Compile Data Set for Download or QSAR
Found 3 Enz. Inhib. hit(s) with Target = 'Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit beta isoform' and Ligand = 'BDBM50347076'
LigandPNGBDBM50347076(CHEMBL1796761)copy SMILEScopy InChI
Affinity DataKi:  19nMAssay Description:Apparent binding affinity to PI3Kbeta using PIP3 as substrate after 30 mins by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2057GCQPubMed
LigandPNGBDBM50347076(CHEMBL1796761)copy SMILEScopy InChI
Affinity DataIC50: 22nMAssay Description:Inhibition of PI3Kbeta using PIP3 as substrate after 30 mins by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2057GCQPubMed
LigandPNGBDBM50347076(CHEMBL1796761)copy SMILEScopy InChI
Affinity DataIC50: 60nMAssay Description:Inhibition of PI3KbetaMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29G5N57PubMed