Compile Data Set for Download or QSAR
Found 3 Enz. Inhib. hit(s) with Target = 'Testis-specific serine/threonine-protein kinase 1' and Ligand = 'BDBM50279383'
TargetTestis-specific serine/threonine-protein kinase 1(Homo sapiens (Human))
Chinese Academy of Medical Sciences & Peking Union Medical College

Curated by ChEMBL
LigandPNGBDBM50279383(CHEMBL484806 | sodium 2,2'-(biphenyl-4,4'-diyl)bis...)copy SMILEScopy InChI
Affinity DataIC50: 1.44E+4nMAssay Description:Inhibition of TSSK1 (unknown origin)-catalyzed phosphorylation of AALVRQMSVAFFFK substrate by LC-MS based HTP assay in absence of Pep8-(O2)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2348K8KPubMed
TargetTestis-specific serine/threonine-protein kinase 1(Homo sapiens (Human))
Chinese Academy of Medical Sciences & Peking Union Medical College

Curated by ChEMBL
LigandPNGBDBM50279383(CHEMBL484806 | sodium 2,2'-(biphenyl-4,4'-diyl)bis...)copy SMILEScopy InChI
Affinity DataIC50: 1.91E+4nMAssay Description:Inhibition of TSSK1 (unknown origin)-catalyzed phosphorylation of AALVRQMSVAFFFK substrate by LC-MS based HTP assay in presence of Pep8-(O2)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2348K8KPubMed
TargetTestis-specific serine/threonine-protein kinase 1(Homo sapiens (Human))
Chinese Academy of Medical Sciences & Peking Union Medical College

Curated by ChEMBL
LigandPNGBDBM50279383(CHEMBL484806 | sodium 2,2'-(biphenyl-4,4'-diyl)bis...)copy SMILEScopy InChI
Affinity DataIC50: 2.48E+4nMAssay Description:Inhibition of TSSK1 (unknown origin)-catalyzed phosphorylation of AALVRQMSVAFFFK substrate by luminescent kinase assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2348K8KPubMed