvl-1 PDZ domain (247 to 337 residues) (unknown origin) expressed in Escherichia coli BL21 (DE3) by SPR analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2N58P84PubMed
TargetSegment polarity protein dishevelled homolog DVL-1(Homo sapiens (Human))
St. Jude Children's Research Hospital

Curated by ChEMBL
LigandPNGBDBM50177708(CHEMBL3814619)copy SMILEScopy InChI
Affinity DataKd:  3.83E+4nMAssay Description:Binding affinity to His-tagged Dvl-1 PDZ domain (247 to 337 residues) (unknown origin) expressed in Escherichia coli BL21 (DE3) by SPR analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2N58P84PubMed
TargetSegment polarity protein dishevelled homolog DVL-1(Homo sapiens (Human))
St. Jude Children's Research Hospital

Curated by ChEMBL
LigandPNGBDBM50177707(CHEMBL3814506)copy SMILEScopy InChI
Affinity DataKd:  1.52E+5nMAssay Description:Binding affinity to His-tagged Dvl-1 PDZ domain (247 to 337 residues) (unknown origin) expressed in Escherichia coli BL21 (DE3) by SPR analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2N58P84PubMed
TargetSegment polarity protein dishevelled homolog DVL-1(Homo sapiens (Human))
St. Jude Children's Research Hospital

Curated by ChEMBL
LigandPNGBDBM50177706(CHEMBL3814441)copy SMILEScopy InChI
Affinity DataKd:  2.51E+5nMAssay Description:Binding affinity to His-tagged Dvl-1 PDZ domain (247 to 337 residues) (unknown origin) expressed in Escherichia coli BL21 (DE3) by SPR analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2N58P84PubMed
TargetSegment polarity protein dishevelled homolog DVL-1(Homo sapiens (Human))
St. Jude Children's Research Hospital

Curated by ChEMBL
LigandPNGBDBM50177705(CHEMBL3815146)copy SMILEScopy InChI
Affinity DataKd:  3.11E+5nMAssay Description:Binding affinity to His-tagged Dvl-1 PDZ domain (247 to 337 residues) (unknown origin) expressed in Escherichia coli BL21 (DE3) by SPR analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2N58P84PubMed
TargetSegment polarity protein dishevelled homolog DVL-1(Homo sapiens (Human))
St. Jude Children's Research Hospital

Curated by ChEMBL
LigandPNGBDBM50177704(CHEMBL3814273)copy SMILEScopy InChI
Affinity DataKd:  1.39E+5nMAssay Description:Binding affinity to His-tagged Dvl-1 PDZ domain (247 to 337 residues) (unknown origin) expressed in Escherichia coli BL21 (DE3) by SPR analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2N58P84PubMed
TargetSegment polarity protein dishevelled homolog DVL-1(Homo sapiens (Human))
St. Jude Children's Research Hospital

Curated by ChEMBL
LigandPNGBDBM50177703(CHEMBL3814879)copy SMILEScopy InChI
Affinity DataKd:  6.24E+4nMAssay Description:Binding affinity to His-tagged Dvl-1 PDZ domain (247 to 337 residues) (unknown origin) expressed in Escherichia coli BL21 (DE3) by SPR analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2N58P84PubMed
TargetSegment polarity protein dishevelled homolog DVL-1(Homo sapiens (Human))
St. Jude Children's Research Hospital

Curated by ChEMBL
LigandPNGBDBM50177714(CHEMBL3813775)copy SMILEScopy InChI
Affinity DataKd:  2.68E+5nMAssay Description:Binding affinity to His-tagged Dvl-1 PDZ domain (247 to 337 residues) (unknown origin) expressed in Escherichia coli BL21 (DE3) by SPR analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2N58P84PubMed
TargetSegment polarity protein dishevelled homolog DVL-1(Homo sapiens (Human))
St. Jude Children's Research Hospital

Curated by ChEMBL
LigandPNGBDBM50177679(CHEMBL3814761)copy SMILEScopy InChI
Affinity DataKd:  9.54E+5nMMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NP28F9PubMed
TargetSegment polarity protein dishevelled homolog DVL-1(Homo sapiens (Human))
St. Jude Children's Research Hospital

Curated by ChEMBL
LigandPNGBDBM50177708(CHEMBL3814619)copy SMILEScopy InChI
Affinity DataKd:  2nMAssay Description:Binding affinity to His-tagged Dvl-1 PDZ domain (247 to 337 residues) (unknown origin) expressed in Escherichia coli BL21 (DE3) assessed as dissociat...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2N58P84PubMed
TargetSegment polarity protein dishevelled homolog DVL-1(Homo sapiens (Human))
St. Jude Children's Research Hospital

