Compile Data Set for Download or QSAR
Found 23 Enz. Inhib. hit(s) with all data for assayid = 2 entry = 50011174
TargetD(2) dopamine receptor(Homo sapiens (Human))
Cracow University of Technology

Curated by ChEMBL
LigandPNGBDBM50545435(CHEMBL4641609)copy SMILEScopy InChI
Affinity DataKi:  1nMAssay Description:Displacement of [3H]-raclopride from human D2L receptor expressed in HEK293 cell membranes measured after 1 hr by microbeta counting methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2D50RJBPubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Cracow University of Technology

Curated by ChEMBL
LigandPNGBDBM50545449(CHEMBL4642981)copy SMILEScopy InChI
Affinity DataKi:  1nMAssay Description:Displacement of [3H]-raclopride from human D2L receptor expressed in HEK293 cell membranes measured after 1 hr by microbeta counting methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2D50RJBPubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Cracow University of Technology

Curated by ChEMBL
LigandPNGBDBM50545442(CHEMBL4648581)copy SMILEScopy InChI
Affinity DataKi:  9nMAssay Description:Displacement of [3H]-raclopride from human D2L receptor expressed in HEK293 cell membranes measured after 1 hr by microbeta counting methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2D50RJBPubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Cracow University of Technology

Curated by ChEMBL
LigandPNGBDBM50048817(2-[6-(4-Benzo[d]isothiazol-3-yl-piperazin-1-yl)-he...)copy SMILEScopy InChI
Affinity DataKi:  10nMAssay Description:Displacement of [3H]-raclopride from human D2L receptor expressed in HEK293 cell membranes measured after 1 hr by microbeta counting methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2D50RJBPubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Cracow University of Technology

Curated by ChEMBL
LigandPNGBDBM50545453(CHEMBL4645793)copy SMILEScopy InChI
Affinity DataKi:  14nMAssay Description:Displacement of [3H]-raclopride from human D2L receptor expressed in HEK293 cell membranes measured after 1 hr by microbeta counting methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2D50RJBPubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Cracow University of Technology

Curated by ChEMBL
LigandPNGBDBM50545452(CHEMBL4638308)copy SMILEScopy InChI
Affinity DataKi:  16nMAssay Description:Displacement of [3H]-raclopride from human D2L receptor expressed in HEK293 cell membranes measured after 1 hr by microbeta counting methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2D50RJBPubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Cracow University of Technology

Curated by ChEMBL
LigandPNGBDBM50545443(CHEMBL4643450)copy SMILEScopy InChI
Affinity DataKi:  16nMAssay Description:Displacement of [3H]-raclopride from human D2L receptor expressed in HEK293 cell membranes measured after 1 hr by microbeta counting methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2D50RJBPubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Cracow University of Technology

Curated by ChEMBL
LigandPNGBDBM50545447(CHEMBL4642594)copy SMILEScopy InChI
Affinity DataKi:  18nMAssay Description:Displacement of [3H]-raclopride from human D2L receptor expressed in HEK293 cell membranes measured after 1 hr by microbeta counting methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2D50RJBPubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Cracow University of Technology

Curated by ChEMBL
LigandPNGBDBM50545456(CHEMBL4645525)copy SMILEScopy InChI
Affinity DataKi:  27nMAssay Description:Displacement of [3H]-raclopride from human D2L receptor expressed in HEK293 cell membranes measured after 1 hr by microbeta counting methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2D50RJBPubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Cracow University of Technology

Curated by ChEMBL
LigandPNGBDBM50545455(CHEMBL4636031)copy SMILEScopy InChI
Affinity DataKi:  31nMAssay Description:Displacement of [3H]-raclopride from human D2L receptor expressed in HEK293 cell membranes measured after 1 hr by microbeta counting methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2D50RJBPubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Cracow University of Technology

Curated by ChEMBL
LigandPNGBDBM50545454(CHEMBL4641296)copy SMILEScopy InChI
Affinity DataKi:  31nMAssay Description:Displacement of [3H]-raclopride from human D2L receptor expressed in HEK293 cell membranes measured after 1 hr by microbeta counting methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2D50RJBPubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Cracow University of Technology

