Found 1 Enz. Inhib. hit(s) with Target = 'Thyroid hormone receptor alpha' and Ligand = 'BDBM50274812'
TargetThyroid hormone receptor alpha(Homo sapiens (Human))
Metabasis Therapeutics, Inc.
Curated by ChEMBL
Metabasis Therapeutics, Inc.
Curated by ChEMBL
Affinity DataKi: 3.74nMAssay Description:Displacement of [125I]3,5,3'-triiodo-L-thyronine from His-tagged human recombinant TRalpha1 by scintillation proximity assayMore data for this Ligand-Target Pair