Compile Data Set for Download or QSAR
Found 665 of ic50 data for polymerid = 4601,4602
TargetGlycylpeptide N-tetradecanoyltransferase(Candida albicans (Yeast))
Second Military Medical University

Curated by ChEMBL
LigandPNGBDBM50121716((3-methyl-4-(3-(pyridin-3-ylmethylamino)propoxy)be...)copy SMILEScopy InChI
Affinity DataIC50: 0.390nMAssay Description:Inhibition of Candida albicans N-myristoyltransferseMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2RV0ND9PubMed
TargetGlycylpeptide N-tetradecanoyltransferase(Candida albicans (Yeast))
Second Military Medical University

Curated by ChEMBL
LigandPNGBDBM50121716((3-methyl-4-(3-(pyridin-3-ylmethylamino)propoxy)be...)copy SMILEScopy InChI
Affinity DataIC50: 0.390nMAssay Description:Inhibition of Candida albicans N-myristoyltransferseMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2RV0ND9PubMed
TargetGlycylpeptide N-tetradecanoyltransferase(Candida albicans (Yeast))
Second Military Medical University

Curated by ChEMBL
LigandPNGBDBM50457393(CHEMBL3220375)copy SMILEScopy InChI
Affinity DataIC50: 0.490nMAssay Description:Inhibition of Candida albicans ATCC 90028 NMT using GLTISKLFRR-NH2 as substrate assessed as reduction in [3H]-myristoylated peptide reaction product ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26112X4PubMed
TargetGlycylpeptide N-tetradecanoyltransferase(Candida albicans (Yeast))
Second Military Medical University

Curated by ChEMBL
LigandPNGBDBM50207643((1S,3R)-N-(2-(cyclopentanecarboxamido)benzo[d]thia...)copy SMILEScopy InChI
Affinity DataIC50: 0.490nMAssay Description:Inhibition of Candida albicans N-myristoyltransferseMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2RV0ND9PubMed
TargetGlycylpeptide N-tetradecanoyltransferase(Candida albicans (Yeast))
Second Military Medical University

Curated by ChEMBL
LigandPNGBDBM50207643((1S,3R)-N-(2-(cyclopentanecarboxamido)benzo[d]thia...)copy SMILEScopy InChI
Affinity DataIC50: 0.490nMAssay Description:Inhibition of Candida albicans N-myristoyltransferseMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2RV0ND9PubMed
TargetGlycylpeptide N-tetradecanoyltransferase 1(Homo sapiens (Human))
Frontier Medicines

Curated by ChEMBL
LigandPNGBDBM50520331(CHEMBL4445137)copy SMILEScopy InChI
Affinity DataIC50: 1nMAssay Description:Inhibition of human N-myristoyltransferase assessed as reduction in CoASH production by fluorogenic detection based assayMore data for this Ligand-Target Pair
TargetGlycylpeptide N-tetradecanoyltransferase(Candida albicans (Yeast))
Second Military Medical University

Curated by ChEMBL
LigandPNGBDBM50121720((1-METHYL-1H-IMIDAZOL-2-YL)-(3-METHYL-4-{3-[(PYRID...)copy SMILEScopy InChI
Affinity DataIC50: 1nMAssay Description:Inhibition activity against C. albicans Nmt and human Nmt as assessed by IC50 using myristoyl-CoA (0.5 uM) and peptide substrate GLTISKLFRR-NH2 (0.5 ...More data for this Ligand-Target Pair
TargetGlycylpeptide N-tetradecanoyltransferase 1(Homo sapiens (Human))
Frontier Medicines

Curated by ChEMBL
LigandPNGBDBM50520331(CHEMBL4445137)copy SMILEScopy InChI
Affinity DataIC50: 1nMAssay Description:Inhibition of human NMT1 by fluorescence methodMore data for this Ligand-Target Pair
TargetGlycylpeptide N-tetradecanoyltransferase 1(Homo sapiens (Human))
Frontier Medicines

