Compile Data Set for Download or QSAR
Found 4 Enz. Inhib. hit(s) with Target = 'Leucyl-cystinyl aminopeptidase' and Ligand = 'BDBM271252'
TargetLeucyl-cystinyl aminopeptidase(Homo sapiens (Human))
Astellas Pharma Inc.; KOTOBUKI PHARMACEUTICALS CO., LTD.

US Patent
LigandPNGBDBM271252(US10059720, Example 67 | US10975091, Example 67)copy SMILEScopy InChI
Affinity DataIC50: 1.80nMAssay Description:HEK293 cells forced to transiently express hP-LAP (J Biol Chem 1996; 271: 56-61) were prepared by lipofection, homogenized, and then subjected to ult...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2XD13Q5US Patent
TargetLeucyl-cystinyl aminopeptidase(Homo sapiens (Human))
Astellas Pharma Inc.; KOTOBUKI PHARMACEUTICALS CO., LTD.

US Patent
LigandPNGBDBM271252(US10059720, Example 67 | US10975091, Example 67)copy SMILEScopy InChI
Affinity DataIC50: 1.80nMAssay Description:hP-LAP: HEK293 cells forced to transiently express hP-LAP were prepared by lipofection, homogenized, and then subjected to ultracentrifugation at 100...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2FF3WHRUS Patent
TargetLeucyl-cystinyl aminopeptidase(Rattus norvegicus)
Astellas Pharma Inc.; KOTOBUKI PHARMACEUTICAL CO., LTD.

US Patent
LigandPNGBDBM271252(US10059720, Example 67 | US10975091, Example 67)copy SMILEScopy InChI
Affinity DataIC50: 1.90nMAssay Description:IRAP: Rat epididymal fat pads were homogenized and subjected to ultracentrifugation at 100,000×g for 30 minutes to obtain microsomes containing IRAP....More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2FF3WHRUS Patent
TargetLeucyl-cystinyl aminopeptidase(Rattus norvegicus)
Astellas Pharma Inc.; KOTOBUKI PHARMACEUTICAL CO., LTD.

US Patent
LigandPNGBDBM271252(US10059720, Example 67 | US10975091, Example 67)copy SMILEScopy InChI
Affinity DataIC50: 1.90nMAssay Description:Rat epididymal fat pads were homogenized and subjected to ultracentrifugation at 100,000×g for 30 minutes to obtain microsomes containing IRAP. The m...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2XD13Q5US Patent