TargetSodium-dependent dopamine transporter(MOUSE)
Universit£ degli Studi di Urbino Carlo Bo
Curated by ChEMBL
Universit£ degli Studi di Urbino Carlo Bo
Curated by ChEMBL
Affinity DataIC50: 5nMAssay Description:Inhibitory concentration against human Adenosine A3 receptor expressed in HEK293 cells using 0.1 nM [3H]AB-MECAMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(MOUSE)
Universit£ degli Studi di Urbino Carlo Bo
Curated by ChEMBL
Universit£ degli Studi di Urbino Carlo Bo
Curated by ChEMBL
Affinity DataIC50: 13nMAssay Description:Inhibition of mouse DAT expressed in HEK293 cells assessed as reduction in [3H]-DA uptakeMore data for this Ligand-Target Pair
Affinity DataIC50: 22nMAssay Description:Competitive inhibition against [3H]cocaine binding to cocaine receptor in bovine striatal tissueMore data for this Ligand-Target Pair
Affinity DataIC50: 22nMAssay Description:Competitive inhibition against [3H]cocaine binding to cocaine receptor in bovine striatal tissueMore data for this Ligand-Target Pair
Affinity DataIC50: 37nMAssay Description:In vitro inhibitory activity towards [3H]cocaine binding to rat striatal tissueMore data for this Ligand-Target Pair
Affinity DataIC50: 65nMAssay Description:In vitro inhibitory activity towards [3H]cocaine binding to rat striatal tissueMore data for this Ligand-Target Pair
Affinity DataIC50: 137nMAssay Description:Competitive inhibition against [3H]cocaine binding to cocaine receptor in bovine striatal tissueMore data for this Ligand-Target Pair
Affinity DataIC50: 137nMAssay Description:Competitive inhibition against [3H]cocaine binding to cocaine receptor in bovine striatal tissueMore data for this Ligand-Target Pair
Affinity DataIC50: 139nMAssay Description:Competitive inhibition against [3H]cocaine binding to cocaine receptor in bovine striatal tissueMore data for this Ligand-Target Pair
Affinity DataIC50: 192nMAssay Description:Competitive inhibition against [3H]cocaine binding to cocaine receptor in bovine striatal tissueMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(MOUSE)
Universit£ degli Studi di Urbino Carlo Bo
Curated by ChEMBL
Universit£ degli Studi di Urbino Carlo Bo
Curated by ChEMBL
Affinity DataIC50: 200nMAssay Description:Inhibition of mouse DAT expressed in HEK293 cells assessed as reduction in [3H]-DA uptakeMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(MOUSE)
Universit£ degli Studi di Urbino Carlo Bo
Curated by ChEMBL
Universit£ degli Studi di Urbino Carlo Bo
Curated by ChEMBL
Affinity DataIC50: 940nMAssay Description:Inhibition of mouse DAT expressed in HEK293 cells assessed as reduction in [3H]-DA uptakeMore data for this Ligand-Target Pair
Affinity DataIC50: 1.09E+3nMAssay Description:In vitro inhibitory activity towards [3H]cocaine binding to rat striatal tissueMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(MOUSE)
Universit£ degli Studi di Urbino Carlo Bo
Curated by ChEMBL
Universit£ degli Studi di Urbino Carlo Bo
Curated by ChEMBL
Affinity DataIC50: 1.17E+3nMAssay Description:Inhibition of mouse DAT expressed in HEK293 cells assessed as reduction in [3H]-DA uptakeMore data for this Ligand-Target Pair
Affinity DataIC50: 2.07E+3nMAssay Description:In vitro inhibitory activity towards [3H]cocaine binding to rat striatal tissueMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(MOUSE)
Universit£ degli Studi di Urbino Carlo Bo
Curated by ChEMBL
Universit£ degli Studi di Urbino Carlo Bo
Curated by ChEMBL
Affinity DataIC50: 2.29E+3nMAssay Description:Inhibition of mouse DAT expressed in HEK293 cells assessed as reduction in [3H]-DA uptakeMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(MOUSE)
Universit£ degli Studi di Urbino Carlo Bo
Curated by ChEMBL
Universit£ degli Studi di Urbino Carlo Bo
Curated by ChEMBL
Affinity DataIC50: 3.26E+3nMAssay Description:Inhibition of mouse DAT expressed in HEK293 cells assessed as reduction in [3H]-DA uptakeMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(MOUSE)
Universit£ degli Studi di Urbino Carlo Bo
Curated by ChEMBL
Universit£ degli Studi di Urbino Carlo Bo
Curated by ChEMBL
Affinity DataIC50: 4.30E+3nMAssay Description:Inhibition of mouse DAT expressed in HEK293 cells assessed as reduction in [3H]-DA uptakeMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(MOUSE)
