Compile Data Set for Download or QSAR
Found 2 Enz. Inhib. hit(s) with Target = 'Excitatory amino acid transporter 2' and Ligand = 'BDBM50180145'
TargetExcitatory amino acid transporter 2(Homo sapiens (Human))
University of Berne

Curated by ChEMBL
LigandPNGBDBM50180145((1R,4S,5R,6S)-3-azabicyclo[3.3.0]octane-4,6-dicarb...)copy SMILEScopy InChI
Affinity DataKi:  5.20E+4nMAssay Description:Inhibition of human GLT1 expressed in Xenopus laevis Oocytes assessed as reduction of [3H]-glutamate uptake after 10 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27081NRPubMed
TargetExcitatory amino acid transporter 2(Homo sapiens (Human))
University of Berne

Curated by ChEMBL
LigandPNGBDBM50180145((1R,4S,5R,6S)-3-azabicyclo[3.3.0]octane-4,6-dicarb...)copy SMILEScopy InChI
Affinity DataKi:  5.20E+4nMAssay Description:Activity against human EAAT2 transfected in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2GM86WBPubMed