Curated by ChEMBL
LigandPNGBDBM185107(US9156811, DDD100868)copy SMILEScopy InChI
Affinity DataIC50: 2nMpH: 7.4 T: 2°CAssay Description:Measurement of the ability of compounds to inhibit the NMT-1 and/or NMT-2 enzyme isoforms of human, trypanosome (T. brucei), leishmanial (L. major) a...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2K35SGMUS Patent
TargetGlycylpeptide N-tetradecanoyltransferase(Candida albicans (Yeast))
Second Military Medical University

Curated by ChEMBL
LigandPNGBDBM50207640(CHEMBL254011 | N-(2-(cyclobutanecarboxamido)benzo[...)copy SMILEScopy InChI
Affinity DataIC50: 2.30nMAssay Description:Inhibition of Candida albicans N-myristoyltransferseMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2RV0ND9PubMed
TargetGlycylpeptide N-tetradecanoyltransferase(Candida albicans (Yeast))
Second Military Medical University

Curated by ChEMBL
LigandPNGBDBM50207640(CHEMBL254011 | N-(2-(cyclobutanecarboxamido)benzo[...)copy SMILEScopy InChI
Affinity DataIC50: 2.30nMAssay Description:Inhibition of Candida albicans N-myristoyltransferseMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2RV0ND9PubMed
TargetGlycylpeptide N-tetradecanoyltransferase(Candida albicans (Yeast))
Second Military Medical University

Curated by ChEMBL
LigandPNGBDBM50207612(CHEMBL400892 | N-(2-(cyclopropanecarboxamido)benzo...)copy SMILEScopy InChI
Affinity DataIC50: 2.40nMAssay Description:Inhibition of Candida albicans N-myristoyltransferseMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2RV0ND9PubMed
TargetGlycylpeptide N-tetradecanoyltransferase(Candida albicans (Yeast))
Second Military Medical University

Curated by ChEMBL
LigandPNGBDBM50207612(CHEMBL400892 | N-(2-(cyclopropanecarboxamido)benzo...)copy SMILEScopy InChI
Affinity DataIC50: 2.40nMAssay Description:Inhibition of Candida albicans N-myristoyltransferseMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2RV0ND9PubMed
TargetGlycylpeptide N-tetradecanoyltransferase 1(Homo sapiens (Human))
Frontier Medicines

Curated by ChEMBL
LigandPNGBDBM50364113(CHEMBL1230468)copy SMILEScopy InChI
Affinity DataIC50: 3nMAssay Description:Inhibition of human N-myristoyltransferase 1 assessed as transfer of [3H]-myristic acid to a biotinylated substrate peptide (GCGGSKVKPQPPQAK(biotin)-...More data for this Ligand-Target Pair
TargetGlycylpeptide N-tetradecanoyltransferase 1(Homo sapiens (Human))
Frontier Medicines

Curated by ChEMBL
LigandPNGBDBM184902(US9156811, DDD86481)copy SMILEScopy InChI
Affinity DataIC50: 3nMpH: 7.4 T: 2°CAssay Description:Measurement of the ability of compounds to inhibit the NMT-1 and/or NMT-2 enzyme isoforms of human, trypanosome (T. brucei), leishmanial (L. major) a...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2K35SGMUS Patent
TargetGlycylpeptide N-tetradecanoyltransferase 1(Homo sapiens (Human))
Frontier Medicines

Curated by ChEMBL
LigandPNGBDBM50364113(CHEMBL1230468)copy SMILEScopy InChI
Affinity DataIC50: 3nMAssay Description:Inhibition of human N-myristoyltransferase 1 using [3H]myristoyl-CoA and GCGGSKVKPQPPQAK(biotin)-amide as substrate preincubated for 5 mins prior sub...More data for this Ligand-Target Pair
TargetGlycylpeptide N-tetradecanoyltransferase 1(Homo sapiens (Human))
Frontier Medicines

Curated by ChEMBL
LigandPNGBDBM184977(US9156811, DDD88646)copy SMILEScopy InChI
Affinity DataIC50: 3nMpH: 7.4 T: 2°CAssay Description:Measurement of the ability of compounds to inhibit the NMT-1 and/or NMT-2 enzyme isoforms of human, trypanosome (T. brucei), leishmanial (L. major) a...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2K35SGMUS Patent
TargetGlycylpeptide N-tetradecanoyltransferase 1(Homo sapiens (Human))
Frontier Medicines

