Compile Data Set for Download or QSAR
Found 33 of ic50 data for polymerid = 49000493,49000494,49000496
TargetSodium-dependent dopamine transporter(MOUSE)
Universit£ degli Studi di Urbino Carlo Bo

Curated by ChEMBL
LigandPNGBDBM22165(1-{2-[bis(4-fluorophenyl)methoxy]ethyl}-4-(3-pheny...)copy SMILEScopy InChI
Affinity DataIC50: 5nMAssay Description:Inhibitory concentration against human Adenosine A3 receptor expressed in HEK293 cells using 0.1 nM [3H]AB-MECAMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28C9X1XPubMed
TargetSodium-dependent dopamine transporter(MOUSE)
Universit£ degli Studi di Urbino Carlo Bo

Curated by ChEMBL
LigandPNGBDBM50005536(42-548 | 5-(4-Chloro-phenyl)-2,5-dihydro-3H-imidaz...)copy SMILEScopy InChI
Affinity DataIC50: 13nMAssay Description:Inhibition of mouse DAT expressed in HEK293 cells assessed as reduction in [3H]-DA uptakeMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Z60RBZPubMed
TargetSodium-dependent dopamine transporter(BOVINE)
University of Maryland

Curated by ChEMBL
LigandPNGBDBM50366564(CHEMBL1790051 | CHEMBL83729 | WIN-35065-2)copy SMILEScopy InChI
Affinity DataIC50: 22nMAssay Description:Competitive inhibition against [3H]cocaine binding to cocaine receptor in bovine striatal tissueMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2BG2PMNPubMed
TargetSodium-dependent dopamine transporter(BOVINE)
University of Maryland

Curated by ChEMBL
LigandPNGBDBM50366564(CHEMBL1790051 | CHEMBL83729 | WIN-35065-2)copy SMILEScopy InChI
Affinity DataIC50: 22nMAssay Description:Competitive inhibition against [3H]cocaine binding to cocaine receptor in bovine striatal tissueMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2BG2PMNPubMed
TargetSodium-dependent dopamine transporter(BOVINE)
University of Maryland

Curated by ChEMBL
LigandPNGBDBM50011397(8-Methyl-3-(3-nitro-phenylcarbamoyloxy)-8-aza-bicy...)copy SMILEScopy InChI
Affinity DataIC50: 37nMAssay Description:In vitro inhibitory activity towards [3H]cocaine binding to rat striatal tissueMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2X34Z21PubMed
TargetSodium-dependent dopamine transporter(BOVINE)
University of Maryland

Curated by ChEMBL
LigandPNGBDBM22418(Cocaine | Cocaine (-) | methyl (1R,2R,3S,5S)-3-(be...)copy SMILEScopy InChI
Affinity DataIC50: 65nMAssay Description:In vitro inhibitory activity towards [3H]cocaine binding to rat striatal tissueMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2X34Z21PubMed
TargetSodium-dependent dopamine transporter(BOVINE)
University of Maryland

Curated by ChEMBL
LigandPNGBDBM50015692(8-Methyl-3-(4-nitro-phenyl)-8-aza-bicyclo[3.2.1]oc...)copy SMILEScopy InChI
Affinity DataIC50: 137nMAssay Description:Competitive inhibition against [3H]cocaine binding to cocaine receptor in bovine striatal tissueMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2BG2PMNPubMed
TargetSodium-dependent dopamine transporter(BOVINE)
University of Maryland

Curated by ChEMBL
LigandPNGBDBM50015692(8-Methyl-3-(4-nitro-phenyl)-8-aza-bicyclo[3.2.1]oc...)copy SMILEScopy InChI
Affinity DataIC50: 137nMAssay Description:Competitive inhibition against [3H]cocaine binding to cocaine receptor in bovine striatal tissueMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2BG2PMNPubMed
TargetSodium-dependent dopamine transporter(BOVINE)
University of Maryland

Curated by ChEMBL
LigandPNGBDBM22418(Cocaine | Cocaine (-) | methyl (1R,2R,3S,5S)-3-(be...)copy SMILEScopy InChI
Affinity DataIC50: 139nMAssay Description:Competitive inhibition against [3H]cocaine binding to cocaine receptor in bovine striatal tissueMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2BG2PMNPubMed
TargetSodium-dependent dopamine transporter(BOVINE)
University of Maryland

Curated by ChEMBL
LigandPNGBDBM50015695(3-(4-Amino-phenyl)-8-methyl-8-aza-bicyclo[3.2.1]oc...)copy SMILEScopy InChI
Affinity DataIC50: 192nMAssay Description:Competitive inhibition against [3H]cocaine binding to cocaine receptor in bovine striatal tissueMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2BG2PMNPubMed
TargetSodium-dependent dopamine transporter(MOUSE)
Universit£ degli Studi di Urbino Carlo Bo

