Compile Data Set for Download or QSAR
Found 4 Enz. Inhib. hit(s) with Target = 'Urokinase-type plasminogen activator' and Ligand = 'BDBM772'
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
Axys Pharmaceuticals Corporation

LigandPNGBDBM772(Benzamidine | CHEMBL79897 | [amino(phenyl)methylid...)copy SMILEScopy InChI
Affinity DataKi:  5.00E+3nMAssay Description:Each enzyme was assayed with a set of different concentrations of each inhibitor. After addition of the appropriate substrate, the rate of hydrolysis...More data for this Ligand-Target Pair
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
Axys Pharmaceuticals Corporation

LigandPNGBDBM772(Benzamidine | CHEMBL79897 | [amino(phenyl)methylid...)copy SMILEScopy InChI
Affinity DataKi:  9.50E+4nMAssay Description:Each enzyme was assayed with a set of different concentrations of each inhibitor. After addition of the appropriate substrate, the rate of hydrolysis...More data for this Ligand-Target Pair
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
Axys Pharmaceuticals Corporation

LigandPNGBDBM772(Benzamidine | CHEMBL79897 | [amino(phenyl)methylid...)copy SMILEScopy InChI
Affinity DataKi:  9.70E+4nM ΔG°:  -22.7kJ/molepH: 7.4 T: 2°CAssay Description:Each enzyme was assayed with a set of different concentrations of each inhibitor. After addition of the appropriate substrate, the rate of hydrolysis...More data for this Ligand-Target Pair
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
Axys Pharmaceuticals Corporation

LigandPNGBDBM772(Benzamidine | CHEMBL79897 | [amino(phenyl)methylid...)copy SMILEScopy InChI
Affinity DataKi:  1.80E+5nM ΔG°:  -21.4kJ/molepH: 8.0 T: 2°CAssay Description:The measurements were carried out on a microplate reader. Two concentrations of the substrate and five concentrations of the inhibitor were used in t...More data for this Ligand-Target Pair