Curated by ChEMBL
LigandPNGBDBM184848(US9156811, DDD85646)copy SMILEScopy InChI
Affinity DataIC50: 3nMpH: 7.4 T: 2°CAssay Description:Measurement of the ability of compounds to inhibit the NMT-1 and/or NMT-2 enzyme isoforms of human, trypanosome (T. brucei), leishmanial (L. major) a...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2K35SGMUS Patent
TargetGlycylpeptide N-tetradecanoyltransferase 1(Homo sapiens (Human))
Frontier Medicines

Curated by ChEMBL
LigandPNGBDBM184854(US9156811, DDD86206)copy SMILEScopy InChI
Affinity DataIC50: 3nMpH: 7.4 T: 2°CAssay Description:Measurement of the ability of compounds to inhibit the NMT-1 and/or NMT-2 enzyme isoforms of human, trypanosome (T. brucei), leishmanial (L. major) a...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2K35SGMUS Patent
TargetGlycylpeptide N-tetradecanoyltransferase(Candida albicans (Yeast))
Second Military Medical University

Curated by ChEMBL
LigandPNGBDBM50207620(CHEMBL254010 | N-(2-isobutyramidobenzo[d]thiazol-6...)copy SMILEScopy InChI
Affinity DataIC50: 3.30nMAssay Description:Inhibition of Candida albicans N-myristoyltransferseMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2RV0ND9PubMed
TargetGlycylpeptide N-tetradecanoyltransferase(Candida albicans (Yeast))
Second Military Medical University

Curated by ChEMBL
LigandPNGBDBM50207620(CHEMBL254010 | N-(2-isobutyramidobenzo[d]thiazol-6...)copy SMILEScopy InChI
Affinity DataIC50: 3.30nMAssay Description:Inhibition of Candida albicans N-myristoyltransferseMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2RV0ND9PubMed
TargetGlycylpeptide N-tetradecanoyltransferase 1(Homo sapiens (Human))
Frontier Medicines

Curated by ChEMBL
LigandPNGBDBM50033480(CHEMBL3357697)copy SMILEScopy InChI
Affinity DataIC50: 4nMAssay Description:Inhibition of human N-myristoyltransferase 1 assessed as transfer of [3H]-myristic acid to a biotinylated substrate peptide (GCGGSKVKPQPPQAK(biotin)-...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ZC84G2PubMed
TargetGlycylpeptide N-tetradecanoyltransferase 1(Homo sapiens (Human))
Frontier Medicines

Curated by ChEMBL
LigandPNGBDBM50033485(CHEMBL3357702)copy SMILEScopy InChI
Affinity DataIC50: 4nMAssay Description:Inhibition of human N-myristoyltransferase 1 assessed as transfer of [3H]-myristic acid to a biotinylated substrate peptide (GCGGSKVKPQPPQAK(biotin)-...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ZC84G2PubMed
TargetGlycylpeptide N-tetradecanoyltransferase 1(Homo sapiens (Human))
Frontier Medicines

Curated by ChEMBL
LigandPNGBDBM50033616(CHEMBL3358119)copy SMILEScopy InChI
Affinity DataIC50: 4nMAssay Description:Inhibition of human N-myristoyltransferase 1 assessed as transfer of [3H]-myristic acid to a biotinylated substrate peptide (GCGGSKVKPQPPQAK(biotin)-...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ZC84G2PubMed
TargetGlycylpeptide N-tetradecanoyltransferase 1(Homo sapiens (Human))
Frontier Medicines

Curated by ChEMBL
LigandPNGBDBM50364113(CHEMBL1230468)copy SMILEScopy InChI
Affinity DataIC50: 4nMAssay Description:Inhibition of human NMT1 using [3H]-myristoyl-coA/biotinylated CAP5.5 as substrate after 15 mins by scintillation/luminescence counting methodMore data for this Ligand-Target Pair
TargetGlycylpeptide N-tetradecanoyltransferase 1(Homo sapiens (Human))
Frontier Medicines

Curated by ChEMBL
LigandPNGBDBM184978(US9156811, DDD90022)copy SMILEScopy InChI
Affinity DataIC50: 4nMpH: 7.4 T: 2°CAssay Description:Measurement of the ability of compounds to inhibit the NMT-1 and/or NMT-2 enzyme isoforms of human, trypanosome (T. brucei), leishmanial (L. major) a...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2K35SGMUS Patent
TargetGlycylpeptide N-tetradecanoyltransferase 1(Homo sapiens (Human))
Frontier Medicines

