Found 20 Enz. Inhib. hit(s) with Target = 'Purine nucleoside phosphorylase' and Ligand = 'BDBM50195587'
TargetPurine nucleoside phosphorylase(Homo sapiens (Human))
Industrial Research Limited
Curated by ChEMBL
Industrial Research Limited
Curated by ChEMBL
Affinity DataKi: 0.0560nMAssay Description:Inhibition of human PNP by xanthine-oxidase coupled assayMore data for this Ligand-Target Pair
TargetPurine nucleoside phosphorylase(Homo sapiens (Human))
Industrial Research Limited
Curated by ChEMBL
Industrial Research Limited
Curated by ChEMBL
Affinity DataKi: 0.0560nMAssay Description:Inhbitory activity of compound against human purine nucleoside phosphorylase (PNP)More data for this Ligand-Target Pair
TargetPurine nucleoside phosphorylase(Homo sapiens (Human))
Industrial Research Limited
Curated by ChEMBL
Industrial Research Limited
Curated by ChEMBL
Affinity DataKi: 0.0560nMAssay Description:Dissociation constant against Human Purine Nucleoside Phosphorylase was reportedMore data for this Ligand-Target Pair
TargetPurine nucleoside phosphorylase(Homo sapiens (Human))
Industrial Research Limited
Curated by ChEMBL
Industrial Research Limited
Curated by ChEMBL
Affinity DataKi: 0.0560nMAssay Description:Equilibrium dissociation constant determined against human purine nucleoside phosphorylase (PNP) after slow-onset inhibitionMore data for this Ligand-Target Pair
TargetPurine nucleoside phosphorylase(Homo sapiens (Human))
Industrial Research Limited
Curated by ChEMBL
Industrial Research Limited
Curated by ChEMBL
Affinity DataKi: 0.0579nMAssay Description:Equilibrium binding affinity to wild type human PNPMore data for this Ligand-Target Pair
Affinity DataKi: 0.600nMAssay Description:Inhibition of Plasmodium falciparum His-tagged PNP assessed as inhibitor constant for enzyme-inhibitor-substrate complex formationMore data for this Ligand-Target Pair
Affinity DataKi: 0.860nMAssay Description:Inhibition of Plasmodium falciparum PNP expressed in Escherichia coli BL21(DE3) cells by spectrophotometryMore data for this Ligand-Target Pair
TargetPurine nucleoside phosphorylase(Homo sapiens (Human))
Industrial Research Limited
Curated by ChEMBL
Industrial Research Limited
Curated by ChEMBL
Affinity DataKi: 1.80nMAssay Description:Inhibition of human PNP activityMore data for this Ligand-Target Pair
TargetPurine nucleoside phosphorylase(Homo sapiens (Human))
Industrial Research Limited
Curated by ChEMBL
Industrial Research Limited
Curated by ChEMBL
Affinity DataKi: 3.30nMAssay Description:Binding affinity towards Human Purine Nucleoside Phosphorylase was reportedMore data for this Ligand-Target Pair
TargetPurine nucleoside phosphorylase(Homo sapiens (Human))
Industrial Research Limited
Curated by ChEMBL
Industrial Research Limited
Curated by ChEMBL
Affinity DataKi: 3.30nMAssay Description:Initial binding affinity to wild type human PNPMore data for this Ligand-Target Pair
TargetPurine nucleoside phosphorylase(Homo sapiens (Human))
Industrial Research Limited
Curated by ChEMBL
Industrial Research Limited
Curated by ChEMBL
Affinity DataKi: 3.30nMAssay Description:Inhibition of human purine nucleoside phosphorylase; Initial rate.More data for this Ligand-Target Pair
Affinity DataKi: 29nMAssay Description:Inhibition of Plasmodium falciparum His-tagged PNP assessed as inhibitor constant for enzyme-inhibitor complex formationMore data for this Ligand-Target Pair
TargetPurine nucleoside phosphorylase(Bos taurus (bovine))
Tokyo University of Pharmacy and Life Sciences
Curated by ChEMBL
Tokyo University of Pharmacy and Life Sciences
Curated by ChEMBL
Affinity DataKi: 41nMAssay Description:Inhibition of calf spleen PNP assessed as inhibition of 7-methylguanosine phosphorolysis after 50 mins by spectrophotometry in presence of 50 mM inor...More data for this Ligand-Target Pair
TargetPurine nucleoside phosphorylase(Homo sapiens (Human))
Industrial Research Limited
Curated by ChEMBL
Industrial Research Limited
Curated by ChEMBL
Affinity DataKi: 72nMAssay Description:Inhibition of human PNP assessed as inhibitor constant for enzyme-inhibitor-substrate complex formationMore data for this Ligand-Target Pair
TargetPurine nucleoside phosphorylase(Homo sapiens (Human))
Industrial Research Limited
Curated by ChEMBL
Industrial Research Limited
Curated by ChEMBL
TargetPurine nucleoside phosphorylase(Homo sapiens (Human))
Industrial Research Limited
Curated by ChEMBL
Industrial Research Limited
Curated by ChEMBL
Affinity DataIC50: 3.5nMAssay Description:Inhibition of human PNP activityMore data for this Ligand-Target Pair
TargetPurine nucleoside phosphorylase(Homo sapiens (Human))
Industrial Research Limited
Curated by ChEMBL
Industrial Research Limited
Curated by ChEMBL
Affinity DataIC50: 100nMAssay Description:Inhibition of human purine nucleoside phosphorylaseMore data for this Ligand-Target Pair
TargetPurine nucleoside phosphorylase(Homo sapiens (Human))
Industrial Research Limited
Curated by ChEMBL
Industrial Research Limited
Curated by ChEMBL
Affinity DataKd: 0.0560nMAssay Description:Inhibition of human PNPMore data for this Ligand-Target Pair
TargetPurine nucleoside phosphorylase(Bos taurus (bovine))
Tokyo University of Pharmacy and Life Sciences
Curated by ChEMBL
Tokyo University of Pharmacy and Life Sciences
Curated by ChEMBL
Affinity DataKd: 0.0230nMAssay Description:Binding affinity to calf recombinant PNP expressed in Escherichia coli BL21 (DE3) by isothermal titration calorimetryMore data for this Ligand-Target Pair
TargetPurine nucleoside phosphorylase(Homo sapiens (Human))
Industrial Research Limited
Curated by ChEMBL
Industrial Research Limited
Curated by ChEMBL
Affinity DataKd: 0.0580nMAssay Description:Binding affinity to human PNPMore data for this Ligand-Target Pair