Compile Data Set for Download or QSAR
Found 2 Enz. Inhib. hit(s) with Target = 'Excitatory amino acid transporter 4' and Ligand = 'BDBM86712'
TargetExcitatory amino acid transporter 4(Rattus norvegicus)
University of Groningen

Curated by ChEMBL
LigandPNGBDBM86712(CAS_868359-05-1 | N-[4-(2-BROMO-4,5-DIFLUOROPHENOX...)copy SMILEScopy InChI
Affinity DataIC50: 1.50E+3nMAssay Description:Inhibition of rat EAAT4 expressed in tsA201 cells assessed as reduction in [3H]-D-Asp uptake incubated for 4 mins by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2G44ST4PubMed
TargetExcitatory amino acid transporter 4(Rattus norvegicus)
University of Groningen

Curated by ChEMBL
LigandPNGBDBM86712(CAS_868359-05-1 | N-[4-(2-BROMO-4,5-DIFLUOROPHENOX...)copy SMILEScopy InChI
Affinity DataIC50: 1.50E+3nMAssay Description:Inhibition of rat EAAT4 expressed in tsA201 cells assessed as reduction in [3H]-D-Asp uptake incubated for 4 mins by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2G44ST4PubMed