Curated by ChEMBL
LigandPNGBDBM50177707(CHEMBL3814506)copy SMILEScopy InChI
Affinity DataKd:  3.80nMAssay Description:Binding affinity to His-tagged Dvl-1 PDZ domain (247 to 337 residues) (unknown origin) expressed in Escherichia coli BL21 (DE3) assessed as dissociat...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2N58P84PubMed
TargetSegment polarity protein dishevelled homolog DVL-1(Homo sapiens (Human))
St. Jude Children's Research Hospital

Curated by ChEMBL
LigandPNGBDBM50177706(CHEMBL3814441)copy SMILEScopy InChI
Affinity DataKd:  1.20nMAssay Description:Binding affinity to His-tagged Dvl-1 PDZ domain (247 to 337 residues) (unknown origin) expressed in Escherichia coli BL21 (DE3) assessed as dissociat...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2N58P84PubMed
TargetSegment polarity protein dishevelled homolog DVL-1(Homo sapiens (Human))
St. Jude Children's Research Hospital

Curated by ChEMBL
LigandPNGBDBM50177705(CHEMBL3815146)copy SMILEScopy InChI
Affinity DataKd:  1.70nMAssay Description:Binding affinity to His-tagged Dvl-1 PDZ domain (247 to 337 residues) (unknown origin) expressed in Escherichia coli BL21 (DE3) assessed as dissociat...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2N58P84PubMed
TargetSegment polarity protein dishevelled homolog DVL-1(Homo sapiens (Human))
St. Jude Children's Research Hospital

Curated by ChEMBL
LigandPNGBDBM50177704(CHEMBL3814273)copy SMILEScopy InChI
Affinity DataKd:  1.5nMAssay Description:Binding affinity to His-tagged Dvl-1 PDZ domain (247 to 337 residues) (unknown origin) expressed in Escherichia coli BL21 (DE3) assessed as dissociat...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2N58P84PubMed
TargetSegment polarity protein dishevelled homolog DVL-1(Homo sapiens (Human))
St. Jude Children's Research Hospital

Curated by ChEMBL
LigandPNGBDBM50177703(CHEMBL3814879)copy SMILEScopy InChI
Affinity DataKd:  3.20nMAssay Description:Binding affinity to His-tagged Dvl-1 PDZ domain (247 to 337 residues) (unknown origin) expressed in Escherichia coli BL21 (DE3) assessed as dissociat...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2N58P84PubMed
TargetSegment polarity protein dishevelled homolog DVL-1(Homo sapiens (Human))
St. Jude Children's Research Hospital

Curated by ChEMBL
LigandPNGBDBM50177679(CHEMBL3814761)copy SMILEScopy InChI
Affinity DataKd:  1.06E+4nMAssay Description:Binding affinity to TMR-labeled Dvl-1 PDZ domain (unknown origin) expressed in Escherichia coli by fluorescence spectroscopyMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2N58P84PubMed
TargetSegment polarity protein dishevelled homolog DVL-1(Mus musculus)
Yonsei University

Curated by ChEMBL
LigandPNGBDBM50177678(CHEMBL3815136)copy SMILEScopy InChI
Affinity DataKd:  2.37E+5nMAssay Description:Binding affinity to TMR-linked 15N-labeled mouse Dvl-1 domain ( 247 to 341 residues) by fluorescence spectroscopyMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2N58P84PubMed
TargetSegment polarity protein dishevelled homolog DVL-1(Homo sapiens (Human))
St. Jude Children's Research Hospital

Curated by ChEMBL
LigandPNGBDBM50601473(CHEMBL5170789)copy SMILES
Affinity DataKd:  3.45E+4nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NP28F9PubMed
TargetSegment polarity protein dishevelled homolog DVL-1(Homo sapiens (Human))
St. Jude Children's Research Hospital

Curated by ChEMBL
LigandPNGBDBM50177676(CHEMBL3814041)copy SMILEScopy InChI
Affinity DataKd:  7.83E+5nMAssay Description:Binding affinity to His-tagged Dvl-1 PDZ domain (247 to 337 residues) (unknown origin) expressed in Escherichia coli BL21 (DE3) by SPR analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2N58P84PubMed
TargetSegment polarity protein dishevelled homolog DVL-1(Homo sapiens (Human))
St. Jude Children's Research Hospital

Curated by ChEMBL
LigandPNGBDBM50177677(CHEMBL3814692)copy SMILEScopy InChI
Affinity DataKd:  186nMAssay Description:Binding affinity to His-tagged Dvl-1 PDZ domain (247 to 337 residues) (unknown origin) expressed in Escherichia coli BL21 (DE3) by fluorescence spect...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2N58P84PubMed