Compile Data Set for Download or QSAR
Found 3 Enz. Inhib. hit(s) with Target = 'Free fatty acid receptor 1' and Ligand = 'BDBM168162'
TargetFree fatty acid receptor 1(Homo sapiens (Human))
SRMLSC

US Patent
LigandPNGBDBM168162(US9688642, 10)copy SMILEScopy InChI
Affinity DataEC50:  8nMT: 2°CAssay Description:Compounds were tested in a calcium flux assay using transfected HEK293 cells stably expressing either human GPR40 or rat GPR40. Human GPR40 expressin...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2QV3JQXUS Patent
TargetFree fatty acid receptor 1(Homo sapiens (Human))
SRMLSC

US Patent
LigandPNGBDBM168162(US9688642, 10)copy SMILEScopy InChI
Affinity DataEC50:  7.5nMAssay Description:Agonist activity at human GPR40 transfected in HEK293 cells assessed as increase in intracellular calcium level incubated for 1 hr by Fluo-8 dye base...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21R6V4XPubMed
TargetFree fatty acid receptor 1(Rattus norvegicus)
SRMLSC

US Patent
LigandPNGBDBM168162(US9688642, 10)copy SMILEScopy InChI
Affinity DataEC50:  31nMT: 2°CAssay Description:Compounds were tested in a calcium flux assay using transfected HEK293 cells stably expressing either human GPR40 or rat GPR40. Human GPR40 expressin...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2QV3JQXUS Patent