Compile Data Set for Download or QSAR
Found 4 Enz. Inhib. hit(s) with Target = 'Urotensin-2 receptor' and Ligand = 'BDBM50413014'
TargetUrotensin-2 receptor(Homo sapiens (Human))
GlaxoSmithKline

Curated by ChEMBL
LigandPNGBDBM50413014(CHEMBL497171)copy SMILEScopy InChI
Affinity DataKi:  3.98nMAssay Description:Displacement of [125I]human urotensin 2 from human recombinant urotensin 2 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2GH9K5TPubMed
TargetUrotensin-2 receptor(Felis catus)
GlaxoSmithKline

Curated by ChEMBL
LigandPNGBDBM50413014(CHEMBL497171)copy SMILEScopy InChI
Affinity DataKi:  631nMAssay Description:Displacement of [125I]human urotensin 2 from cat urotensin 2 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2GH9K5TPubMed
TargetUrotensin-2 receptor(Homo sapiens (Human))
GlaxoSmithKline

Curated by ChEMBL
LigandPNGBDBM50413014(CHEMBL497171)copy SMILEScopy InChI
Affinity DataIC50: 501nMAssay Description:Antagonist activity at human recombinant urotensin 2 receptor expressed in HEK293 cells assessed as inhibition of intercellular calcium mobilization ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2GH9K5TPubMed
TargetUrotensin-2 receptor(Homo sapiens (Human))
GlaxoSmithKline

Curated by ChEMBL
LigandPNGBDBM50413014(CHEMBL497171)copy SMILEScopy InChI
Affinity DataKd:  100nMAssay Description:Antagonist activity at human urotensin 2 receptor by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2GH9K5TPubMed