Compile Data Set for Download or QSAR
Found 386 of ec50 data for polymerid = 9460
TargetLysophosphatidic acid receptor 1(Homo sapiens (Human))TBA
LigandPNGUS11912686, Compound 314(Preparation of (R)-1-(2,5-difluoropyridin-3-yl)eth...)
Affinity DataEC50:  2.90nMMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails
TargetLysophosphatidic acid receptor 1(Homo sapiens (Human))TBA
Affinity DataEC50:  5nMMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails
TargetLysophosphatidic acid receptor 1(Homo sapiens (Human))TBA
Affinity DataEC50:  5.20nMMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails
TargetLysophosphatidic acid receptor 1(Homo sapiens (Human))TBA
Affinity DataEC50:  7.30nMMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails
TargetLysophosphatidic acid receptor 1(Homo sapiens (Human))TBA
Affinity DataEC50:  8.30nMMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails
TargetLysophosphatidic acid receptor 1(Homo sapiens (Human))TBA
LigandPNGBDBM50430006(CHEMBL2335048)copy SMILEScopy InChI
Affinity DataEC50:  8.40nMAssay Description:Agonist activity at human LPA1 receptor transfected in HEK293 cells after 1 hr by TGFalpha shedding assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2SN0B9GPubMed
TargetLysophosphatidic acid receptor 1(Homo sapiens (Human))TBA
Affinity DataEC50:  8.60nMMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails
TargetLysophosphatidic acid receptor 1(Homo sapiens (Human))TBA
LigandPNGUS11912686, Compound 318(Preparation of (R)-1-(2-chloropyridin-3-yl)ethyl (...)
Affinity DataEC50:  9.5nMMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails
TargetLysophosphatidic acid receptor 1(Homo sapiens (Human))TBA
LigandPNGBDBM50430010(CHEMBL2335047)copy SMILEScopy InChI
Affinity DataEC50:  10nMAssay Description:Agonist activity at human LPA1 receptor transfected in HEK293 cells after 1 hr by TGFalpha shedding assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2SN0B9GPubMed
TargetLysophosphatidic acid receptor 1(Homo sapiens (Human))TBA
Affinity DataEC50:  10.9nMMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails
TargetLysophosphatidic acid receptor 1(Homo sapiens (Human))TBA
LigandPNGBDBM50430008(CHEMBL2335050)copy SMILEScopy InChI
Affinity DataEC50:  11nMAssay Description:Agonist activity at human LPA1 receptor transfected in HEK293 cells after 1 hr by TGFalpha shedding assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2SN0B9GPubMed
TargetLysophosphatidic acid receptor 1(Homo sapiens (Human))TBA
Affinity DataEC50:  11.2nMMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails
TargetLysophosphatidic acid receptor 1(Homo sapiens (Human))TBA
Affinity DataEC50:  11.7nMMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails
TargetLysophosphatidic acid receptor 1(Homo sapiens (Human))TBA
Affinity DataEC50:  11.9nMMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails
TargetLysophosphatidic acid receptor 1(Homo sapiens (Human))TBA
LigandPNGBDBM50430007(CHEMBL2335051)copy SMILEScopy InChI
Affinity DataEC50:  12nMAssay Description:Agonist activity at human LPA1 receptor transfected in HEK293 cells after 1 hr by TGFalpha shedding assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2SN0B9GPubMed
TargetLysophosphatidic acid receptor 1(Homo sapiens (Human))TBA
LigandPNGUS11912686, Compound 315(Preparation of (R)-1-(2-chloropyridin-3-yl)ethyl (...)
