Found 2 Enz. Inhib. hit(s) with Target = 'Histone acetyltransferase GCN5' and Ligand = 'BDBM53290' TargetHistone acetyltransferase GCN5(Saccharomyces cerevisiae S288c)
Mayo Clinic College of Medicine
Curated by ChEMBL
Mayo Clinic College of Medicine
Curated by ChEMBL
Affinity DataIC50: 130nMAssay Description:Inhibition of Vps75-stimulated recombinant Saccharomyces cerevisiae histone acetyltransferase Rtt109 using [3H]-acetyl-CoA assessed as acetate incorp...More data for this Ligand-Target Pair
TargetHistone acetyltransferase GCN5(Saccharomyces cerevisiae S288c)
Mayo Clinic College of Medicine
Curated by ChEMBL
Mayo Clinic College of Medicine
Curated by ChEMBL
Affinity DataIC50: 1.20E+3nMAssay Description:Inhibition of yeast histone acetyltransferase Gcn5-Ada2-Ada3 complex using tetramer and [3H]-acetyl-CoA assessed as acetate incorporation after 30 mi...More data for this Ligand-Target Pair
