Compile Data Set for Download or QSAR
Found 3 Enz. Inhib. hit(s) with Target = 'Serine/threonine-protein kinase receptor R3 [166-493]' and Ligand = 'BDBM451777'
TargetSerine/threonine-protein kinase receptor R3 [166-493](Homo sapiens (Human))
Novartis AG

US Patent
LigandPNGBDBM451777(US10710980, Example 9 | US10947218, Example 9)copy SMILEScopy InChI
Affinity DataIC50: 127nMAssay Description:In the applied method, this separation takes place inside a chip that contains a complex capillary system for simultaneous analysis of 12 samples (“1...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2DF6V81US Patent
TargetSerine/threonine-protein kinase receptor R3 [166-493](Homo sapiens (Human))
Novartis AG

US Patent
LigandPNGBDBM451777(US10710980, Example 9 | US10947218, Example 9)copy SMILEScopy InChI
Affinity DataIC50: 127nMAssay Description:A kinase selectivity panel which measures substrate peptide phosphorylation was set-up for wild-type ALK2 (aa172-499), ALK2 FOP mutant (aa172-499 R20...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q24F1TVVUS Patent
TargetSerine/threonine-protein kinase receptor R3 [166-493](Homo sapiens (Human))
Novartis AG

US Patent
LigandPNGBDBM451777(US10710980, Example 9 | US10947218, Example 9)copy SMILEScopy InChI
Affinity DataIC50: 310nMAssay Description:A kinase selectivity panel which measures substrate peptide phosphorylation was set-up for wild-type ALK2 (aa172-499), ALK2 FOP mutant (aa172-499 R20...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q24F1TVVUS Patent