Universit£ degli Studi di Urbino Carlo Bo
Curated by ChEMBL
Universit£ degli Studi di Urbino Carlo Bo
Curated by ChEMBL
Affinity DataIC50: 5.01E+3nMAssay Description:Inhibition of mouse GAT3 expressed in HEK293 cells by [3H]GABA uptake assayMore data for this Ligand-Target Pair
Affinity DataIC50: 5.60E+3nMAssay Description:In vitro inhibitory activity towards [3H]cocaine binding to rat striatal tissueMore data for this Ligand-Target Pair
Affinity DataIC50: 1.10E+4nMAssay Description:Competitive inhibition against [3H]cocaine binding to cocaine receptor in bovine striatal tissueMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(MOUSE)
Universit£ degli Studi di Urbino Carlo Bo
Curated by ChEMBL
Universit£ degli Studi di Urbino Carlo Bo
Curated by ChEMBL
Affinity DataIC50: 1.15E+4nMAssay Description:Inhibition of mouse GAT3 expressed in HEK293 cells by [3H]GABA uptake assayMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(MOUSE)
Universit£ degli Studi di Urbino Carlo Bo
Curated by ChEMBL
Universit£ degli Studi di Urbino Carlo Bo
Curated by ChEMBL
Affinity DataIC50: 1.70E+4nMAssay Description:Inhibition of mouse GAT3 expressed in HEK293 cells by [3H]GABA uptake assayMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(MOUSE)
Universit£ degli Studi di Urbino Carlo Bo
Curated by ChEMBL
Universit£ degli Studi di Urbino Carlo Bo
Curated by ChEMBL
Affinity DataIC50: 2.69E+4nMAssay Description:Inhibition of mouse GAT3 expressed in HEK293 cells by [3H]GABA uptake assayMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(MOUSE)
Universit£ degli Studi di Urbino Carlo Bo
Curated by ChEMBL
Universit£ degli Studi di Urbino Carlo Bo
Curated by ChEMBL
Affinity DataIC50: 3.02E+4nMAssay Description:Inhibition of mouse GAT3 expressed in HEK293 cells by [3H]GABA uptake assayMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(MOUSE)
Universit£ degli Studi di Urbino Carlo Bo
Curated by ChEMBL
Universit£ degli Studi di Urbino Carlo Bo
Curated by ChEMBL
Affinity DataIC50: 3.63E+4nMAssay Description:Inhibition of mouse GAT3 expressed in HEK293 cells by [3H]GABA uptake assayMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(MOUSE)
Universit£ degli Studi di Urbino Carlo Bo
Curated by ChEMBL
Universit£ degli Studi di Urbino Carlo Bo
Curated by ChEMBL
Affinity DataIC50: 4.27E+4nMAssay Description:Inhibition of mouse GAT3 expressed in HEK293 cells by [3H]GABA uptake assayMore data for this Ligand-Target Pair
Affinity DataIC50: 6.33E+4nMAssay Description:In vitro inhibitory activity towards [3H]cocaine binding to rat striatal tissueMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(MOUSE)
Universit£ degli Studi di Urbino Carlo Bo
Curated by ChEMBL
Universit£ degli Studi di Urbino Carlo Bo
Curated by ChEMBL
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of mouse GAT3 expressed in HEK293 cells by [3H]GABA uptake assayMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(MOUSE)
Universit£ degli Studi di Urbino Carlo Bo
Curated by ChEMBL
Universit£ degli Studi di Urbino Carlo Bo
Curated by ChEMBL
Affinity DataIC50: 1.41E+5nMAssay Description:Inhibition of mouse GAT3 expressed in HEK293 cells by [3H]GABA uptake assayMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(MOUSE)
Universit£ degli Studi di Urbino Carlo Bo
Curated by ChEMBL
Universit£ degli Studi di Urbino Carlo Bo
Curated by ChEMBL
Affinity DataIC50: 2.69E+5nMAssay Description:Inhibition of mouse GAT3 expressed in HEK293 cells by [3H]GABA uptake assayMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(MOUSE)
Universit£ degli Studi di Urbino Carlo Bo
Curated by ChEMBL
Universit£ degli Studi di Urbino Carlo Bo
Curated by ChEMBL
Affinity DataIC50: 3.09E+5nMAssay Description:Inhibition of mouse GAT3 expressed in HEK293 cells by [3H]GABA uptake assayMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(MOUSE)
Universit£ degli Studi di Urbino Carlo Bo
Curated by ChEMBL
Universit£ degli Studi di Urbino Carlo Bo
Curated by ChEMBL
Affinity DataIC50: 3.39E+5nMAssay Description:Inhibition of mouse GAT3 expressed in HEK293 cells by [3H]GABA uptake assayMore data for this Ligand-Target Pair