Compile Data Set for Download or QSAR
Found 4 Enz. Inhib. hit(s) with Target = 'Melanocortin receptor 3' and Ligand = 'BDBM50565827'
TargetMelanocortin receptor 3(Homo sapiens (Human))TBA
LigandPNGBDBM50565827(CHEMBL4794990)copy SMILES
Affinity DataKi:  0.352nMAssay Description:Displacement of [125I]-[NIe,DPhe7]-alpha-MSH from human MC3R expressed in HEK293 cell membranes incubated for 120 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2C53QMNPubMed
TargetMelanocortin receptor 3(Homo sapiens (Human))TBA
LigandPNGBDBM50565827(CHEMBL4794990)copy SMILES
Affinity DataKi:  0.355nMAssay Description:Displacement of [125I]-[NIe,DPhe7]-alpha-MSH from human MC3R expressed in HEK293 cell membranes incubated for 120 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2C53QMNPubMed
TargetMelanocortin receptor 3(Homo sapiens (Human))TBA
LigandPNGBDBM50565827(CHEMBL4794990)copy SMILES
Affinity DataIC50: 345nMAssay Description:Antagonist activity at human MC3R expressed in HEK293 cells expressing the GScAMP22F cAMP reporter assessed as reduction in alpha-MSH-induced cAMP ac...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2C53QMNPubMed
TargetMelanocortin receptor 3(Homo sapiens (Human))TBA
LigandPNGBDBM50565827(CHEMBL4794990)copy SMILES
Affinity DataIC50: 347nMAssay Description:Antagonist activity at human MC3R expressed in HEK293 cells expressing the GScAMP22F cAMP reporter assessed as reduction in alpha-MSH-induced cAMP ac...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2C53QMNPubMed