Compile Data Set for Download or QSAR
Found 3 Enz. Inhib. hit(s) with Target = 'MAP kinase-interacting serine/threonine-protein kinase 1' and Ligand = 'BDBM50298223'
TargetMAP kinase-interacting serine/threonine-protein kinase 1(Homo sapiens (Human))
University of South Australia

Curated by ChEMBL
LigandPNGBDBM50298223(CGP-57380 | CHEMBL1240885 | CHEMBL576817 | N-(4-fl...)copy SMILEScopy InChI
Affinity DataKi:  1.01E+3nMAssay Description:Inhibition of Mnk1 (unknown origin) pre-incubated for 10 mins before eIF4E peptide substrate addition by ADP-Glo kinase assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28917K3PubMed
TargetMAP kinase-interacting serine/threonine-protein kinase 1(Homo sapiens (Human))
University of South Australia

Curated by ChEMBL
LigandPNGBDBM50298223(CGP-57380 | CHEMBL1240885 | CHEMBL576817 | N-(4-fl...)copy SMILEScopy InChI
Affinity DataIC50: 870nMAssay Description:Inhibition of MNK1 in the presence of 50uM ATPMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27082B4PubMed
TargetMAP kinase-interacting serine/threonine-protein kinase 1(Homo sapiens (Human))
University of South Australia

Curated by ChEMBL
LigandPNGBDBM50298223(CGP-57380 | CHEMBL1240885 | CHEMBL576817 | N-(4-fl...)copy SMILEScopy InChI
Affinity DataIC50: 870nMAssay Description:Inhibition of MNK1More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Z038CPPubMed