BindingDB PrimarySearch

Found 3 Enz. Inhib. hit(s) with Target = 'Dual specificity tyrosine-phosphorylation-regulated kinase 2' and Ligand = 'BDBM246383'

Dual specificity tyrosine-phosphorylation-regulated kinase 2(Homo sapiens (Human))TBA

BDBM246383(US9446044, 69)copy SMILEScopy InChI

IC50: 3.20nMAssay Description:Inhibition of DYRK2 (unknown origin)More data for this Ligand-Target Pair

PDB MMDB NCI pathway KEGG
UniProtKB/SwissProt
B.MOAD antibodypedia GoogleScholar

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Details
BindingDB Entry DOI: 10.7270/Q2GH9NMGPubMed PDB

3D Structure (crystal)

Dual specificity tyrosine-phosphorylation-regulated kinase 2(Homo sapiens (Human))TBA

BDBM246383(US9446044, 69)copy SMILEScopy InChI

IC50: 323nMMore data for this Ligand-Target Pair

PDB MMDB NCI pathway KEGG
UniProtKB/SwissProt
B.MOAD antibodypedia GoogleScholar

Purchase MCE
PC cid PC sid PDB

Details PDB

3D Structure (crystal)

Dual specificity tyrosine-phosphorylation-regulated kinase 2(Homo sapiens (Human))TBA

BDBM246383(US9446044, 69)copy SMILEScopy InChI

IC50: 3.00E+3nMAssay Description:Inhibition of DYRK2 (unknown origin) by NanoBRET cellular target engagement assayMore data for this Ligand-Target Pair

PDB MMDB NCI pathway KEGG
UniProtKB/SwissProt
B.MOAD antibodypedia GoogleScholar

Purchase MCE
PC cid PC sid PDB

Details Article
BindingDB Entry DOI: 10.7270/Q2KD22MPPubMed PDB

3D Structure (crystal)