Compile Data Set for Download or QSAR
Found 3 Enz. Inhib. hit(s) with Target = 'Casein kinase I isoform gamma-2' and Ligand = 'BDBM50400744'
TargetCasein kinase I isoform gamma-2(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50400744(CHEMBL2203560)copy SMILEScopy InChI
Affinity DataIC50: 26nMAssay Description:Inhibition of CK1-gamma 2 using biotin[long chain]-KKRRRAL{pS}VATLPGL substrate in presence of 32 uM ATPMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21V5G41PubMed
TargetCasein kinase I isoform gamma-2(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50400744(CHEMBL2203560)copy SMILEScopy InChI
Affinity DataIC50: 840nMAssay Description:Inhibition of human CK1-gamma2 in HEK293 cells assessed as inhibition of doxcycline-induced LRP6 phosphorylation after 2 hrs by electrochemiluminesce...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21V5G41PubMed
TargetCasein kinase I isoform gamma-2(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50400744(CHEMBL2203560)copy SMILEScopy InChI
Affinity DataIC50: 1.30E+3nMAssay Description:Inhibition of CK1-gamma2 in human RKO cell assessed as inhibition of Wnt3a-induced Wnt signaling treated 1 hr prior to Wnt3a ligand addition measured...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21V5G41PubMed