Compile Data Set for Download or QSAR
Found 2 Enz. Inhib. hit(s) with Target = 'Bromodomain-containing protein 4 [368-440]' and Ligand = 'BDBM249273'
TargetBromodomain-containing protein 4 [368-440](Homo sapiens (Human))
Gilead Sciences Inc

US Patent
LigandPNGBDBM249273(US10017501, Compound 1020-1 | US9458145, 1020-1)copy SMILEScopy InChI
Affinity DataIC50: 97.6nMAssay Description:Binding of the two tandem bromodomains, BRD4-1 and BRD4-2, to an acetylated histone H4 peptide was measured using a homogeneous time resolved fluores...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2CV4M3ZUS Patent
TargetBromodomain-containing protein 4 [368-440](Homo sapiens (Human))
Gilead Sciences Inc

US Patent
LigandPNGBDBM249273(US10017501, Compound 1020-1 | US9458145, 1020-1)copy SMILEScopy InChI
Affinity DataIC50: 97.6nMpH: 7.5 T: 2°CAssay Description:Binding of the two tandem bromodomains, BRD4-1 and BRD4-2, to an acetylated histone H4 peptide was measured using a homogeneous time resolved fluores...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q26Q1W53US Patent