Compile Data Set for Download or QSAR
Found 1 Enz. Inhib. hit(s) with Target = 'Protein farnesyltransferase/geranylgeranyltransferase type-1 subunit alpha' and Ligand = 'BDBM13331'
TargetProtein farnesyltransferase/geranylgeranyltransferase type-1 subunit alpha(Rattus norvegicus (rat))
University of Washington at Seattle

LigandPNGBDBM13331(N-tert-butyl-2-({6-isocyano-1-[(1-methyl-1H-imidaz...)copy SMILEScopy InChI
Affinity DataIC50: 1.80nMAssay Description:Assays for PFT activity were performed with a PFT-specific scintillation assay (SPA) kit (Amersham Biosciences, Piscataway, NJ). IC50 values were cal...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BC3WSQPubMed