Compile Data Set for Download or QSAR
Found 28 Enz. Inhib. hit(s) with all data for entry = 50045747
TargetMAP kinase-interacting serine/threonine-protein kinase 2(Homo sapiens (Human))
University of South Australia

Curated by ChEMBL
LigandPNGBDBM50079470(CHEMBL3417199)copy SMILEScopy InChI
Affinity DataKi:  240nMAssay Description:Inhibition of Mnk2 (unknown origin) pre-incubated for 10 mins before eIF4E peptide substrate addition by ADP-Glo kinase assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28917K3PubMed
TargetMAP kinase-interacting serine/threonine-protein kinase 2(Homo sapiens (Human))
University of South Australia

Curated by ChEMBL
LigandPNGBDBM50079405(CHEMBL3417205)copy SMILEScopy InChI
Affinity DataKi:  340nMAssay Description:Inhibition of Mnk2 (unknown origin) pre-incubated for 10 mins before eIF4E peptide substrate addition by ADP-Glo kinase assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28917K3PubMed
TargetMAP kinase-interacting serine/threonine-protein kinase 2(Homo sapiens (Human))
University of South Australia

Curated by ChEMBL
LigandPNGBDBM50079471(CHEMBL3417198)copy SMILEScopy InChI
Affinity DataKi:  350nMAssay Description:Inhibition of Mnk2 (unknown origin) pre-incubated for 10 mins before eIF4E peptide substrate addition by ADP-Glo kinase assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28917K3PubMed
TargetMAP kinase-interacting serine/threonine-protein kinase 2(Homo sapiens (Human))
University of South Australia

Curated by ChEMBL
LigandPNGBDBM50298223(CGP-57380 | CHEMBL1240885 | CHEMBL576817 | N-(4-fl...)copy SMILEScopy InChI
Affinity DataKi:  880nMAssay Description:Inhibition of Mnk2 (unknown origin) pre-incubated for 10 mins before eIF4E peptide substrate addition by ADP-Glo kinase assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28917K3PubMed
TargetMAP kinase-interacting serine/threonine-protein kinase 2(Homo sapiens (Human))
University of South Australia

Curated by ChEMBL
LigandPNGBDBM50079403(CHEMBL3417207)copy SMILEScopy InChI
Affinity DataKi:  900nMAssay Description:Inhibition of Mnk2 (unknown origin) pre-incubated for 10 mins before eIF4E peptide substrate addition by ADP-Glo kinase assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28917K3PubMed
TargetMAP kinase-interacting serine/threonine-protein kinase 1(Homo sapiens (Human))
University of South Australia

Curated by ChEMBL
LigandPNGBDBM50298223(CGP-57380 | CHEMBL1240885 | CHEMBL576817 | N-(4-fl...)copy SMILEScopy InChI
Affinity DataKi:  1.01E+3nMAssay Description:Inhibition of Mnk1 (unknown origin) pre-incubated for 10 mins before eIF4E peptide substrate addition by ADP-Glo kinase assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28917K3PubMed
TargetMAP kinase-interacting serine/threonine-protein kinase 2(Homo sapiens (Human))
University of South Australia

Curated by ChEMBL
LigandPNGBDBM50079402(CHEMBL3417208)copy SMILEScopy InChI
Affinity DataKi:  1.60E+3nMAssay Description:Inhibition of Mnk2 (unknown origin) pre-incubated for 10 mins before eIF4E peptide substrate addition by ADP-Glo kinase assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28917K3PubMed
TargetMAP kinase-interacting serine/threonine-protein kinase 1(Homo sapiens (Human))
University of South Australia

Curated by ChEMBL
LigandPNGBDBM50079470(CHEMBL3417199)copy SMILEScopy InChI
Affinity DataKi:  2.06E+3nMAssay Description:Inhibition of Mnk1 (unknown origin) pre-incubated for 10 mins before eIF4E peptide substrate addition by ADP-Glo kinase assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28917K3PubMed
TargetMAP kinase-interacting serine/threonine-protein kinase 1(Homo sapiens (Human))
University of South Australia

