Compile Data Set for Download or QSAR
Found 2 Enz. Inhib. hit(s) with Target = '5-hydroxytryptamine receptor 1A' and Ligand = 'BDBM50048817'
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Cracow University of Technology

Curated by ChEMBL
LigandPNGBDBM50048817(2-[6-(4-Benzo[d]isothiazol-3-yl-piperazin-1-yl)-he...)copy SMILEScopy InChI
Affinity DataKi:  18nMAssay Description:Displacement of [3H]8-OH-DPAT from human 5HT1A receptor expressed in HEK293 cell membranes measured after 1 hr by microbeta counting methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2D50RJBPubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Glaxo Wellcome Inc.

Curated by ChEMBL
LigandPNGBDBM50048817(2-[6-(4-Benzo[d]isothiazol-3-yl-piperazin-1-yl)-he...)copy SMILEScopy InChI
Affinity DataIC50: 0.760nMAssay Description:Inhibition of [3H]-8-OH-DPAT binding at serotonin 5-hydroxytryptamine 1A receptor from rat hippocampus tissue.More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TQ60MNPubMed