Curated by ChEMBL
LigandPNGBDBM185101(US9156811, DDD100807)copy SMILEScopy InChI
Affinity DataIC50: 4nMpH: 7.4 T: 2°CAssay Description:Measurement of the ability of compounds to inhibit the NMT-1 and/or NMT-2 enzyme isoforms of human, trypanosome (T. brucei), leishmanial (L. major) a...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2K35SGMUS Patent
TargetGlycylpeptide N-tetradecanoyltransferase 1(Homo sapiens (Human))
Frontier Medicines

Curated by ChEMBL
LigandPNGBDBM50033418(CHEMBL3357685)copy SMILEScopy InChI
Affinity DataIC50: 4nMAssay Description:Inhibition of human N-myristoyltransferase 1 assessed as transfer of [3H]-myristic acid to a biotinylated substrate peptide (GCGGSKVKPQPPQAK(biotin)-...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ZC84G2PubMed
TargetGlycylpeptide N-tetradecanoyltransferase(Candida albicans (Yeast))
Second Military Medical University

Curated by ChEMBL
LigandPNGBDBM50109879(CHEMBL155301 | Non peptidic, 4 | {3-[2-(2,3-Difluo...)copy SMILEScopy InChI
Affinity DataIC50: 4nMAssay Description:Inhibition activity against C. albicans Nmt and human Nmt as assessed by IC50 using myristoyl-CoA (0.5 uM) and peptide substrate GLTISKLFRR-NH2 (0.5 ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BV7F0CPubMed
TargetGlycylpeptide N-tetradecanoyltransferase 1(Homo sapiens (Human))
Frontier Medicines

Curated by ChEMBL
LigandPNGBDBM185092(US9156811, DDD100798)copy SMILEScopy InChI
Affinity DataIC50: 4nMpH: 7.4 T: 2°CAssay Description:Measurement of the ability of compounds to inhibit the NMT-1 and/or NMT-2 enzyme isoforms of human, trypanosome (T. brucei), leishmanial (L. major) a...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2K35SGMUS Patent
TargetGlycylpeptide N-tetradecanoyltransferase 1(Homo sapiens (Human))
Frontier Medicines

Curated by ChEMBL
LigandPNGBDBM184988(US9156811, DDD90107)copy SMILEScopy InChI
Affinity DataIC50: 5nMpH: 7.4 T: 2°CAssay Description:Measurement of the ability of compounds to inhibit the NMT-1 and/or NMT-2 enzyme isoforms of human, trypanosome (T. brucei), leishmanial (L. major) a...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2K35SGMUS Patent
TargetGlycylpeptide N-tetradecanoyltransferase 1(Homo sapiens (Human))
Frontier Medicines

Curated by ChEMBL
LigandPNGBDBM184943(US9156811, DDD88193)copy SMILEScopy InChI
Affinity DataIC50: 5nMpH: 7.4 T: 2°CAssay Description:Measurement of the ability of compounds to inhibit the NMT-1 and/or NMT-2 enzyme isoforms of human, trypanosome (T. brucei), leishmanial (L. major) a...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2K35SGMUS Patent
TargetGlycylpeptide N-tetradecanoyltransferase 1(Homo sapiens (Human))
Frontier Medicines

Curated by ChEMBL
LigandPNGBDBM50033618(CHEMBL3358121)copy SMILEScopy InChI
Affinity DataIC50: 5nMAssay Description:Inhibition of human N-myristoyltransferase 1 assessed as transfer of [3H]-myristic acid to a biotinylated substrate peptide (GCGGSKVKPQPPQAK(biotin)-...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ZC84G2PubMed
TargetGlycylpeptide N-tetradecanoyltransferase 1(Homo sapiens (Human))
Frontier Medicines

