Compile Data Set for Download or QSAR
Found 3 Enz. Inhib. hit(s) with Target = 'Retinoic acid receptor alpha' and Ligand = 'BDBM50143833'
TargetRetinoic acid receptor alpha(Homo sapiens (Human))
GlaxoSmithKline Research and Development

Curated by ChEMBL
LigandPNGBDBM50143833((E)-3-[4-(5,5,8,8-Tetramethyl-5,6,7,8-tetrahydro-n...)copy SMILEScopy InChI
Affinity DataKi: >1.00E+3nMAssay Description:Binding affinity for retinoic acid receptor alpha (RARalpha), using 9-cis-[3H]-retinoic acidMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KH0MRCPubMed
TargetRetinoic acid receptor alpha(Homo sapiens (Human))
GlaxoSmithKline Research and Development

Curated by ChEMBL
LigandPNGBDBM50143833((E)-3-[4-(5,5,8,8-Tetramethyl-5,6,7,8-tetrahydro-n...)copy SMILEScopy InChI
Affinity DataEC50: >1.00E+4nMAssay Description:Effective concentration for retinoic acid receptor alpha induced lipogenesis in C3H10T1/2 clone 8 fibroblast cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KH0MRCPubMed
TargetRetinoic acid receptor alpha(Homo sapiens (Human))
GlaxoSmithKline Research and Development

Curated by ChEMBL
LigandPNGBDBM50143833((E)-3-[4-(5,5,8,8-Tetramethyl-5,6,7,8-tetrahydro-n...)copy SMILEScopy InChI
Affinity DataEC50: >1.00E+4nMAssay Description:Effective concentration for Retinoic acid receptor alpha activity in CV-1 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KH0MRCPubMed