Compile Data Set for Download or QSAR
Found 1 Enz. Inhib. hit(s) with Target = 'Glutaminyl-peptide cyclotransferase' and Ligand = 'BDBM3740'
TargetGlutaminyl-peptide cyclotransferase(Homo sapiens (Human))
Probiodrug AG

US Patent
LigandPNGBDBM3740(US8530670, 27)copy SMILEScopy InChI
Affinity DataKi:  4.60nM ΔG°:  -48.4kJ/mole IC50: 46.1nMT: 2°CAssay Description:This novel assay was used to determine the kinetic parameters for most of the QC substrate. QC activity was analyzed spectrophotometrically using a ...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2PK0DTDUS Patent