Compile Data Set for Download or QSAR
Found 37 of ic50 data for polymerid = 2395
LigandPNGBDBM50590284(CHEMBL5192316)copy SMILES
Affinity DataIC50: 10nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27S7SQ9PubMed
LigandPNGBDBM50590283(CHEMBL5169766 | US20230303547, Reference Example D)copy SMILES
Affinity DataIC50: 10nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27S7SQ9PubMed
LigandPNGBDBM50431630(KRX-0401 | PERIFOSINE)copy SMILEScopy InChI
Affinity DataIC50: 50nMMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BV7MNZPubMed
LigandPNGBDBM53421(4-Cyclohexyl-2-phenyl-quinazoline | 4-cyclohexyl-2...)copy SMILEScopy InChI
Affinity DataIC50: 600nMAssay Description:Inhibition of UCHL3 in human H1299 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KW5G7PPubMed
LigandPNGBDBM50594731(CHEMBL1241028)copy SMILES
Affinity DataIC50: 600nMMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BV7MNZPubMed
LigandPNGBDBM50069764(CHEMBL3407501)copy SMILEScopy InChI
Affinity DataIC50: 2.16E+3nMMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BV7MNZPubMed
LigandPNGBDBM50594730(CHEMBL5193983)copy SMILES
Affinity DataIC50: 5.00E+3nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BV7MNZPubMed
LigandPNGBDBM50594729(CHEBI:27485 | CHEMBL1397260)copy SMILES
Affinity DataIC50: 1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BV7MNZPubMed
LigandPNGBDBM50538571(CHEMBL4635160)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human GST-tagged UCHL3 expressed in Escherichia coli assessed as cleavage of Ubiquitin-Rhodamine110-glycine to Ubiquitin and Rhodamine1...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2XK8K2TPubMed
LigandPNGBDBM65518(5-Chloro-1-[(2,5-dichlorophenyl)methyl]-1H-indole-...)copy SMILEScopy InChI
Affinity DataIC50: 1.41E+4nMpH: 7.5 T: 2°CAssay Description:Ubiquitin-7-amino-4-methylcoumarin (Ub-AMC) was generated as previously described.(7) The enzymatic reaction was conducted in fluorometric assay buff...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21J97WDPubMed
LigandPNGBDBM50442907(Acetyl Isogambogic Acid | CHEMBL3039433)copy SMILEScopy InChI
Affinity DataIC50: 1.54E+4nMpH: 7.5 T: 2°CAssay Description:Ubiquitin-7-amino-4-methylcoumarin (Ub-AMC) was generated as previously described.(7) The enzymatic reaction was conducted in fluorometric assay buff...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21J97WDPubMed
LigandPNGBDBM50326012(3-(acetoxyimino)-5-bromo-1-(3,4-dichlorobenzyl)ind...)copy SMILEScopy InChI
Affinity DataIC50: 1.70E+4nMAssay Description:Inhibition of UCHL3 in human H1299 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KW5G7PPubMed
LigandPNGBDBM50326014(3-(acetoxyimino)-1-(3,4-dichlorobenzyl)-5-iodoindo...)copy SMILEScopy InChI
Affinity DataIC50: 2.30E+4nMAssay Description:Inhibition of UCHL3 in human H1299 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KW5G7PPubMed
LigandPNGBDBM200235(Rifampicin | cid_5381226)copy SMILEScopy InChI
Affinity DataIC50: 2.48E+4nMpH: 7.5 T: 2°CAssay Description:Ubiquitin-7-amino-4-methylcoumarin (Ub-AMC) was generated as previously described.(7) The enzymatic reaction was conducted in fluorometric assay buff...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21J97WDPubMed
LigandPNGBDBM50594733(CHEMBL4303698)copy SMILES
Affinity DataIC50: 2.50E+4nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BV7MNZPubMed
LigandPNGBDBM50326013(3-(acetoxyimino)-5-bromo-1-(2,5-dichlorobenzyl)ind...)copy SMILEScopy InChI