Curated by ChEMBL
LigandPNGBDBM50033482(CHEMBL3357699)copy SMILEScopy InChI
Affinity DataIC50: 5nMAssay Description:Inhibition of human N-myristoyltransferase 1 assessed as transfer of [3H]-myristic acid to a biotinylated substrate peptide (GCGGSKVKPQPPQAK(biotin)-...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ZC84G2PubMed
TargetGlycylpeptide N-tetradecanoyltransferase 1(Homo sapiens (Human))
Frontier Medicines

Curated by ChEMBL
LigandPNGBDBM50033617(CHEMBL3358120)copy SMILEScopy InChI
Affinity DataIC50: 5nMAssay Description:Inhibition of human NMT1 using [3H]-myristoyl-coA/biotinylated CAP5.5 as substrate after 15 mins by scintillation/luminescence counting methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25141NZPubMed
TargetGlycylpeptide N-tetradecanoyltransferase 1(Homo sapiens (Human))
Frontier Medicines

Curated by ChEMBL
LigandPNGBDBM184992(US9156811, DDD90118)copy SMILEScopy InChI
Affinity DataIC50: 5nMpH: 7.4 T: 2°CAssay Description:Measurement of the ability of compounds to inhibit the NMT-1 and/or NMT-2 enzyme isoforms of human, trypanosome (T. brucei), leishmanial (L. major) a...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2K35SGMUS Patent
TargetGlycylpeptide N-tetradecanoyltransferase 1(Homo sapiens (Human))
Frontier Medicines

Curated by ChEMBL
LigandPNGBDBM185083(US9156811, DDD100169)copy SMILEScopy InChI
Affinity DataIC50: 5nMpH: 7.4 T: 2°CAssay Description:Measurement of the ability of compounds to inhibit the NMT-1 and/or NMT-2 enzyme isoforms of human, trypanosome (T. brucei), leishmanial (L. major) a...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2K35SGMUS Patent
TargetGlycylpeptide N-tetradecanoyltransferase 1(Homo sapiens (Human))
Frontier Medicines

Curated by ChEMBL
LigandPNGBDBM50033617(CHEMBL3358120)copy SMILEScopy InChI
Affinity DataIC50: 5nMAssay Description:Inhibition of human N-myristoyltransferase 1 assessed as transfer of [3H]-myristic acid to a biotinylated substrate peptide (GCGGSKVKPQPPQAK(biotin)-...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ZC84G2PubMed
TargetGlycylpeptide N-tetradecanoyltransferase(Candida albicans (Yeast))
Second Military Medical University

Curated by ChEMBL
LigandPNGBDBM50109882(3-(3-methyl-2-((2,3,4-trifluorophenoxy)methyl)benz...)copy SMILEScopy InChI
Affinity DataIC50: 5.70nMAssay Description:Inhibition of Candida albicans N-myristoyltransferseMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2RV0ND9PubMed
TargetGlycylpeptide N-tetradecanoyltransferase(Candida albicans (Yeast))
Second Military Medical University

Curated by ChEMBL
LigandPNGBDBM50109882(3-(3-methyl-2-((2,3,4-trifluorophenoxy)methyl)benz...)copy SMILEScopy InChI
Affinity DataIC50: 5.70nMAssay Description:Inhibition of Candida albicans N-myristoyltransferseMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2RV0ND9PubMed
TargetGlycylpeptide N-tetradecanoyltransferase(Candida albicans (Yeast))
Second Military Medical University

Curated by ChEMBL
LigandPNGBDBM50109882(3-(3-methyl-2-((2,3,4-trifluorophenoxy)methyl)benz...)copy SMILEScopy InChI
Affinity DataIC50: 5.70nMAssay Description:Inhibition of Candida albicans ATCC 90028 NMT using GLTISKLFRR-NH2 as substrate assessed as reduction in [3H]-myristoylated peptide reaction product ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26112X4PubMed
TargetGlycylpeptide N-tetradecanoyltransferase 1(Homo sapiens (Human))
Frontier Medicines

Curated by ChEMBL
LigandPNGBDBM185061(US9156811, DDD100144)copy SMILEScopy InChI
Affinity DataIC50: 6nMpH: 7.4 T: 2°CAssay Description:Measurement of the ability of compounds to inhibit the NMT-1 and/or NMT-2 enzyme isoforms of human, trypanosome (T. brucei), leishmanial (L. major) a...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2K35SGMUS Patent
TargetGlycylpeptide N-tetradecanoyltransferase 1(Homo sapiens (Human))
Frontier Medicines