Curated by ChEMBL
LigandPNGBDBM50545444(CHEMBL4635603)copy SMILEScopy InChI
Affinity DataKi:  33nMAssay Description:Displacement of [3H]-raclopride from human D2L receptor expressed in HEK293 cell membranes measured after 1 hr by microbeta counting methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2D50RJBPubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Cracow University of Technology

Curated by ChEMBL
LigandPNGBDBM50545436(CHEMBL4645308)copy SMILEScopy InChI
Affinity DataKi:  35nMAssay Description:Displacement of [3H]-raclopride from human D2L receptor expressed in HEK293 cell membranes measured after 1 hr by microbeta counting methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2D50RJBPubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Cracow University of Technology

Curated by ChEMBL
LigandPNGBDBM50545445(CHEMBL4644906)copy SMILEScopy InChI
Affinity DataKi:  39nMAssay Description:Displacement of [3H]-raclopride from human D2L receptor expressed in HEK293 cell membranes measured after 1 hr by microbeta counting methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2D50RJBPubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Cracow University of Technology

Curated by ChEMBL
LigandPNGBDBM50545441(CHEMBL4645292)copy SMILEScopy InChI
Affinity DataKi:  41nMAssay Description:Displacement of [3H]-raclopride from human D2L receptor expressed in HEK293 cell membranes measured after 1 hr by microbeta counting methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2D50RJBPubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Cracow University of Technology

Curated by ChEMBL
LigandPNGBDBM50545439(CHEMBL4639203)copy SMILEScopy InChI
Affinity DataKi:  55nMAssay Description:Displacement of [3H]-raclopride from human D2L receptor expressed in HEK293 cell membranes measured after 1 hr by microbeta counting methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2D50RJBPubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Cracow University of Technology

Curated by ChEMBL
LigandPNGBDBM50545446(CHEMBL4637294)copy SMILEScopy InChI
Affinity DataKi:  56nMAssay Description:Displacement of [3H]-raclopride from human D2L receptor expressed in HEK293 cell membranes measured after 1 hr by microbeta counting methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2D50RJBPubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Cracow University of Technology

Curated by ChEMBL
LigandPNGBDBM50545448(CHEMBL4646868)copy SMILEScopy InChI
Affinity DataKi:  59nMAssay Description:Displacement of [3H]-raclopride from human D2L receptor expressed in HEK293 cell membranes measured after 1 hr by microbeta counting methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2D50RJBPubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Cracow University of Technology

Curated by ChEMBL
LigandPNGBDBM50545451(CHEMBL4638388)copy SMILEScopy InChI
Affinity DataKi:  106nMAssay Description:Displacement of [3H]-raclopride from human D2L receptor expressed in HEK293 cell membranes measured after 1 hr by microbeta counting methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2D50RJBPubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Cracow University of Technology

Curated by ChEMBL
LigandPNGBDBM50545450(CHEMBL4648390)copy SMILEScopy InChI
Affinity DataKi:  164nMAssay Description:Displacement of [3H]-raclopride from human D2L receptor expressed in HEK293 cell membranes measured after 1 hr by microbeta counting methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2D50RJBPubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Cracow University of Technology

Curated by ChEMBL
LigandPNGBDBM50545440(CHEMBL4636435)copy SMILEScopy InChI
Affinity DataKi:  168nMAssay Description:Displacement of [3H]-raclopride from human D2L receptor expressed in HEK293 cell membranes measured after 1 hr by microbeta counting methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2D50RJBPubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Cracow University of Technology

Curated by ChEMBL
LigandPNGBDBM50545437(CHEMBL4635363)copy SMILEScopy InChI
Affinity DataKi:  225nMAssay Description:Displacement of [3H]-raclopride from human D2L receptor expressed in HEK293 cell membranes measured after 1 hr by microbeta counting methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2D50RJBPubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Cracow University of Technology

Curated by ChEMBL
LigandPNGBDBM50545438(CHEMBL4632519)copy SMILEScopy InChI
Affinity DataKi:  370nMAssay Description:Displacement of [3H]-raclopride from human D2L receptor expressed in HEK293 cell membranes measured after 1 hr by microbeta counting methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2D50RJBPubMed