Affinity DataIC50: 2.50E+4nMAssay Description:Inhibition of UCHL3 in human H1299 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KW5G7PPubMed
LigandPNGBDBM205457((2R,4aS,6aR,6aS,14aS,14bR)-10-hydroxy-2,4a,6a,6a,9...)copy SMILEScopy InChI
Affinity DataIC50: 3.21E+4nMpH: 7.5 T: 2°CAssay Description:Ubiquitin-7-amino-4-methylcoumarin (Ub-AMC) was generated as previously described.(7) The enzymatic reaction was conducted in fluorometric assay buff...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21J97WDPubMed
LigandPNGBDBM50326015(5-(4-butylphenyl)-4-(4-isopropylphenyl)-4H-1,2,4-t...)copy SMILEScopy InChI
Affinity DataIC50: 4.70E+4nMAssay Description:Inhibition of UCHL3 in human H1299 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KW5G7PPubMed
LigandPNGBDBM50594732(CHEMBL5195092)copy SMILES
Affinity DataIC50: 4.70E+4nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BV7MNZPubMed
LigandPNGBDBM50242207(CHEMBL455364 | Mangiferin)copy SMILEScopy InChI
Affinity DataIC50: 5.26E+4nMpH: 7.5 T: 2°CAssay Description:Ubiquitin-7-amino-4-methylcoumarin (Ub-AMC) was generated as previously described.(7) The enzymatic reaction was conducted in fluorometric assay buff...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21J97WDPubMed
LigandPNGBDBM24778(2-methyl-1,4-dihydronaphthalene-1,4-dione | 2-meth...)copy SMILEScopy InChI
Affinity DataIC50: 7.10E+4nMAssay Description:Inhibition of UCHL3 in human H1299 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KW5G7PPubMed
LigandPNGBDBM24778(2-methyl-1,4-dihydronaphthalene-1,4-dione | 2-meth...)copy SMILEScopy InChI
Affinity DataIC50: 7.10E+4nMMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BV7MNZPubMed
LigandPNGBDBM50552483(CHEMBL4763594)copy SMILES
Affinity DataIC50: 7.40E+4nMAssay Description:Inhibition of recombinant human UCHL3 assessed as reduction in cleavage of Ubiquitin-Rhodamine110-glycine to Ubiquitin and Rhodamine110-glycine using...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2R49VFDPubMed
LigandPNGBDBM50538549(CHEMBL4641424)copy SMILEScopy InChI
Affinity DataIC50: 8.00E+4nMAssay Description:Inhibition of human GST-tagged UCHL3 expressed in Escherichia coli assessed as cleavage of Ubiquitin-Rhodamine110-glycine to Ubiquitin and Rhodamine1...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2XK8K2TPubMed
LigandPNGBDBM50270667(CHEMBL4130194)copy SMILEScopy InChI
Affinity DataIC50: 8.00E+4nMAssay Description:Inhibition of human GST-tagged UCHL3 expressed in Escherichia coli assessed as cleavage of Ubiquitin-Rhodamine110-glycine to Ubiquitin and Rhodamine1...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2XK8K2TPubMed
LigandPNGBDBM23421(1-benzyl-3-hydroxy-4-[(5-methylfuran-2-yl)carbonyl...)copy SMILEScopy InChI
Affinity DataIC50: 1.03E+5nMpH: 7.8 T: 2°CAssay Description:Enzyme reactions were carried out on Costar 96-well black assay plates. After the reaction, AMC fluorescence (excitation wavelength: 355 nm, emission...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ZK5DZKPubMed
LigandPNGBDBM50069762(CHEMBL3182437 | ML323 | US9802904, 87)copy SMILEScopy InChI
Affinity DataIC50: 1.14E+5nMpH: 7.5 T: 2°CAssay Description:Ubiquitin-7-amino-4-methylcoumarin (Ub-AMC) was generated as previously described.(7) The enzymatic reaction was conducted in fluorometric assay buff...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21J97WDPubMed
