Found 5 Enz. Inhib. hit(s) with Target = 'Excitatory amino acid transporter 2' and Ligand = 'BDBM86712' TargetExcitatory amino acid transporter 2(Homo sapiens (Human))
Wyeth Research
Curated by PDSP Ki Database
Wyeth Research
Curated by PDSP Ki Database
3D Structure (crystal)TargetExcitatory amino acid transporter 2(Homo sapiens (Human))
Wyeth Research
Curated by PDSP Ki Database
Wyeth Research
Curated by PDSP Ki Database
Affinity DataIC50: 71nMAssay Description:Inhibition of human EAAT2 expressed in HEK293 cells assessed as reduction in [3H]-D-Asp uptake incubated for 4 mins by scintillation counting methodMore data for this Ligand-Target Pair
TargetExcitatory amino acid transporter 2(Homo sapiens (Human))
Wyeth Research
Curated by PDSP Ki Database
Wyeth Research
Curated by PDSP Ki Database
Affinity DataIC50: 71nMAssay Description:Inhibition of human EAAT2 expressed in HEK293 cells assessed as reduction in [3H]-D-Asp uptake incubated for 4 mins by scintillation counting methodMore data for this Ligand-Target Pair
TargetExcitatory amino acid transporter 2(Homo sapiens (Human))
Wyeth Research
Curated by PDSP Ki Database
Wyeth Research
Curated by PDSP Ki Database
Affinity DataIC50: 80nMAssay Description:Inhibitory concentration against glutamate uptake in HEK cells expressing human Excitatory amino acid transporter 2More data for this Ligand-Target Pair
TargetExcitatory amino acid transporter 2(Homo sapiens (Human))
Wyeth Research
Curated by PDSP Ki Database
Wyeth Research
Curated by PDSP Ki Database
Affinity DataIC50: 130nMAssay Description:Inhibitory concentration against glutamate uptake in oocytes expressing in human Excitatory amino acid transporter 2More data for this Ligand-Target Pair
