Compile Data Set for Download or QSAR
Found 6 Enz. Inhib. hit(s) with all data for assayid = 3 entry = 8086
TargetSerine protease 1(Homo sapiens (Human))
Medical University of Bialystok

LigandPNGBDBM233006(H-D-Ser-Ala-Arg-NH-(CH2)6-NH2 (5))copy SMILEScopy InChI
Affinity DataKi:  2.50E+3nMpH: 7.5Assay Description:Determination of amidolytic activity was performed as described previously [Okada et al., Chem. Pharm. Bull., 36:1289-1297]. Detailed description of ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q23R0RR3PubMed
TargetSerine protease 1(Homo sapiens (Human))
Medical University of Bialystok

LigandPNGBDBM233009(H-D-Ser-Ala-Arg-NH-(CH2)9-NH2 (8))copy SMILEScopy InChI
Affinity DataKi:  5.00E+3nMpH: 7.5Assay Description:Determination of amidolytic activity was performed as described previously [Okada et al., Chem. Pharm. Bull., 36:1289-1297]. Detailed description of ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q23R0RR3PubMed
TargetSerine protease 1(Homo sapiens (Human))
Medical University of Bialystok

LigandPNGBDBM233012(H-D-Ser-Ala-Arg-NH-(CH2)4-OH (11))copy SMILEScopy InChI
Affinity DataKi:  1.00E+4nMpH: 7.5Assay Description:Determination of amidolytic activity was performed as described previously [Okada et al., Chem. Pharm. Bull., 36:1289-1297]. Detailed description of ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q23R0RR3PubMed
TargetSerine protease 1(Homo sapiens (Human))
Medical University of Bialystok

LigandPNGBDBM233008(H-D-Ser-Ala-Arg-NH-(CH2)8-NH2 (7))copy SMILEScopy InChI
Affinity DataKi:  1.00E+4nMpH: 7.5Assay Description:Determination of amidolytic activity was performed as described previously [Okada et al., Chem. Pharm. Bull., 36:1289-1297]. Detailed description of ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q23R0RR3PubMed
TargetSerine protease 1(Homo sapiens (Human))
Medical University of Bialystok

LigandPNGBDBM233011(H-D-Ser-Ala-Arg-NH-(CH2)3-OH (10))copy SMILEScopy InChI
Affinity DataKi:  1.50E+4nMpH: 7.5Assay Description:Determination of amidolytic activity was performed as described previously [Okada et al., Chem. Pharm. Bull., 36:1289-1297]. Detailed description of ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q23R0RR3PubMed
TargetSerine protease 1(Homo sapiens (Human))
Medical University of Bialystok

LigandPNGBDBM233007(H-D-Ser-Ala-Arg-NH-(CH2)7-NH2 (6))copy SMILEScopy InChI
Affinity DataKi:  3.00E+4nMpH: 7.5Assay Description:Determination of amidolytic activity was performed as described previously [Okada et al., Chem. Pharm. Bull., 36:1289-1297]. Detailed description of ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q23R0RR3PubMed