Compile Data Set for Download or QSAR
Found 3 Enz. Inhib. hit(s) with Target = 'Metabotropic glutamate receptor 4' and Ligand = 'BDBM50241580'
TargetMetabotropic glutamate receptor 4(Homo sapiens (Human))
Prexton Therapeutics

Curated by ChEMBL
LigandPNGBDBM50241580(CHEMBL4089083)copy SMILEScopy InChI
Affinity DataEC50:  79nMAssay Description:Positive allosteric modulation of recombinant human mGlu4 receptor expressed in HEK293 cells co-expressing Gi/Gq assessed as increase in glutamate-in...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2GF0WNQPubMed
TargetMetabotropic glutamate receptor 4(Homo sapiens (Human))
Prexton Therapeutics

Curated by ChEMBL
LigandPNGBDBM50241580(CHEMBL4089083)copy SMILEScopy InChI
Affinity DataEC50: >1.50E+4nMAssay Description:Positive allosteric modulation of recombinant human mGlu4 receptor expressed in HEK293 cells co-expressing chimeric G protein assessed as increase in...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2GF0WNQPubMed
TargetMetabotropic glutamate receptor 4(Rattus norvegicus (Rat))
Prexton Therapeutics

Curated by ChEMBL
LigandPNGBDBM50241580(CHEMBL4089083)copy SMILEScopy InChI
Affinity DataEC50:  47nMAssay Description:Positive allosteric modulation of rat mGlu4 receptor expressed in HEK293 cells co-expressing Gi/Gq assessed as increase in glutamate-induced calcium ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2GF0WNQPubMed