Compile Data Set for Download or QSAR
Found 2 Enz. Inhib. hit(s) with Target = 'Urotensin-2 receptor' and Ligand = 'BDBM50302239'
TargetUrotensin-2 receptor(Homo sapiens (Human))
Johnson& Johnson Pharmaceutical Research& Development

Curated by ChEMBL
LigandPNGBDBM50302239(2-(4-amino-1-(3,4-dimethoxyphenyl)butyl)-4-(4-((R)...)copy SMILEScopy InChI
Affinity DataKi:  3.20E+3nMAssay Description:Displacement of [125I]urotensin 2 from urotensin 2 receptor in human RMS13 cells by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2S75GD7PubMed
TargetUrotensin-2 receptor(RAT)
Johnson& Johnson Pharmaceutical Research& Development

Curated by ChEMBL
LigandPNGBDBM50302239(2-(4-amino-1-(3,4-dimethoxyphenyl)butyl)-4-(4-((R)...)copy SMILEScopy InChI
Affinity DataIC50: 200nMAssay Description:Antagonist activity at rat urotensin 2 receptor expressed in CHOK1 cells assessed as inhibition of urotensin 2-induced intracellular calcium mobiliza...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2S75GD7PubMed