Curated by ChEMBL
LigandPNGBDBM50079403(CHEMBL3417207)copy SMILEScopy InChI
Affinity DataKi:  2.15E+3nMAssay Description:Inhibition of Mnk1 (unknown origin) pre-incubated for 10 mins before eIF4E peptide substrate addition by ADP-Glo kinase assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28917K3PubMed
TargetMAP kinase-interacting serine/threonine-protein kinase 1(Homo sapiens (Human))
University of South Australia

Curated by ChEMBL
LigandPNGBDBM50079405(CHEMBL3417205)copy SMILEScopy InChI
Affinity DataKi:  2.33E+3nMAssay Description:Inhibition of Mnk1 (unknown origin) pre-incubated for 10 mins before eIF4E peptide substrate addition by ADP-Glo kinase assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28917K3PubMed
TargetMAP kinase-interacting serine/threonine-protein kinase 2(Homo sapiens (Human))
University of South Australia

Curated by ChEMBL
LigandPNGBDBM50079449(CHEMBL3417204)copy SMILEScopy InChI
Affinity DataKi:  2.63E+3nMAssay Description:Inhibition of Mnk2 (unknown origin) pre-incubated for 10 mins before eIF4E peptide substrate addition by ADP-Glo kinase assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28917K3PubMed
TargetMAP kinase-interacting serine/threonine-protein kinase 2(Homo sapiens (Human))
University of South Australia

Curated by ChEMBL
LigandPNGBDBM50079466(CHEMBL3417203)copy SMILEScopy InChI
Affinity DataKi:  3.17E+3nMAssay Description:Inhibition of Mnk2 (unknown origin) pre-incubated for 10 mins before eIF4E peptide substrate addition by ADP-Glo kinase assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28917K3PubMed
TargetMAP kinase-interacting serine/threonine-protein kinase 1(Homo sapiens (Human))
University of South Australia

Curated by ChEMBL
LigandPNGBDBM50079402(CHEMBL3417208)copy SMILEScopy InChI
Affinity DataKi:  4.51E+3nMAssay Description:Inhibition of Mnk1 (unknown origin) pre-incubated for 10 mins before eIF4E peptide substrate addition by ADP-Glo kinase assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28917K3PubMed
TargetMAP kinase-interacting serine/threonine-protein kinase 1(Homo sapiens (Human))
University of South Australia

Curated by ChEMBL
LigandPNGBDBM50079471(CHEMBL3417198)copy SMILEScopy InChI
Affinity DataKi:  4.82E+3nMAssay Description:Inhibition of Mnk1 (unknown origin) pre-incubated for 10 mins before eIF4E peptide substrate addition by ADP-Glo kinase assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28917K3PubMed
TargetMAP kinase-interacting serine/threonine-protein kinase 1(Homo sapiens (Human))
University of South Australia

Curated by ChEMBL
LigandPNGBDBM50079449(CHEMBL3417204)copy SMILEScopy InChI
Affinity DataKi:  5.00E+3nMAssay Description:Inhibition of Mnk1 (unknown origin) pre-incubated for 10 mins before eIF4E peptide substrate addition by ADP-Glo kinase assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28917K3PubMed
TargetMAP kinase-interacting serine/threonine-protein kinase 1(Homo sapiens (Human))
University of South Australia

Curated by ChEMBL
LigandPNGBDBM50079466(CHEMBL3417203)copy SMILEScopy InChI
Affinity DataKi:  5.40E+3nMAssay Description:Inhibition of Mnk1 (unknown origin) pre-incubated for 10 mins before eIF4E peptide substrate addition by ADP-Glo kinase assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28917K3PubMed
TargetMAP kinase-interacting serine/threonine-protein kinase 2(Homo sapiens (Human))
University of South Australia

Curated by ChEMBL
LigandPNGBDBM50079467(CHEMBL3417202)copy SMILEScopy InChI
Affinity DataKi:  5.99E+3nMAssay Description:Inhibition of Mnk2 (unknown origin) pre-incubated for 10 mins before eIF4E peptide substrate addition by ADP-Glo kinase assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28917K3PubMed
TargetMAP kinase-interacting serine/threonine-protein kinase 2(Homo sapiens (Human))
University of South Australia