Curated by ChEMBL
LigandPNGBDBM22418(Cocaine | Cocaine (-) | methyl (1R,2R,3S,5S)-3-(be...)copy SMILEScopy InChI
Affinity DataIC50: 200nMAssay Description:Inhibition of mouse DAT expressed in HEK293 cells assessed as reduction in [3H]-DA uptakeMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Z60RBZPubMed
TargetSodium-dependent dopamine transporter(MOUSE)
Universit£ degli Studi di Urbino Carlo Bo

Curated by ChEMBL
LigandPNGBDBM50236804(CHEMBL4066973)copy SMILEScopy InChI
Affinity DataIC50: 940nMAssay Description:Inhibition of mouse DAT expressed in HEK293 cells assessed as reduction in [3H]-DA uptakeMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Z60RBZPubMed
TargetSodium-dependent dopamine transporter(BOVINE)
University of Maryland

Curated by ChEMBL
LigandPNGBDBM50011396(8-Methyl-3-(4-nitro-phenylcarbamoyloxy)-8-aza-bicy...)copy SMILEScopy InChI
Affinity DataIC50: 1.09E+3nMAssay Description:In vitro inhibitory activity towards [3H]cocaine binding to rat striatal tissueMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2X34Z21PubMed
TargetSodium-dependent dopamine transporter(MOUSE)
Universit£ degli Studi di Urbino Carlo Bo

Curated by ChEMBL
LigandPNGBDBM50236796(CHEMBL4093756)copy SMILEScopy InChI
Affinity DataIC50: 1.17E+3nMAssay Description:Inhibition of mouse DAT expressed in HEK293 cells assessed as reduction in [3H]-DA uptakeMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Z60RBZPubMed
TargetSodium-dependent dopamine transporter(BOVINE)
University of Maryland

Curated by ChEMBL
LigandPNGBDBM50011395(3-(3-Amino-phenylcarbamoyloxy)-8-methyl-8-aza-bicy...)copy SMILEScopy InChI
Affinity DataIC50: 2.07E+3nMAssay Description:In vitro inhibitory activity towards [3H]cocaine binding to rat striatal tissueMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2X34Z21PubMed
TargetSodium-dependent dopamine transporter(MOUSE)
Universit£ degli Studi di Urbino Carlo Bo

Curated by ChEMBL
LigandPNGBDBM50069812(CHEMBL3407784)copy SMILEScopy InChI
Affinity DataIC50: 2.29E+3nMAssay Description:Inhibition of mouse DAT expressed in HEK293 cells assessed as reduction in [3H]-DA uptakeMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Z60RBZPubMed
TargetSodium-dependent dopamine transporter(MOUSE)
Universit£ degli Studi di Urbino Carlo Bo

Curated by ChEMBL
LigandPNGBDBM50069813(CHEMBL3407785)copy SMILEScopy InChI
Affinity DataIC50: 3.26E+3nMAssay Description:Inhibition of mouse DAT expressed in HEK293 cells assessed as reduction in [3H]-DA uptakeMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Z60RBZPubMed
TargetSodium-dependent dopamine transporter(MOUSE)
Universit£ degli Studi di Urbino Carlo Bo

Curated by ChEMBL
LigandPNGBDBM50237600(CHEMBL4071867)copy SMILEScopy InChI
Affinity DataIC50: 4.30E+3nMAssay Description:Inhibition of mouse DAT expressed in HEK293 cells assessed as reduction in [3H]-DA uptakeMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Z60RBZPubMed
TargetSodium-dependent dopamine transporter(MOUSE)
Universit£ degli Studi di Urbino Carlo Bo

Curated by ChEMBL
LigandPNGBDBM50039246((S)-1-(2-(tris(4-methoxyphenyl)methoxy)ethyl)piper...)copy SMILEScopy InChI
Affinity DataIC50: 5.01E+3nMAssay Description:Inhibition of mouse GAT3 expressed in HEK293 cells by [3H]GABA uptake assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QR4ZTKPubMed
TargetSodium-dependent dopamine transporter(BOVINE)
University of Maryland

Curated by ChEMBL
LigandPNGBDBM50011394(8-Methyl-3-phenylcarbamoyloxy-8-aza-bicyclo[3.2.1]...)copy SMILEScopy InChI
Affinity DataIC50: 5.60E+3nMAssay Description:In vitro inhibitory activity towards [3H]cocaine binding to rat striatal tissueMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2X34Z21PubMed
TargetSodium-dependent dopamine transporter(BOVINE)
University of Maryland

Curated by ChEMBL
LigandPNGBDBM50015694(3-(2,4-Dinitro-phenyl)-8-methyl-8-aza-bicyclo[3.2....)copy SMILEScopy InChI
Affinity DataIC50: 1.10E+4nMAssay Description:Competitive inhibition against [3H]cocaine binding to cocaine receptor in bovine striatal tissueMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2BG2PMNPubMed
TargetSodium-dependent dopamine transporter(MOUSE)
Universit£ degli Studi di Urbino Carlo Bo