LigandPNGBDBM65524((-)-Aricine | Heterophylline (VAN) | Quinovatine)copy SMILEScopy InChI
Affinity DataIC50: 1.14E+5nMpH: 7.5 T: 2°CAssay Description:Ubiquitin-7-amino-4-methylcoumarin (Ub-AMC) was generated as previously described.(7) The enzymatic reaction was conducted in fluorometric assay buff...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21J97WDPubMed
LigandPNGBDBM23427(5-(4-fluorophenyl)-3-hydroxy-4-[(5-methylfuran-2-y...)copy SMILEScopy InChI
Affinity DataIC50: 1.23E+5nMpH: 7.8 T: 2°CAssay Description:Enzyme reactions were carried out on Costar 96-well black assay plates. After the reaction, AMC fluorescence (excitation wavelength: 355 nm, emission...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ZK5DZKPubMed
LigandPNGBDBM23426(3-hydroxy-5-(4-methoxyphenyl)-1-(1,3,4-thiadiazol-...)copy SMILEScopy InChI
Affinity DataIC50: 1.54E+5nMpH: 7.8 T: 2°CAssay Description:Enzyme reactions were carried out on Costar 96-well black assay plates. After the reaction, AMC fluorescence (excitation wavelength: 355 nm, emission...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ZK5DZKPubMed
LigandPNGBDBM50271098(CHEMBL4129140)copy SMILEScopy InChI
Affinity DataIC50: 2.00E+5nMAssay Description:Inhibition of UCH-L3 (unknown origin) using Ub-AMC as substrate preincubated for 30 mins followed by substrate addition measured after 60 mins by flu...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CR5WVGPubMed
LigandPNGBDBM50608424(CHEMBL5267683)copy SMILES
Affinity DataIC50: 2.00E+5nMMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails
LigandPNGBDBM23425(ChemBridge CNS-Set 7909542, 5 | N-{3-[1-acetyl-5-(...)copy SMILEScopy InChI
Affinity DataIC50: 3.31E+5nMpH: 7.8 T: 2°CAssay Description:Enzyme reactions were carried out on Costar 96-well black assay plates. After the reaction, AMC fluorescence (excitation wavelength: 355 nm, emission...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ZK5DZKPubMed
LigandPNGBDBM23424(ChemBridge CNS-Set 6382507, 4 | N-cyclopropyl-2-[(...)copy SMILEScopy InChI
Affinity DataIC50: 3.34E+5nMpH: 7.8 T: 2°CAssay Description:Enzyme reactions were carried out on Costar 96-well black assay plates. After the reaction, AMC fluorescence (excitation wavelength: 355 nm, emission...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ZK5DZKPubMed
LigandPNGBDBM23429(2-[benzene(3-methoxyphenyl)sulfonamido]-N-cyclopen...)copy SMILEScopy InChI
Affinity DataIC50: 3.86E+5nMpH: 7.8 T: 2°CAssay Description:Enzyme reactions were carried out on Costar 96-well black assay plates. After the reaction, AMC fluorescence (excitation wavelength: 355 nm, emission...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ZK5DZKPubMed
LigandPNGBDBM23430(4-({[5-(furan-2-yl)-4-phenyl-4H-1,2,4-triazol-3-yl...)copy SMILEScopy InChI
Affinity DataIC50: 3.87E+5nMpH: 7.8 T: 2°CAssay Description:Enzyme reactions were carried out on Costar 96-well black assay plates. After the reaction, AMC fluorescence (excitation wavelength: 355 nm, emission...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ZK5DZKPubMed
LigandPNGBDBM23428(ChemBridge CNS-Set 6699002, 8 | N-cyclopropyl-2-[(...)copy SMILEScopy InChI
Affinity DataIC50: 4.01E+5nMpH: 7.8 T: 2°CAssay Description:Enzyme reactions were carried out on Costar 96-well black assay plates. After the reaction, AMC fluorescence (excitation wavelength: 355 nm, emission...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ZK5DZKPubMed