Curated by ChEMBL
LigandPNGBDBM50079468(CHEMBL3417201)copy SMILEScopy InChI
Affinity DataKi:  9.05E+3nMAssay Description:Inhibition of Mnk2 (unknown origin) pre-incubated for 10 mins before eIF4E peptide substrate addition by ADP-Glo kinase assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28917K3PubMed
TargetMAP kinase-interacting serine/threonine-protein kinase 1(Homo sapiens (Human))
University of South Australia

Curated by ChEMBL
LigandPNGBDBM50079472(CHEMBL3417197)copy SMILEScopy InChI
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of Mnk1 (unknown origin) pre-incubated for 10 mins before eIF4E peptide substrate addition by ADP-Glo kinase assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28917K3PubMed
TargetMAP kinase-interacting serine/threonine-protein kinase 1(Homo sapiens (Human))
University of South Australia

Curated by ChEMBL
LigandPNGBDBM50079469(CHEMBL3417200)copy SMILEScopy InChI
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of Mnk1 (unknown origin) pre-incubated for 10 mins before eIF4E peptide substrate addition by ADP-Glo kinase assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28917K3PubMed
TargetMAP kinase-interacting serine/threonine-protein kinase 1(Homo sapiens (Human))
University of South Australia

Curated by ChEMBL
LigandPNGBDBM50079468(CHEMBL3417201)copy SMILEScopy InChI
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of Mnk1 (unknown origin) pre-incubated for 10 mins before eIF4E peptide substrate addition by ADP-Glo kinase assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28917K3PubMed
TargetMAP kinase-interacting serine/threonine-protein kinase 1(Homo sapiens (Human))
University of South Australia

Curated by ChEMBL
LigandPNGBDBM50079467(CHEMBL3417202)copy SMILEScopy InChI
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of Mnk1 (unknown origin) pre-incubated for 10 mins before eIF4E peptide substrate addition by ADP-Glo kinase assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28917K3PubMed
TargetMAP kinase-interacting serine/threonine-protein kinase 1(Homo sapiens (Human))
University of South Australia

Curated by ChEMBL
LigandPNGBDBM50079404(CHEMBL3417206)copy SMILEScopy InChI
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of Mnk1 (unknown origin) pre-incubated for 10 mins before eIF4E peptide substrate addition by ADP-Glo kinase assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28917K3PubMed
TargetMAP kinase-interacting serine/threonine-protein kinase 1(Homo sapiens (Human))
University of South Australia

Curated by ChEMBL
LigandPNGBDBM50079473(CHEMBL3417196)copy SMILEScopy InChI
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of Mnk1 (unknown origin) pre-incubated for 10 mins before eIF4E peptide substrate addition by ADP-Glo kinase assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28917K3PubMed
TargetMAP kinase-interacting serine/threonine-protein kinase 2(Homo sapiens (Human))
University of South Australia

Curated by ChEMBL
LigandPNGBDBM50079472(CHEMBL3417197)copy SMILEScopy InChI
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of Mnk2 (unknown origin) pre-incubated for 10 mins before eIF4E peptide substrate addition by ADP-Glo kinase assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28917K3PubMed
TargetMAP kinase-interacting serine/threonine-protein kinase 2(Homo sapiens (Human))
University of South Australia

Curated by ChEMBL
LigandPNGBDBM50079469(CHEMBL3417200)copy SMILEScopy InChI
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of Mnk2 (unknown origin) pre-incubated for 10 mins before eIF4E peptide substrate addition by ADP-Glo kinase assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28917K3PubMed
TargetMAP kinase-interacting serine/threonine-protein kinase 2(Homo sapiens (Human))
University of South Australia

Curated by ChEMBL
LigandPNGBDBM50079404(CHEMBL3417206)copy SMILEScopy InChI
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of Mnk2 (unknown origin) pre-incubated for 10 mins before eIF4E peptide substrate addition by ADP-Glo kinase assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28917K3PubMed
TargetMAP kinase-interacting serine/threonine-protein kinase 2(Homo sapiens (Human))
University of South Australia

Curated by ChEMBL
LigandPNGBDBM50079473(CHEMBL3417196)copy SMILEScopy InChI
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of Mnk2 (unknown origin) pre-incubated for 10 mins before eIF4E peptide substrate addition by ADP-Glo kinase assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28917K3PubMed