Curated by ChEMBL
LigandPNGBDBM50063514(CHEMBL3398504)copy SMILEScopy InChI
Affinity DataIC50: 1.15E+4nMAssay Description:Inhibition of mouse GAT3 expressed in HEK293 cells by [3H]GABA uptake assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QR4ZTKPubMed
TargetSodium-dependent dopamine transporter(MOUSE)
Universit£ degli Studi di Urbino Carlo Bo

Curated by ChEMBL
LigandPNGBDBM50063512(CHEMBL3398502)copy SMILEScopy InChI
Affinity DataIC50: 1.70E+4nMAssay Description:Inhibition of mouse GAT3 expressed in HEK293 cells by [3H]GABA uptake assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QR4ZTKPubMed
TargetSodium-dependent dopamine transporter(MOUSE)
Universit£ degli Studi di Urbino Carlo Bo

Curated by ChEMBL
LigandPNGBDBM50063513(CHEMBL3398496)copy SMILEScopy InChI
Affinity DataIC50: 2.69E+4nMAssay Description:Inhibition of mouse GAT3 expressed in HEK293 cells by [3H]GABA uptake assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QR4ZTKPubMed
TargetSodium-dependent dopamine transporter(MOUSE)
Universit£ degli Studi di Urbino Carlo Bo

Curated by ChEMBL
LigandPNGBDBM50063500(CHEMBL3398506)copy SMILEScopy InChI
Affinity DataIC50: 3.02E+4nMAssay Description:Inhibition of mouse GAT3 expressed in HEK293 cells by [3H]GABA uptake assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QR4ZTKPubMed
TargetSodium-dependent dopamine transporter(MOUSE)
Universit£ degli Studi di Urbino Carlo Bo

Curated by ChEMBL
LigandPNGBDBM50063510(CHEMBL3398494)copy SMILEScopy InChI
Affinity DataIC50: 3.63E+4nMAssay Description:Inhibition of mouse GAT3 expressed in HEK293 cells by [3H]GABA uptake assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QR4ZTKPubMed
TargetSodium-dependent dopamine transporter(MOUSE)
Universit£ degli Studi di Urbino Carlo Bo

Curated by ChEMBL
LigandPNGBDBM50063498(CHEMBL3398501)copy SMILEScopy InChI
Affinity DataIC50: 4.27E+4nMAssay Description:Inhibition of mouse GAT3 expressed in HEK293 cells by [3H]GABA uptake assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QR4ZTKPubMed
TargetSodium-dependent dopamine transporter(BOVINE)
University of Maryland

Curated by ChEMBL
LigandPNGBDBM50011398(3-(4-Amino-phenylcarbamoyloxy)-8-methyl-8-aza-bicy...)copy SMILEScopy InChI
Affinity DataIC50: 6.33E+4nMAssay Description:In vitro inhibitory activity towards [3H]cocaine binding to rat striatal tissueMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2X34Z21PubMed
TargetSodium-dependent dopamine transporter(MOUSE)
Universit£ degli Studi di Urbino Carlo Bo

Curated by ChEMBL
LigandPNGBDBM50063503(CHEMBL3398499)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of mouse GAT3 expressed in HEK293 cells by [3H]GABA uptake assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QR4ZTKPubMed
TargetSodium-dependent dopamine transporter(MOUSE)
Universit£ degli Studi di Urbino Carlo Bo

Curated by ChEMBL
LigandPNGBDBM50063509((S)-Homoproline | CHEMBL1164855)copy SMILEScopy InChI
Affinity DataIC50: 1.41E+5nMAssay Description:Inhibition of mouse GAT3 expressed in HEK293 cells by [3H]GABA uptake assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QR4ZTKPubMed
TargetSodium-dependent dopamine transporter(MOUSE)
Universit£ degli Studi di Urbino Carlo Bo

Curated by ChEMBL
LigandPNGBDBM50063502(CHEMBL3398495)copy SMILEScopy InChI
Affinity DataIC50: 2.69E+5nMAssay Description:Inhibition of mouse GAT3 expressed in HEK293 cells by [3H]GABA uptake assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QR4ZTKPubMed
TargetSodium-dependent dopamine transporter(MOUSE)
Universit£ degli Studi di Urbino Carlo Bo

Curated by ChEMBL
LigandPNGBDBM50063501(CHEMBL3398490)copy SMILEScopy InChI
Affinity DataIC50: 3.09E+5nMAssay Description:Inhibition of mouse GAT3 expressed in HEK293 cells by [3H]GABA uptake assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QR4ZTKPubMed
TargetSodium-dependent dopamine transporter(MOUSE)
Universit£ degli Studi di Urbino Carlo Bo

Curated by ChEMBL
LigandPNGBDBM50063499((R)-Homoproline | CHEMBL1163348)copy SMILEScopy InChI
Affinity DataIC50: 3.39E+5nMAssay Description:Inhibition of mouse GAT3 expressed in HEK293 cells by [3H]GABA uptake assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QR4ZTKPubMed