Compile Data Set for Download or QSAR
Found 1 Enz. Inhib. hit(s) with Target = 'Kelch-like ECH-associated protein 1' and Ligand = 'BDBM50502734'
TargetKelch-like ECH-associated protein 1(Homo sapiens (Human))
Temple University School of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50502734(CHEMBL4442320 | US11479539, Compound 42)copy SMILEScopy InChI
Affinity DataEC50:  33nMAssay Description:Inhibition of KEAP1 interaction with Nrf2 in human HEK293 cells transfected with ARE-LUC assessed as activation of Nrf2 signaling pathway measured af...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QZ2F72PubMed