Found 2 Enz. Inhib. hit(s) with Target = 'Histone acetyltransferase GCN5' and Ligand = 'BDBM50076483'
TargetHistone acetyltransferase GCN5(Saccharomyces cerevisiae S288c)
Mayo Clinic College of Medicine
Curated by ChEMBL
Mayo Clinic College of Medicine
Curated by ChEMBL
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibition of Vps75-stimulated recombinant Saccharomyces cerevisiae histone acetyltransferase Rtt109 using Asf1-dH3-H4 as substrate assessed as coenz...More data for this Ligand-Target Pair
TargetHistone acetyltransferase GCN5(Saccharomyces cerevisiae S288c)
Mayo Clinic College of Medicine
Curated by ChEMBL
Mayo Clinic College of Medicine
Curated by ChEMBL
Affinity DataIC50: 1.30E+4nMAssay Description:Inhibition of Vps75-stimulated recombinant Saccharomyces cerevisiae histone acetyltransferase Rtt109 using Asf1-dH3-H4 as substrate assessed as coenz...More data for this Ligand-Target Pair