Compile Data Set for Download or QSAR
Found 1 Enz. Inhib. hit(s) with Target = 'Tyrosine-protein kinase ABL1 [T315I]' and Ligand = 'BDBM81735'
TargetTyrosine-protein kinase ABL1 [T315I](Homo sapiens (Human))
ARIAD Pharmaceuticals Inc

LigandPNGBDBM81735(PPY-B)copy SMILEScopy InChI
Affinity DataIC50: 9nMpH: 7.4 T: 2°CAssay Description:Inhibition of wild-type Abl and Abl T315I kinase activity was measured in a homogeneous time-resolved fluorescence resonance energy transfer (TR-FRET...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q228063TPubMed