Affinity DataKi: 3.98nMAssay Description:Displacement of [125I]human urotensin 2 from human recombinant urotensin 2 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 631nMAssay Description:Displacement of [125I]human urotensin 2 from cat urotensin 2 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 501nMAssay Description:Antagonist activity at human recombinant urotensin 2 receptor expressed in HEK293 cells assessed as inhibition of intercellular calcium mobilization ...More data for this Ligand-Target Pair
Affinity DataKd: 100nMAssay Description:Antagonist activity at human urotensin 2 receptor by FLIPR assayMore data for this Ligand-Target Pair