BindingDB PrimarySearch

Found 1 Enz. Inhib. hit(s) with Target = 'Gag-Pol polyprotein [588-1027,K691N,Y769C]/[588-1147,K691N,Y769C]' and Ligand = 'BDBM27609'

Gag-Pol polyprotein [588-1027,K691N,Y769C]/[588-1147,K691N,Y769C](Human immunodeficiency virus type 1)
Roche Palo Alto LLC

BDBM27609(3-{[4-bromo-3-(3-chloro-5-cyanophenoxy)-2-fluoroph...)copy SMILEScopy InChI

IC50: 15nM EC50: 53nMpH: 8.0 T: 2°CAssay Description:IC50s were obtained from the inhibition of the RNA-dependent DNA polymerase activity of the HIV-1 reverse transcriptase enzyme using a primer extensi...More data for this Ligand-Target Pair

PDB MMDB
UniProtKB/SwissProt
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PC cid PC sid Similars

Details Article
BindingDB Entry DOI: 10.7270/Q2TQ5ZV0PubMed