Curated by ChEMBL
LigandPNGBDBM184937(US9156811, DDD88186)copy SMILEScopy InChI
Affinity DataIC50: 6nMpH: 7.4 T: 2°CAssay Description:Measurement of the ability of compounds to inhibit the NMT-1 and/or NMT-2 enzyme isoforms of human, trypanosome (T. brucei), leishmanial (L. major) a...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2K35SGMUS Patent
TargetGlycylpeptide N-tetradecanoyltransferase 1(Homo sapiens (Human))
Frontier Medicines

Curated by ChEMBL
LigandPNGBDBM185108(US9156811, DDD100869)copy SMILEScopy InChI
Affinity DataIC50: 6nMpH: 7.4 T: 2°CAssay Description:Measurement of the ability of compounds to inhibit the NMT-1 and/or NMT-2 enzyme isoforms of human, trypanosome (T. brucei), leishmanial (L. major) a...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2K35SGMUS Patent
TargetGlycylpeptide N-tetradecanoyltransferase 1(Homo sapiens (Human))
Frontier Medicines

Curated by ChEMBL
LigandPNGBDBM50364135(CHEMBL1951295)copy SMILEScopy InChI
Affinity DataIC50: 7nMAssay Description:Inhibition of human N-myristoyltransferase 1 using [3H]myristoyl-CoA and GCGGSKVKPQPPQAK(biotin)-amide as substrate preincubated for 5 mins prior sub...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25Q4WK9PubMed
TargetGlycylpeptide N-tetradecanoyltransferase 1(Homo sapiens (Human))
Frontier Medicines

Curated by ChEMBL
LigandPNGBDBM184965(US9156811, DDD88558)copy SMILEScopy InChI
Affinity DataIC50: 7nMpH: 7.4 T: 2°CAssay Description:Measurement of the ability of compounds to inhibit the NMT-1 and/or NMT-2 enzyme isoforms of human, trypanosome (T. brucei), leishmanial (L. major) a...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2K35SGMUS Patent
TargetGlycylpeptide N-tetradecanoyltransferase 1(Homo sapiens (Human))
Frontier Medicines

Curated by ChEMBL
LigandPNGBDBM184860(US9156811, DDD86213)copy SMILEScopy InChI
Affinity DataIC50: 7nMpH: 7.4 T: 2°CAssay Description:Measurement of the ability of compounds to inhibit the NMT-1 and/or NMT-2 enzyme isoforms of human, trypanosome (T. brucei), leishmanial (L. major) a...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2K35SGMUS Patent
TargetGlycylpeptide N-tetradecanoyltransferase 1(Homo sapiens (Human))
Frontier Medicines

Curated by ChEMBL
LigandPNGBDBM185078(US9156811, DDD100164)copy SMILEScopy InChI
Affinity DataIC50: 7nMpH: 7.4 T: 2°CAssay Description:Measurement of the ability of compounds to inhibit the NMT-1 and/or NMT-2 enzyme isoforms of human, trypanosome (T. brucei), leishmanial (L. major) a...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2K35SGMUS Patent
TargetGlycylpeptide N-tetradecanoyltransferase 1(Homo sapiens (Human))
Frontier Medicines

Curated by ChEMBL
LigandPNGBDBM184920(US9156811, DDD87767)copy SMILEScopy InChI
Affinity DataIC50: 8nMpH: 7.4 T: 2°CAssay Description:Measurement of the ability of compounds to inhibit the NMT-1 and/or NMT-2 enzyme isoforms of human, trypanosome (T. brucei), leishmanial (L. major) a...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2K35SGMUS Patent
TargetGlycylpeptide N-tetradecanoyltransferase 1(Homo sapiens (Human))
Frontier Medicines

Curated by ChEMBL
LigandPNGBDBM50033619(CHEMBL3358122)copy SMILEScopy InChI
Affinity DataIC50: 8nMAssay Description:Inhibition of human N-myristoyltransferase 1 assessed as transfer of [3H]-myristic acid to a biotinylated substrate peptide (GCGGSKVKPQPPQAK(biotin)-...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ZC84G2PubMed
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