Affinity DataEC50:  12.7nMMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails
TargetLysophosphatidic acid receptor 1(Homo sapiens (Human))TBA
Affinity DataEC50:  13nMMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails
TargetLysophosphatidic acid receptor 1(Homo sapiens (Human))TBA
Affinity DataEC50:  14.5nMMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails
TargetLysophosphatidic acid receptor 1(Homo sapiens (Human))TBA
LigandPNGBDBM50430012(CHEMBL357053)copy SMILEScopy InChI
Affinity DataEC50:  15nMAssay Description:Agonist activity at human LPA1 receptor transfected in HEK293 cells after 1 hr by TGFalpha shedding assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2SN0B9GPubMed
TargetLysophosphatidic acid receptor 1(Homo sapiens (Human))TBA
Affinity DataEC50:  16nMMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails
TargetLysophosphatidic acid receptor 1(Homo sapiens (Human))TBA
Affinity DataEC50:  16.1nMMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails
TargetLysophosphatidic acid receptor 1(Homo sapiens (Human))TBA
Affinity DataEC50:  16.2nMMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails
TargetLysophosphatidic acid receptor 1(Homo sapiens (Human))TBA
Affinity DataEC50:  16.3nMMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails
TargetLysophosphatidic acid receptor 1(Homo sapiens (Human))TBA
Affinity DataEC50:  16.6nMMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails
TargetLysophosphatidic acid receptor 1(Homo sapiens (Human))TBA
Affinity DataEC50:  16.6nMMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails
TargetLysophosphatidic acid receptor 1(Homo sapiens (Human))TBA
LigandPNGBDBM50381022(CHEMBL2017139)copy SMILEScopy InChI
Affinity DataEC50:  17nMAssay Description:Agonist activity at human LPA1 receptor transfected in HEK293 cells after 1 hr by TGFalpha shedding assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2SN0B9GPubMed
TargetLysophosphatidic acid receptor 1(Homo sapiens (Human))TBA
Affinity DataEC50:  17nMMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails
TargetLysophosphatidic acid receptor 1(Homo sapiens (Human))TBA
LigandPNGBDBM50148348((R)-Octadec-9-enoic acid 2-hydroxy-3-phosphonooxy-...)copy SMILEScopy InChI
Affinity DataEC50:  17nMAssay Description:Agonistic activity against lysophosphatidic acid receptor 1 using [35S]-GTP-gammaS as radioligand tested in vitroMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2D50MDWPubMed
TargetLysophosphatidic acid receptor 1(Homo sapiens (Human))TBA
Affinity DataEC50:  17.3nMMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails
TargetLysophosphatidic acid receptor 1(Homo sapiens (Human))TBA
Affinity DataEC50:  17.7nMMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails
TargetLysophosphatidic acid receptor 1(Homo sapiens (Human))TBA
LigandPNGBDBM50148348((R)-Octadec-9-enoic acid 2-hydroxy-3-phosphonooxy-...)copy SMILEScopy InChI
Affinity DataEC50:  18nMAssay Description:Agonist activity at human LPA1 receptor transfected in HEK293 cells after 1 hr by TGFalpha shedding assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2SN0B9GPubMed
TargetLysophosphatidic acid receptor 1(Homo sapiens (Human))TBA
Affinity DataEC50:  18.1nMMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails
TargetLysophosphatidic acid receptor 1(Homo sapiens (Human))TBA
Affinity DataEC50:  19.1nMMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails
TargetLysophosphatidic acid receptor 1(Homo sapiens (Human))TBA
Affinity DataEC50:  19.3nMMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails
TargetLysophosphatidic acid receptor 1(Homo sapiens (Human))TBA
Affinity DataEC50:  19.3nMMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails
TargetLysophosphatidic acid receptor 1(Homo sapiens (Human))TBA
Affinity DataEC50:  19.5nMMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails
TargetLysophosphatidic acid receptor 1(Homo sapiens (Human))TBA
Affinity DataEC50:  20.4nMMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails
TargetLysophosphatidic acid receptor 1(Homo sapiens (Human))TBA
Affinity DataEC50:  21.1nMMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails
TargetLysophosphatidic acid receptor 1(Homo sapiens (Human))TBA
Affinity DataEC50:  21.5nMMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails
TargetLysophosphatidic acid receptor 1(Homo sapiens (Human))TBA
Affinity DataEC50:  22.4nMMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails
TargetLysophosphatidic acid receptor 1(Homo sapiens (Human))TBA
Affinity DataEC50:  22.8nMMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails
TargetLysophosphatidic acid receptor 1(Homo sapiens (Human))TBA
Affinity DataEC50:  22.8nMMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails
TargetLysophosphatidic acid receptor 1(Homo sapiens (Human))TBA
Affinity DataEC50:  22.8nMMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails
TargetLysophosphatidic acid receptor 1(Homo sapiens (Human))TBA
Affinity DataEC50:  23.4nMMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails
TargetLysophosphatidic acid receptor 1(Homo sapiens (Human))TBA
Affinity DataEC50:  23.7nMMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails
TargetLysophosphatidic acid receptor 1(Homo sapiens (Human))TBA
LigandPNGBDBM50430011(CHEMBL153043)copy SMILEScopy InChI
Affinity DataEC50:  24nMAssay Description:Agonist activity at human LPA1 receptor transfected in HEK293 cells after 1 hr by TGFalpha shedding assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2SN0B9GPubMed
TargetLysophosphatidic acid receptor 1(Homo sapiens (Human))TBA
Affinity DataEC50:  24nMMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails
TargetLysophosphatidic acid receptor 1(Homo sapiens (Human))TBA
Affinity DataEC50:  25.5nMMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails
TargetLysophosphatidic acid receptor 1(Homo sapiens (Human))TBA
LigandPNGBDBM50430009(CHEMBL2335049)copy SMILEScopy InChI
Affinity DataEC50:  26nMAssay Description:Agonist activity at human LPA1 receptor transfected in HEK293 cells after 1 hr by TGFalpha shedding assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2SN0B9GPubMed
TargetLysophosphatidic acid receptor 1(Homo sapiens (Human))TBA
Affinity DataEC50:  26.5nMMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails
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