Compile Data Set for Download or QSAR
Found 4 Enz. Inhib. hit(s) with Target = 'Thromboxane A2 receptor' and Ligand = 'BDBM50353636'
TargetThromboxane A2 receptor(MOUSE)
University of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM50353636(CHEMBL1829802)copy SMILEScopy InChI
Affinity DataIC50: 91nMAssay Description:Antagonist activity at mouse prostanoid TP receptor expressed in QBI-HEK 293A cells assessed as inhibition of 1-BOP-induced increase in inositol mono...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2H995KGPubMed
TargetThromboxane A2 receptor(Homo sapiens (Human))
University of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM50353636(CHEMBL1829802)copy SMILEScopy InChI
Affinity DataIC50: 377nMAssay Description:Antagonist activity at human prostanoid TP receptor expressed in QBI-HEK 293A cells assessed as inhibition of 1-BOP-induced increase in inositol mono...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2H995KGPubMed
TargetThromboxane A2 receptor(Homo sapiens (Human))
University of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM50353636(CHEMBL1829802)copy SMILEScopy InChI
Affinity DataKd:  359nMAssay Description:Displacement of [3H]SQ-29548 from human prostanoid TP receptor expressed in QBI-HEK 293A cells after 2 hrs by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2H995KGPubMed
TargetThromboxane A2 receptor(MOUSE)
University of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM50353636(CHEMBL1829802)copy SMILEScopy InChI
Affinity DataKd:  17nMAssay Description:Displacement of [3H]SQ-29548 from mouse prostanoid TP receptor expressed in QBI-HEK 293A cells after 2 hrs by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2H995KGPubMed